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Structure-based drug optimization and biological evaluation of tetrahydroquinolin derivatives as selective and potent CBP bromodomain inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 22, 页码: 7
作者:  Bi, Xiaoyang;  Chen, Yu;  Sun, Zhongya;  Lu, Wenchao;  Xu, Pan
收藏  |  浏览/下载:20/0  |  提交时间:2021/05/24
Design, synthesis, and biological evaluation of tetrahydroquinolin derivatives as potent inhibitors of CBP bromodomain 期刊论文
BIOORGANIC CHEMISTRY, 2020, 卷号: 101, 页码: 11
作者:  Chen, Yu;  Bi, Xiaoyang;  Zhang, Fengcai;  Sun, Zhongya;  Xu, Pan
收藏  |  浏览/下载:23/0  |  提交时间:2020/12/24
Discovery of novel CBP bromodomain inhibitors through TR-FRET-based high-throughput screening 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 卷号: 41, 期号: 2, 页码: 286-292
作者:  Zhang, Feng-cai;  Sun, Zhong-ya;  Liao, Li-ping;  Zuo, Yu;  Zhang, Dan
收藏  |  浏览/下载:29/0  |  提交时间:2020/07/01
discoveryofnovelcbpbromodomaininhibitorsthroughtrfretbasedhighthroughputscreening 期刊论文
actapharmacologicasinica, 2020, 卷号: 41, 期号: 2, 页码: 285
作者:  Zhang Fengcai;  Sun Zhongya;  Liao Liping;  Zuo Yu;  Zhang Dan
收藏  |  浏览/下载:35/0  |  提交时间:2020/07/01
Nut Directs p300-Dependent, Genome-Wide H4 Hyperacetylation in Male Germ Cells 期刊论文
CELL REPORTS, 2018, 卷号: 24, 期号: 13, 页码: 3477-+
作者:  Shiota, Hitoshi;  Barral, Sophie;  Buchou, Thierry;  Tan, Minjia;  Coute, Yohann
收藏  |  浏览/下载:66/0  |  提交时间:2019/01/08
Discovery and optimization of 1-(1H-indol-1-yl)ethanone derivatives as CBP/EP300 bromodomain inhibitors for the treatment of castration-resistant prostate cancer 期刊论文
2018, 卷号: 147, 页码: 238
作者:  Xiang, Qiuping[1];  Wang, Chao[1,3];  Zhang, Yan[1];  Xue, Xiaoqian[1];  Song, Ming[1]
收藏  |  浏览/下载:17/0  |  提交时间:2019/12/10
Recognition of Hyperacetylated N-terminus of H2AZ by TbBDF2 from Trypanosoma brucei. 期刊论文
Biochem J, 2017
作者:  Xu,Chao;  Zhang,Jiahai;  Yang,Xiao;  Zhang,Xuecheng;  Wu,Xuelei
收藏  |  浏览/下载:10/0  |  提交时间:2019/04/22
Brd3通过促进IL6基因启动子区乙酰基转移酶CBP的募集和组蛋白H3乙酰化修饰促进IL-6产生 期刊论文
2016, 卷号: 32, 期号: 10, 页码: 1301-1305
作者:  任文汇;  孙东豪;  王春梅;  李楠
收藏  |  浏览/下载:3/0  |  提交时间:2020/01/04
Dimeric structure of p300/CBP associated factor 期刊论文
http://dx.doi.org/10.1186/1472-6807-14-2, 2014
Shi, Shasha; Lin, Juanyu; Cai, Yongfei; Yu, Jiao; Hong, Haiyan; Ji, Kunmei; Downey, Jennifer S.; Lu, Xiaodong; Chen, Ruichuan; Han, Jiahuai; Han, Aidong; 韩家淮; 韩爱东
收藏  |  浏览/下载:5/0  |  提交时间:2015/07/22
Small organic molecules targeting PCAF bromodomain as potent inhibitors of HIV-1 replication 期刊论文
MEDCHEMCOMM, 2013, 卷号: 4, 期号: 4, 页码: 737-740
作者:  Wang Q;  Wang RR;  Zhang BQ;  Zhang S;  Zheng YT[*]
收藏  |  浏览/下载:9/0  |  提交时间:2013/08/28


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