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Design, Synthesis, and Structure-Activity Relationship Study of 2-Oxo-3,4-dihydropyrimido[4,5-d]pyrimidines as New Colony Stimulating Factor 1 Receptor (CSF1R) Kinase Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 页码: 2353-2371
作者:  Xun, Qiuju[1];  Zhang, Zhang[2];  Luo, Jinfeng[3];  Tong, Linjiang[4];  Huang, Minhao[5]
收藏  |  浏览/下载:25/0  |  提交时间:2019/04/22
Design, Synthesis, and Structure-Activity Relationship Study of 2-Oxo-3,4-dihydropyrimido[4,5-d]pyrimidines as New Colony Stimulating Factor 1 Receptor (CSF1R) Kinase Inhibitors 期刊论文
2018, 卷号: 61, 期号: 6, 页码: 2353
作者:  Xun, Qiuju[1,2];  Zhang, Zhang[3];  Luo, Jinfeng[1];  Tong, Linjiang[6];  Huang, Minhao[1,2]
收藏  |  浏览/下载:16/0  |  提交时间:2019/12/10
Design, Synthesis, and Biological Evaluation of 3-(Imidazo[1,2-a]pyrazin-3-ylethynyl)-4-isopropyl-N-(3-((4-methylpiperazin-1-yl)methyl)-5-(trifluoromethyl)phenyl)benzamide as a Dual Inhibitor of Discoidin Domain Receptors 1 and 2 期刊论文
2018, 卷号: 61, 期号: 17, 页码: 7977
作者:  Wang, Zhen[1,2];  Zhang, Yali[3];  Pinkas, Daniel M.[7];  Fox, Alice E.[7];  Luo, Jinfeng[2]
收藏  |  浏览/下载:27/0  |  提交时间:2019/12/17
Discovery of JND3229 as a New EGFR(C797S) Mutant Inhibitor with In Vivo Monodrug Efficacy 期刊论文
2018, 卷号: 9, 期号: 11, 页码: 1123
作者:  Lu, Xiaoyun[1];  Zhang, Tao[2,6,7];  Zhu, Su-Jie[3,4];  Xun, Qiuju[5];  Tong, Lingjiang[2]
收藏  |  浏览/下载:24/0  |  提交时间:2019/12/23
Tetrahydroisoquinoline-7-carboxamide Derivatives as New Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors 期刊论文
2017, 卷号: 8, 期号: 3, 页码: 327
作者:  Wang, Zhen[1,2];  Zhang, Yali[3];  Bartual, Sergio G.[5];  Luo, Jinfeng[2];  Xu, Tingting[4]
收藏  |  浏览/下载:22/0  |  提交时间:2019/12/06


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