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Design, Synthesis, and Structure-Activity Relationship Study of 2-Oxo-3,4-dihydropyrimido[4,5-d]pyrimidines as New Colony Stimulating Factor 1 Receptor (CSF1R) Kinase Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 页码: 2353-2371
作者:  Xun, Qiuju[1];  Zhang, Zhang[2];  Luo, Jinfeng[3];  Tong, Linjiang[4];  Huang, Minhao[5]
收藏  |  浏览/下载:25/0  |  提交时间:2019/04/22
Design, Synthesis, and Structure-Activity Relationship Study of 2-Oxo-3,4-dihydropyrimido[4,5-d]pyrimidines as New Colony Stimulating Factor 1 Receptor (CSF1R) Kinase Inhibitors 期刊论文
2018, 卷号: 61, 期号: 6, 页码: 2353
作者:  Xun, Qiuju[1,2];  Zhang, Zhang[3];  Luo, Jinfeng[1];  Tong, Linjiang[6];  Huang, Minhao[1,2]
收藏  |  浏览/下载:16/0  |  提交时间:2019/12/10
A structure-guided optimization of pyrido[2,3-d]pyrimidin-7-ones as selective inhibitors of EGFR(L858R/T790M) mutant with improved pharmacokinetic properties 期刊论文
2017, 卷号: 126, 期号: [db:dc_citation_issue], 页码: 1107
作者:  Yu, Lei[1,2];  Huang, Minhao[1,2];  Xu, Tianfeng[1,2];  Tong, Linjiang[4];  Yan, Xiao-e[5,6]
收藏  |  浏览/下载:5/0  |  提交时间:2019/12/03
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M) 期刊论文
2015, 卷号: 25, 期号: [db:dc_citation_issue], 页码: 4277
作者:  Chan, Shingpan[1,2];  Han, Kun[3];  Qu, Rong[2,3];  Tong, Linjiang[3];  Li, Yingjun[1,2]
收藏  |  浏览/下载:23/0  |  提交时间:2019/12/03


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