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PI3K alpha inhibitor impairs AKT phosphorylation and synergizes with novel angiogenesis inhibitor AL3810 in human hepatocellular carcinoma 期刊论文
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2021, 卷号: 6, 期号: 1, 页码: 3
作者:  Xie, Qin;  Chi, Shuaishuai;  Fang, Yanfen;  Sun, Yiming;  Meng, Linghua
收藏  |  浏览/下载:18/0  |  提交时间:2021/05/24
N-Cyclic sulfamoylaminoethyl substituted 1,2,5-oxadiazol-3-amines as new indoleamine 2, 3-dioxygenase 1 (IDO1) inhibitors. 期刊论文
CANCER IMMUNOLOGY RESEARCH, 2020, 卷号: 8, 期号: 3, 页码: 51-51
作者:  Chen, Shulun;  Guo, Wei;  Sun, Pu;  Meng, Linghua;  Zhang, Ao
收藏  |  浏览/下载:16/0  |  提交时间:2020/07/01
discoveryandcharacterizationofnaturalproductsasnovelindoleamine23dioxygenase1inhibitorsthroughhighthroughputscreening 期刊论文
actapharmacologicasinica, 2020, 卷号: 41, 期号: 3, 页码: 423
作者:  Guo Wei;  Yao Sheng;  Sun Pu;  Yang Tianbiao;  Tang Chunping
收藏  |  浏览/下载:81/0  |  提交时间:2020/07/01
crisprcas9apowerfultooltowardsprecisionmedicineincancertreatment 期刊论文
actapharmacologicasinica, 2020, 卷号: 41, 期号: 5, 页码: 583
作者:  Xing Hui;  Meng Linghua
收藏  |  浏览/下载:25/0  |  提交时间:2020/07/01
Design, synthesis, and biological evaluation of thieno[3,2-d]pyrimidine derivatives as potential simplified phosphatidylinositol 3-kinase alpha inhibitors 期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2019, 卷号: 94, 期号: 6, 页码: 2013-2022
作者:  Yang, Xiuyan;  Deng, Meng;  Zhang, Xi;  Wang, Yi;  Song, Kun
收藏  |  浏览/下载:75/0  |  提交时间:2020/07/01
HRAS(G12s) mutant mediates resistance to a PI3K alpha inhibitor CYH33 in esophageal squamous cell carcinomas 期刊论文
MOLECULAR CANCER THERAPEUTICS, 2019, 卷号: 18, 期号: 12, 页码: 2
作者:  Wang, Yuxiang;  Zhang, Xu;  Ma, Qingyang;  Zhang, Xi;  Yang, Chunhao
收藏  |  浏览/下载:23/0  |  提交时间:2020/07/01
Design, synthesis and antitumor study of a series of N-Cyclic sulfamoylaminoethyl substituted 1,2,5-oxadiazol-3-amines as new indoleamine 2, 3-dioxygenase 1 (IDO1) inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 179, 页码: 38-55
作者:  Chen, Shulun;  Guo, Wei;  Liu, Xiaohua;  Sun, Pu;  Wang, Yi
收藏  |  浏览/下载:11/0  |  提交时间:2020/07/01
Discovery of Indoleamine 2,3-Dioxygenase 1 (IDO-1) Inhibitors Based on Ortho-Naphthaquinone-Containing Natural Product 期刊论文
MOLECULES, 2019, 卷号: 24, 期号: 6, 页码: 11
作者:  Zhao, Hongchuan;  Sun, Pu;  Guo, Wei;  Wang, Yi;  Zhang, Ao
收藏  |  浏览/下载:8/0  |  提交时间:2020/07/01
Fe3+-sensing by 3,3 ',5,5 '- tetramethylbenzidine-functionalized upconversion nanoparticles 期刊论文
NANOTECHNOLOGY, 2019, 卷号: 30, 页码: 135502
作者:  Meng, Zhipeng;  Wu, Suli;  Zhong, Linghua;  Sun, Xiaoqian;  Li, Lu
收藏  |  浏览/下载:9/0  |  提交时间:2019/12/02
Unbiased screening reveals that blocking exportin 1 overcomes resistance to PI3Kα inhibition in breast cancer 期刊论文
signaltransductionandtargetedtherapy, 2019, 卷号: 4, 期号: 4, 页码: 295
作者:  Liu Xueling;  Wang Bobo;  Wang Yi;  Wang Yuxiang;  Yang Chunhao
收藏  |  浏览/下载:15/0  |  提交时间:2020/07/01


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