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Key Considerations in Targeted Protein Degradation Drug Discovery and Development 期刊论文
FRONTIERS IN CHEMISTRY, 2022, 卷号: 10
作者:  Qin, Liena;  Dai, Han;  Wang, Junfeng
收藏  |  浏览/下载:19/0  |  提交时间:2022/12/23
PROTAC: An Effective Targeted Protein Degradation Strategy for Cancer Therapy 期刊论文
FRONTIERS IN PHARMACOLOGY, 2021, 卷号: 12
作者:  Qi, Si-Min;  Dong, Jinyun;  Xu, Zhi-Yuan;  Cheng, Xiang-Dong;  Zhang, Wei-Dong
收藏  |  浏览/下载:47/0  |  提交时间:2021/06/15
Optimization of piperidine constructed peptidyl derivatives as proteasome inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 29, 页码: 14
作者:  Zhao, Yanmei;  Xu, Lei;  Zhang, Jiankang;  Zhang, Mengmeng;  Lu, Jingyi
收藏  |  浏览/下载:21/0  |  提交时间:2021/05/24
Targeting Protein Neddylation to Inactivate Cullin-RING Ligases by Gossypol: A Lucky Hit or a New Start? 期刊论文
DRUG DESIGN DEVELOPMENT AND THERAPY, 2021, 卷号: 15
作者:  Yu, Qing;  Sun, Yi
收藏  |  浏览/下载:21/0  |  提交时间:2021/03/15
Combinations of proteasome inhibitors with obatoclax are effective for small cell lung cancer 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020
作者:  Yin, Yan-ping;  Shi, Wen-hao;  Deng, Ke;  Liu, Xiao-li;  Li, Hong
收藏  |  浏览/下载:26/0  |  提交时间:2020/12/28
DCZ5248, a novel dual inhibitor of Hsp90 and autophagy, exerts antitumor activity against colon cancer 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 10
作者:  Chen, Xiang-ling;  Liu, Peng;  Zhu, Wei-liang;  Lou, Li-guang
收藏  |  浏览/下载:49/0  |  提交时间:2020/07/01
Xanthohumol, a Prenylated Flavonoid from Hops, Induces Caspase-Dependent Degradation of Oncoprotein BCR-ABL in K562 Cells 期刊论文
ANTIOXIDANTS, 2019, 卷号: 8, 期号: 9
作者:  Lu, Xuxiu;  Geng, Jiajia;  Zhang, Jinman;  Miao, Jinlai;  Liu, Ming
收藏  |  浏览/下载:30/0  |  提交时间:2019/10/29
Xanthohumol, a Prenylated Flavonoid from Hops, Induces Caspase-Dependent Degradation of Oncoprotein BCR-ABL in K562 Cells 期刊论文
ANTIOXIDANTS, 2019, 卷号: 8, 期号: 9
作者:  Lu, Xuxiu;  Geng, Jiajia;  Zhang, Jinman;  Miao, Jinlai;  Liu, Ming
收藏  |  浏览/下载:27/0  |  提交时间:2019/10/29
Covalent docking modelling-based discovery of tripeptidyl epoxyketone proteasome inhibitors composed of aliphatic-heterocycles 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 164, 页码: 602-614
作者:  Dong, Xiao-Wu;  Zhang, Jian-Kang;  Xu, Lei;  Che, Jin-Xin;  Cheng, Gang
收藏  |  浏览/下载:35/0  |  提交时间:2020/07/01
Exploration of novel macrocyclic dipeptide N-benzyl amides as proteasome inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 164, 页码: 423-439
作者:  Yu, Jianjun;  Liu, Jieyu;  Li, Daqiang;  Xu, Lei;  Hong, Duidui
收藏  |  浏览/下载:0/0  |  提交时间:2020/07/01


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