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科研机构
上海药物研究所 [108]
内容类型
期刊论文 [104]
会议论文 [3]
学位论文 [1]
发表日期
2021 [8]
2020 [11]
2019 [4]
2018 [8]
2017 [6]
2016 [6]
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Chemistry [1]
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Define Mesenchymal Stem Cell from Its Fate: Biodisposition of Human Mesenchymal Stem Cells in Normal and Concanavalin A-Induced Liver Injury Mice
期刊论文
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2021, 卷号: 379, 期号: 2, 页码: 125-133
作者:
Han, Li
;
Ma, Chenhui
;
Peng, Huige
;
Wu, Zhitao
;
Xu, Huiming
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2022/01/04
Enhancing the Potential of Miniature-Scale DNA-Compatible Radical Reactions via an Electron Donor-Acceptor Complex and a Reversible Adsorption to Solid Support Strategy
期刊论文
ORGANIC LETTERS, 2021, 卷号: 23, 期号: 19, 页码: 7381-7385
作者:
Lin, Bizhen
;
Lu, Weiwei
;
Chen, Zhen-yu
;
Zhang, Yue
;
Duan, Yin-zhe
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2021/12/01
Effects of Food on the Pharmacokinetic Properties and Mass Balance of Henagliflozin in Healthy Male Volunteers
期刊论文
CLINICAL THERAPEUTICS, 2021, 卷号: 43, 期号: 9, 页码: E264-E273
作者:
Chen, Zhen-dong
;
Chen, Qian
;
Zhu, Yun-ting
;
Zhang, Yi-fan
;
Zhan, Yan
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2022/01/04
henagliflozin
food effects
mass balance
pharmacokinetics
SGLT-2 inhibitor
DNA-encoded C-H functionality via photoredox-mediated hydrogen atom transformation catalysis
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 42, 页码: 4
作者:
Shan, Jinming
;
Ling, Xing
;
Liu, JiaXiang
;
Wang, Xuan
;
Lu, Xiaojie
收藏
  |  
浏览/下载:86/0
  |  
提交时间:2021/08/17
Photoredox
Hydrogen atom transfer
N-Boc saturated heterocycle
DNA Encoded Library (DEL)
Molecular Dynamics Simulations Based on 1-Phenyl-4-Benzoyl-1-Hydro-Triazole ERR alpha Inverse Agonists
期刊论文
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2021, 卷号: 22, 期号: 7, 页码: 14
作者:
Gao, Zhipei
;
Du, Yongli
;
Sheng, Xiehuang
;
Shen, Jingkang
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2021/05/24
ERRα
inverse agonists
1-phenyl-4-benzoyl-1-hydro-triazole
MD simulations
Neonatal cortical astrocytes possess intrinsic potential in neuronal conversion in defined media
期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 12
作者:
Zeng, Peng
;
Hua, Qiu-hong
;
Gong, Jun-yuan
;
Shi, Chang-jie
;
Pi, Xiao-ping
收藏
  |  
浏览/下载:64/0
  |  
提交时间:2021/05/24
cortical astrocytes
neonatal
neuronal conversion
insulin
heterogeneity
Increasing the Sampling Efficiency of Protein Conformational Change by Combining a Modified Replica Exchange Molecular Dynamics and Normal Mode Analysis
期刊论文
JOURNAL OF CHEMICAL THEORY AND COMPUTATION, 2021, 卷号: 17, 期号: 1, 页码: 13-28
作者:
Peng, Cheng
;
Wang, Jinan
;
Shi, Yulong
;
Xu, Zhijian
;
Zhu, Weiliang
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2021/05/24
A Phase I Study to Evaluate the Safety, Tolerability, and Pharmacokinetics of TPN171H, a Novel Phosphodiesterase Type 5 Inhibitor, in Healthy Subjects
期刊论文
DRUG DESIGN DEVELOPMENT AND THERAPY, 2021, 卷号: 15, 页码: 2947-2959
作者:
Qian, Hongjie
;
Chen, Qian
;
Lang, Liyu
;
Zou, Yang
;
Pu, Huahua
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2021/08/17
TPN171H
PDE5 inhibitor
safety
pharmacokinetics
food effect
healthy subjects
Targeted Drugs for Treatment of Pulmonary Arterial Hypertension: Past, Present, and Future Perspectives
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 24, 页码: 15153-15186
作者:
Zheng, Wei
;
Wang, Zhen
;
Jiang, Xiangrui
;
Zhao, Qingjie
;
Shen, Jingshan
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2021/05/24
Intrinsic stability study of L-alpha-glycerylphosphorylcholine with HPLC method development and validation
期刊论文
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2020, 卷号: 188, 页码: 6
作者:
Zhao, Hongwei
;
Sun, Ling
;
Chen, Huanhuan
;
Xiang, Lili
;
Chen, Dongying
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2020/12/24
L-alpha-Glycerylphosphorylcholine
Phosphate ester bond
Forced degradation
HPLC
Intrinsic stability
Kinetics study
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