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Repressing MYC by targeting BET synergizes with selective inhibition of PI3K alpha against B cell lymphoma 期刊论文
CANCER LETTERS, 2022, 卷号: 524, 页码: 206-218
作者:  Chen, Zi-qi;  Cao, Zhe-rui;  Wang, Yi;  Zhang, Xi;  Xu, Lan
收藏  |  浏览/下载:53/0  |  提交时间:2021/12/16
CYH33  MYC  P300  BET  B cell lymphoma  PI3K  
Rhodomeroterpene alleviates macrophage infiltration and the inflammatory response in renal tissue to improve acute kidney injury 期刊论文
FASEB JOURNAL, 2021, 卷号: 35, 期号: 11, 页码: 17
作者:  Wu, Yong-Mei;  Shi, Qing;  Zhu, Peng-Fei;  Ma, Hai-Jian;  Cui, Shi-Chao
收藏  |  浏览/下载:54/0  |  提交时间:2021/12/16
Anti-DLBCL efficacy of DCZ0825 in vitro and in vivo: involvement of the PI3K-AKT-mTOR/JNK pathway 期刊论文
ACTA BIOCHIMICA ET BIOPHYSICA SINICA, 2021, 卷号: 53, 期号: 5, 页码: 575-583
作者:  Hu, Ke;  Li, Bo;  Ma, Ruye;  Yi, Hongfei;  Xu, Zhijian
收藏  |  浏览/下载:68/0  |  提交时间:2021/06/11
lncRNA H19 binds VGF and promotes pNEN progression via PI3K/AKT/CREB signaling (vol 26, pg 643, 2019) 期刊论文
ENDOCRINE-RELATED CANCER, 2021, 卷号: 28, 期号: 4, 页码: X1-X2
作者:  Ji, Meng;  Yao, Yanli;  Liu, Anan;  Shi, Ligang;  Chen, Danlei
收藏  |  浏览/下载:16/0  |  提交时间:2021/08/17
PI3K alpha inhibitor impairs AKT phosphorylation and synergizes with novel angiogenesis inhibitor AL3810 in human hepatocellular carcinoma 期刊论文
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2021, 卷号: 6, 期号: 1, 页码: 3
作者:  Xie, Qin;  Chi, Shuaishuai;  Fang, Yanfen;  Sun, Yiming;  Meng, Linghua
收藏  |  浏览/下载:18/0  |  提交时间:2021/05/24
SAF-248, a novel PI3K delta-selective inhibitor, potently suppresses the growth of diffuse large B-cell lymphoma 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 11
作者:  Zhang, Xi;  Duan, Yu-ting;  Wang, Yi;  Zhao, Xing-dong;  Sun, Yi-ming
收藏  |  浏览/下载:37/0  |  提交时间:2021/05/24
Identification of methyl (5-(6-((4-(methylsulfonyl)piperazin-1-yl)methyl)-4-morpholinopyrrolo[2,1-f][1,2,4]triazin-2-yl)-4-(trifluoromethyl)pyridin-2-yl)carbamate (CYH33) as an orally bioavailable, highly potent, PI3K alpha inhibitor for the treatment of advanced solid tumors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 209, 页码: 10
作者:  Xiang, Hao-Yue;  Wang, Xiang;  Chen, Yan-Hong;  Zhang, Xi;  Tan, Cun
收藏  |  浏览/下载:33/0  |  提交时间:2021/05/24
DCZ3301, an aryl-guanidino agent, inhibits ocular neovascularization via PI3K/AKT and ERK1/2 signaling pathways 期刊论文
EXPERIMENTAL EYE RESEARCH, 2020, 卷号: 201, 页码: 8
作者:  Xu, Kai;  Li, Bo;  Zhang, Shujie;  Hu, Fangyuan;  Xu, Zhijian
收藏  |  浏览/下载:47/0  |  提交时间:2021/05/24
Comprehensive analysis of transcriptomics and metabolomics to understand triptolide-induced liver injury in mice 期刊论文
TOXICOLOGY LETTERS, 2020, 卷号: 333, 页码: 290-302
作者:  Zhao, Jie;  Xie, Cen;  Wang, Kanglong;  Takahashi, Shogo;  Krausz, Kristopher W.
收藏  |  浏览/下载:49/0  |  提交时间:2020/12/21
Emerging roles of class I PI3K inhibitors in modulating tumor microenvironment and immunity 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 8
作者:  Sun, Pu;  Meng, Ling-hua
收藏  |  浏览/下载:39/0  |  提交时间:2020/12/21


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