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浏览/检索结果: 共9条，第1-9条 帮助 限定条件 专题：山东大学    第一署名单位    第一作者单位    通讯作者单位     已选(0)清除 条数/页：5101520253035404550556065707580859095100   排序方式：请选择发表日期升序发表日期降序提交时间升序提交时间降序题名升序题名降序作者升序作者降序 Design, synthesis, and biological evaluation of 2-(5-methyl-1H-pyrazol-1-yl) acetamide derivatives as androgen receptor antagonists 期刊论文 MEDICINAL CHEMISTRY RESEARCH, 2019, 卷号: 28, 期号: 3, 页码: 380-386 作者:  Dong, Junze;  Zhang, Jingya;  Li, Zilu;  Asnake, Solomon;  Zhang, Daoguang 收藏  |  浏览/下载：15/0  |  提交时间：2019/12/11 Androgen receptor  Prostate cancer  Antagonists  Pyrazole derivatives   Discovery of novel pyrazole derivatives as potential anticancer agents in MCL 期刊论文 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 9, 页码: 1060-1064 作者:  Ran, Fansheng;  Liu, Yang;  Zhang, Daoguang;  Liu, Meixia;  Zhao, Guisen 收藏  |  浏览/下载：28/0  |  提交时间：2019/12/11 Mantle cell lymphoma  BTK  Irreversible inhibitors  Anticancer  Pyrazole  derivatives   Discovery of pyrazolopyrimidine derivatives as potent BTK inhibitors with effective anticancer activity in MCL 期刊论文 BIOORGANIC CHEMISTRY, 2019, 卷号: 89 作者:  Ran, Fansheng;  Liu, Yang;  Liu, Meixia;  Zhang, Daoguang;  Wang, Peng 收藏  |  浏览/下载：7/0  |  提交时间：2019/12/11 Mantle cell lymphoma  BTK inhibitors  Anticancer  Selectivity  Patient  cells   Discovery of novel 5-methyl-1H-pyrazole derivatives as potential antiprostate cancer agents: Design, synthesis, molecular modeling, and biological evaluation 期刊论文 CHEMICAL BIOLOGY & DRUG DESIGN, 2018, 卷号: 91, 期号: 6, 页码: 1113-1124 作者:  Zhang, Daoguang;  Asnake, Solomon;  Zhang, Jingya;  Olsson, Per-Erik;  Zhao, Guisen 收藏  |  浏览/下载：2/0  |  提交时间：2019/12/11 androgen receptor  AR antagonist  luciferase reporter gene assay  prostate cancer  pyrazole derivative   Design, synthesis and biological evaluation of AKT inhibitors bearing a piperidin-4-yl appendant 期刊论文 MEDCHEMCOMM, 2018, 卷号: 9, 期号: 8, 页码: 1340-1350 作者:  Zhang, Daoguang;  Tong, Dongdong;  Yang, Dezhi;  Sun, Jing;  Zhang, Fenghe 收藏  |  浏览/下载：5/0  |  提交时间：2019/12/11 Targeting Bruton's tyrosine kinase for the treatment of B cell associated malignancies and autoimmune diseases: Preclinical and clinical developments of small molecule inhibitors 期刊论文 ARCHIV DER PHARMAZIE, 2018, 卷号: 351, 期号: 7 作者:  Zhang, Zhen;  Zhang, Daoguang;  Liu, Yang;  Yang, Dezhi;  Ran, Fansheng 收藏  |  浏览/下载：5/0  |  提交时间：2019/12/11 arthritis  Bruton's tyrosine kinase  BTK inhibitor  leukemia  lymphoma   Structural optimization elaborates novel potent Akt inhibitors with promising anticancer activity 期刊论文 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 138, 页码: 543-551 作者:  Liu, Yang;  Yin, Yanzhen;  Zhang, Zhen;  Li, Carrie J.;  Zhang, Hui 收藏  |  浏览/下载：3/0  |  提交时间：2019/12/12 Akt  Anticancer  Docking  Mantle cell lymphoma  Piperidyl  Pyrrolopyrimidines   Recent Developments in Androgen Receptor Antagonists 期刊论文 ARCHIV DER PHARMAZIE, 2015, 卷号: 348, 期号: 11, 页码: 757-775 作者:  Ran, Fansheng;  Xing, Hualu;  Liu, Yang;  Zhang, Daoguang;  Li, Pengzhan 收藏  |  浏览/下载：4/0  |  提交时间：2019/12/17 Activation function-2  Androgen receptor antagonist  Binding function-3  Ligand binding domain  Prostate cancer   Design and discovery of 5-hydroxy-6-oxo-1,6-dihydropyrimidine-4-carboxamide inhibitors of HIV-1 integrase 期刊论文 Bioorganic and medicinal chemistry, 2014, 卷号: 22, 期号: 19, 页码: 5446-5453 作者:  Zhang, Daoguang;  Debnath, Bikash;  Yu, Shenghui;  Sanchez, Tino Wilson;  Christ, Frauke 收藏  |  浏览/下载：3/0  |  提交时间：2019/12/17 HIV-1 integrase inhibitors  INSTIs  5-Hydroxy-6-oxo-1  6-dihydropyrimidine analogues