CORC

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The Novel RET Inhibitor SYHA1815 Inhibits RET-Driven Cancers and Overcomes Gatekeeper Mutations by Inducing G1 Cell-Cycle Arrest through c-Myc Downregulation 期刊论文
MOLECULAR CANCER THERAPEUTICS, 2021, 卷号: 20, 期号: 11, 页码: 2198-2206
作者:  Jiang, Yuchen;  Peng, Xia;  Ji, Yinchun;  Dai, Yang;  Fang, Yanfen
收藏  |  浏览/下载:28/0  |  提交时间:2021/12/16
Discovery of 1,5-Dihydro-4H-imidazol-4-one Derivatives as Potent, Selective Antagonists of CXC Chemokine Receptor 2 期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2021, 卷号: 12, 期号: 5, 页码: 836-845
作者:  Che, Jinxin;  Wang, Zhilong;  Shen, Zheyuan;  Zhuang, Weihao;  Ying, Huazhou
收藏  |  浏览/下载:60/0  |  提交时间:2021/08/17
GPR52 Antagonist Reduces Huntingtin Levels and Ameliorates Huntington's Disease-Related Phenotypes 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 2, 页码: 941-957
作者:  Wang, Congcong;  Zhang, Yu-Fang;  Guo, Shimeng;  Zhao, Quan;  Zeng, Yanping
收藏  |  浏览/下载:21/0  |  提交时间:2021/05/24
Discovery of selective HDAC/BRD4 dual inhibitors as epigenetic probes 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 209, 页码: 20
作者:  Chen, Jingjing;  Li, Yalei;  Zhang, Jie;  Zhang, Minmin;  Wei, Aihuan
收藏  |  浏览/下载:25/0  |  提交时间:2021/05/24
Targeted Proteomics Combined with Affinity Mass Spectrometry Analysis Reveals Antagonist E7 Acts As an Intracellular Covalent Ligand of Orphan Receptor GPR52 期刊论文
ACS CHEMICAL BIOLOGY, 2020, 卷号: 15, 期号: 12, 页码: 3275-3284
作者:  Ma, Mengna;  Guo, Shimeng;  Lin, Xi;  Li, Shanshan;  Wu, Yiran
收藏  |  浏览/下载:16/0  |  提交时间:2021/05/24
Discovery of Phthalazinone Derivatives as Novel Hepatitis B Virus Capsid Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 15, 页码: 8134-8145
作者:  Chen, Wuhong;  Liu, Feifei;  Zhao, Qiliang;  Ma, Xinna;  Lu, Dong
收藏  |  浏览/下载:34/0  |  提交时间:2020/12/24
NaH Promoted One-Pot Tandem Reactions of 3-(1-Alkynyl) Chromones to Form 2-Nitrogen-Substituted Xanthones 期刊论文
ACS OMEGA, 2020, 卷号: 5, 期号: 22, 页码: 13454-13461
作者:  Duan, Wen-Di;  Zhang, Yu-Fang;  Hu, Youhong
收藏  |  浏览/下载:5/0  |  提交时间:2020/12/24
Base-Promoted Cascade Reactions of 3-(1-Alkynyl)chromones with Pyridinium Ylides to Chromeno[2,3-d]azepine Derivatives 期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2019, 卷号: 84, 期号: 7, 页码: 4467-4472
作者:  Zhang, Yu-Fang;  Duan, Wen-Di;  Chen, Jingjing;  Hu, Youhong
收藏  |  浏览/下载:6/0  |  提交时间:2020/07/01
Visualizing Autophagic Flux during Endothelial Injury with a Pathway-Inspired Tandem-Reaction Based Fluorogenic Probe 期刊论文
THERANOSTICS, 2019, 卷号: 9, 期号: 19, 页码: 5672-5680
作者:  Lei, Yu;  Ren, Wenming;  Wang, Cheng-Kun;  Tao, Rong-Rong;  Xiang, Huai-Jiang
收藏  |  浏览/下载:19/0  |  提交时间:2020/07/01
Fluorescent Imaging of beta-Amyloid Using BODIPY Based Near-Infrared Off-On Fluorescent Probe 期刊论文
BIOCONJUGATE CHEMISTRY, 2018, 卷号: 29, 期号: 10, 页码: 3459-3466
作者:  Ren, Wenming;  Zhang, Jingjing;  Peng, Cheng;  Xiang, Huaijiang;  Chen, Jingjing
收藏  |  浏览/下载:34/0  |  提交时间:2019/01/08


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