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"One-Pot" Synthesis of Molnupiravir from Cytidine 期刊论文
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2022, 卷号: 26, 期号: 2, 页码: 358-364
作者:  Hu, TW (Hu, Tianwen) [1] , [2];  Xie, YC (Xie, Yuanchao) [3];  Zhu, FQ (Zhu, Fuqiang) [4];  Gong, XD (Gong, Xudong) [4];  Liu, Y (Liu, Yin) [2] , [3]
收藏  |  浏览/下载:122/0  |  提交时间:2022/03/23
Design, synthesis, in vitro evaluation of a new pyrrolo[1,2-a]thiazolo[5,4-d]pyrimidinone derivatives as cholinesterase inhibitors against Alzheimer's disease 期刊论文
JOURNAL OF HETEROCYCLIC CHEMISTRY, 2022, 卷号: 59, 期号: 6, 页码: 1086-1101
作者:  Zeng, Y (Zeng, Yan) [1] , [2];  Nie, LF (Nie, Lifei) [1];  Liu, L (Liu, Liu) [1];  Niu, C (Niu, Chao) [1] , [2];  Li, Y (Li, Yi) [1] , [2]
收藏  |  浏览/下载:18/0  |  提交时间:2022/06/21
A novel synthesis of tetrahydrocortisone 3-glucuronide 期刊论文
JOURNAL OF CARBOHYDRATE CHEMISTRY, 2022, 卷号: 41, 期号: 1, 页码: 18-27
作者:  Zhang, Y (Zhang, Yan) [1] , [2] , [3];  Zhang, SQ (Zhang, Suqing) [4];  Li, R (Li, Rui) [5];  Shen, JS (Shen, Jingshan) [3] , [4];  Jiang, XR (Jiang, Xiangrui) [3] , [4]
收藏  |  浏览/下载:21/0  |  提交时间:2022/04/07
Synthesis and antiviral activity of 2 '-deoxy-6 '-substituted carbocyclic nucleosides 期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2021, 页码: 12
作者:  Xue, Haitao;  Guo, Shuang;  Hu, Tianwen;  Wei, Daibao;  Xie, Yuanchao
收藏  |  浏览/下载:37/0  |  提交时间:2022/01/18
Scalable Process for Making 5,7-Dichlorotetrahydroisoquinoline-6-carboxylic Acid Using Methylene as the Protecting Group 期刊论文
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2021, 卷号: 25, 期号: 11, 页码: 2447-2452
作者:  Xu, Wanbin;  Gong, Xudong;  Odilov, Abdullajon;  Hu, Tianwen;  Jiang, Xiangrui
收藏  |  浏览/下载:49/0  |  提交时间:2022/01/18
Facile and Cost-Effective Route for the Synthesis of Simmerafil 期刊论文
ORGANIC PROCESS RESEARCH & DEVELOPMENT, 2021, 卷号: 25, 期号: 11, 页码: 2432-2437
作者:  Odilov, Abdullajon;  Liu, Yin;  Hu, Tianwen;  Jiang, Xiangrui;  Suo, Jin
收藏  |  浏览/下载:20/0  |  提交时间:2022/01/18
Design and development of an oral remdesivir derivative VV116 against SARS-CoV-2 期刊论文
CELL RESEARCH, 2021, 页码: 3
作者:  Xie, Yuanchao;  Yin, Wanchao;  Zhang, Yumin;  Shang, Weijuan;  Wang, Zhen
收藏  |  浏览/下载:105/0  |  提交时间:2021/11/04
TPN672: A Novel Serotonin-Dopamine Receptor Modulator for the Treatment of Schizophrenia 期刊论文
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2021, 卷号: 378, 期号: 1, 页码: 20-30
作者:  Wang, Yu;  He, Yang;  Yang, Feipu;  Abame, Melkamu Alemu;  Wu, Chunhui
收藏  |  浏览/下载:37/0  |  提交时间:2021/11/04
Identification of pyrogallol as a warhead in design of covalent inhibitors for the SARS-CoV-2 3CL protease 期刊论文
NATURE COMMUNICATIONS, 2021, 卷号: 12, 期号: 1, 页码: 12
作者:  Su, Haixia;  Yao, Sheng;  Zhao, Wenfeng;  Zhang, Yumin;  Liu, Jia
收藏  |  浏览/下载:27/0  |  提交时间:2021/08/17
SARS-CoV-2 envelope protein causes acute respiratory distress syndrome (ARDS)-like pathological damages and constitutes an antiviral target 期刊论文
CELL RESEARCH, 2021, 页码: 14
作者:  Xia, Bingqing;  Shen, Xurui;  He, Yang;  Pan, Xiaoyan;  Liu, Feng-Liang
收藏  |  浏览/下载:76/0  |  提交时间:2021/08/17


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