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Optimization of piperidine constructed peptidyl derivatives as proteasome inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 29, 页码: 14
作者:  Zhao, Yanmei;  Xu, Lei;  Zhang, Jiankang;  Zhang, Mengmeng;  Lu, Jingyi
收藏  |  浏览/下载:21/0  |  提交时间:2021/05/24
Combinations of proteasome inhibitors with obatoclax are effective for small cell lung cancer 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020
作者:  Yin, Yan-ping;  Shi, Wen-hao;  Deng, Ke;  Liu, Xiao-li;  Li, Hong
收藏  |  浏览/下载:26/0  |  提交时间:2020/12/28
Bioinspired manganese complexes catalyzed epoxidation for the synthesis of the epoxyketone fragment of carfilzomib 期刊论文
Chinese Chemical Letters, 2019, 卷号: 30, 期号: 3, 页码: 698
作者:  Wei Sun;  Chungu Xia;  Bin Qiu
收藏  |  浏览/下载:15/0  |  提交时间:2019/11/28
Covalent docking modelling-based discovery of tripeptidyl epoxyketone proteasome inhibitors composed of aliphatic-heterocycles 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 164, 页码: 602-614
作者:  Dong, Xiao-Wu;  Zhang, Jian-Kang;  Xu, Lei;  Che, Jin-Xin;  Cheng, Gang
收藏  |  浏览/下载:35/0  |  提交时间:2020/07/01
Development of Macrocyclic Peptides Containing Epoxyketone with Oral Availability as Proteasome Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 61, 期号: 20, 页码: 9177-9204
作者:  Li, Daqiang;  Zhang, Xiaotuan;  Ma, Xiaodong;  Xu, Lei;  Yu, Jianjun
收藏  |  浏览/下载:30/0  |  提交时间:2019/01/08
Enhanced Glioblastoma Targeting Ability of Carfilzomib Enabled by a (D)A7R-Modified Lipid Nanodisk 期刊论文
MOLECULAR PHARMACEUTICS, 2018, 卷号: 15, 期号: 6
作者:  Zhang, Mingfei;  Lu, Linwei;  Ying, Man;  Ruan, Huitong;  Wang, Xiaoyi
收藏  |  浏览/下载:7/0  |  提交时间:2019/12/05
Lenalidomide and Low Dose Dexamethasone Plus Elotuzumab or Carfilzomib for Relapsed or Refractory Multiple Myeloma: A Comparison of Progression-Free Survival with Reconstructed Individual Participant Data 期刊论文
BIOMED RESEARCH INTERNATIONAL, 2018
作者:  Li, Shuo;  Meng, Xiang-Yu;  Maman, Souraka Tapara Dramani;  Xiao, Yong-Nong;  Li, Sheng
收藏  |  浏览/下载:1/0  |  提交时间:2019/12/05
Resveratrol Sensitizes Carfilzomib-Induced Apoptosis via Promoting Oxidative Stress in Multiple Myeloma Cells 期刊论文
2018, 卷号: 9, 页码: 334
作者:  Li, Qian;  Yue, Yuanfang;  Chen, Lin;  Xu, Chang;  Wang, Yan
收藏  |  浏览/下载:5/0  |  提交时间:2020/01/03
Exploration of novel piperazine or piperidine constructed non-covalent peptidyl derivatives as proteasome inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 126, 页码: 1056-1070
作者:  Zhuang, Rangxiao;  Gao, Lixin;  Lv, Xiaoqing;  Xi, Jianjun;  Sheng, Li
收藏  |  浏览/下载:21/0  |  提交时间:2019/01/08
蛋白酶体抑制剂Carfilzomib对子宫内膜癌的抗癌作用研究 学位论文
2017
作者:  王珂
收藏  |  浏览/下载:2/0  |  提交时间:2019/11/26


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