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Discovery of SARS-CoV-2-E channel inhibitors as antiviral candidates 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 7
作者:  Wang, Yi;  Fang, Sui;  Wu, Yan;  Cheng, Xi;  Zhang, Lei-ke
收藏  |  浏览/下载:101/0  |  提交时间:2021/08/17
Discovery of 2-(5-(quinolin-6-yl)-1,3,4-oxadiazol-2-yl)acetamide derivatives as novel PI3K alpha inhibitors via docking-based virtual screening 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 29, 页码: 9
作者:  Gu, Dongyan;  Cheng, Gang;  Zhang, Mengmeng;  Zhou, Yu-Bo;  Li, Jia
收藏  |  浏览/下载:15/0  |  提交时间:2021/05/24
In Silico Screening-Based Discovery of Novel Inhibitors of Human Cyclic GMP-AMP Synthase: A Cross-Validation Study of Molecular Docking and Experimental Testing 期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2020, 卷号: 60, 期号: 6, 页码: 3265-3276
作者:  Zhao, Wenfeng;  Xiong, Muya;  Yuan, Xiaojing;  Li, Minjun;  Sun, Hongbin
收藏  |  浏览/下载:17/0  |  提交时间:2020/12/24
Design, Synthesis, and Biological Evaluation of 8-Mercapto-3,7-Dihydro-1H-Purine-2,6-Diones as Potent Inhibitors of SIRT1, SIRT2, SIRT3, and SIRT5 期刊论文
MOLECULES, 2020, 卷号: 25, 期号: 12, 页码: 18
作者:  Han, Haozhen;  Li, Chunpu;  Li, Man;  Yang, Lisheng;  Zhao, Sen
收藏  |  浏览/下载:35/0  |  提交时间:2020/12/24
Identification of catalytic and non-catalytic activity inhibitors against PRC2-EZH2 complex through multiple high-throughput screening campaigns 期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2020, 页码: 27
作者:  Zhou, Yan;  Du, Dao-Hai;  Wang, Jia;  Cai, Xiao-Qing;  Deng, Alicia X.
收藏  |  浏览/下载:102/0  |  提交时间:2020/07/01
High-throughput screening campaign identifies a small molecule agonist of the relaxin family peptide receptor 4 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 9
作者:  Lin, Guang-yao;  Lin, Lin;  Cai, Xiao-qing;  Dai, An-tao;  Zhu, Yue
收藏  |  浏览/下载:27/0  |  提交时间:2020/07/01
Discovery and characterization of natural products as novel indoleamine 2,3-dioxygenase 1 inhibitors through high-throughput screening 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 卷号: 41, 期号: 3, 页码: 423-431
作者:  Guo, Wei;  Yao, Sheng;  Sun, Pu;  Yang, Tian-biao;  Tang, Chun-ping
收藏  |  浏览/下载:79/0  |  提交时间:2020/07/01
discoveryandcharacterizationofnaturalproductsasnovelindoleamine23dioxygenase1inhibitorsthroughhighthroughputscreening 期刊论文
actapharmacologicasinica, 2020, 卷号: 41, 期号: 3, 页码: 423
作者:  Guo Wei;  Yao Sheng;  Sun Pu;  Yang Tianbiao;  Tang Chunping
收藏  |  浏览/下载:81/0  |  提交时间:2020/07/01
Discovery of New and Potent InhA Inhibitors as Antituberculosis Agents: Structure-Based Virtual Screening Validated by Biological Assays and X-ray Crystallography 期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2020, 卷号: 60, 期号: 1, 页码: 226-234
作者:  Kamsri, Pharit;  Hanwarinroj, Chayanin;  Phusi, Naruedon;  Pornprom, Thimpika;  Chayajarus, Kampanart
收藏  |  浏览/下载:23/0  |  提交时间:2020/07/01
The identification of novel small-molecule inhibitors targeting WDR5-MLL1 interaction through fluorescence polarization based high-throughput screening 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 4, 页码: 638-645
作者:  Ye, Xiaoqing;  Zhang, Rukang;  Lian, Fulin;  Zhang, Weiyao;  Lu, Wenchao
收藏  |  浏览/下载:3/0  |  提交时间:2020/07/01


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