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上海药物研究所 [13]
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Development of a traditional Chinese medicine-based agent for the treatment of cancer cachexia
期刊论文
JOURNAL OF CACHEXIA SARCOPENIA AND MUSCLE, 2022
作者:
Wu, Kun-Chang
;
Chu, Po-Chen
;
Cheng, Yu-Jung
;
Li, Chia-Ing
;
Tian, Jingkui
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2022/12/23
Cachexia
Traditional Chinese medicine
Muscle atrophy
C-26 tumour-bearing model
Caenorhabditis elegans model
Discovery of 5-(3-bromo-2-(2,3-dibromo-4,5-dimethoxybenzyl)-4,5-dimethoxybenzylidene)thiazolidine-2,4-dione as a novel potent protein tyrosine phosphatase 1B inhibitor with antidiabetic properties
期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 108, 页码: 13
作者:
Jiang, Bo
;
Luo, Jiao
;
Guo, Shuju
;
Wang, Lijun
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2021/05/11
Type 2 diabetes mellitus
Protein tyrosine phosphatase 1B inhibitors
Thiazolidinedione
Insulin signaling
Anti-diabetic activities
Valve-based consecutive bioprinting method for multimaterial tissue-like constructs with controllable interfaces
期刊论文
BIOFABRICATION, 2021, 卷号: 13, 期号: 3, 页码: 1-12
作者:
Wang HR(王赫然)
;
Guo K(郭凯)
;
Zhang LM(张黎明)
;
Zhu HX(朱慧轩)
;
Li SJ(李世杰)
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2021/04/24
bioprinting
multimaterial construct
material interface
printing efficiency
vascularized tissue
Antidiabetic activity in vitro and in vivo of BDB, a selective inhibitor of protein tyrosine phosphatase 1B, fromRhodomela confervoides
期刊论文
BRITISH JOURNAL OF PHARMACOLOGY, 2020, 卷号: 177, 期号: 19, 页码: 4464-4480
作者:
Luo, Jiao
;
Zheng, Meiling
;
Jiang, Bo
;
Li, Chao
;
Guo, Shuju
收藏
  |  
浏览/下载:136/0
  |  
提交时间:2020/09/29
bromophenol
PTP1B inhibitor
selectivity
cell permeability
oral bioavailability
TGR5 agonist ameliorates insulin resistance in skeletal muscles and improves glucose homeostasis in diabetic mice
期刊论文
METABOLISM-CLINICAL AND EXPERIMENTAL, 2019, 卷号: 99, 页码: 45-56
作者:
Huang, Suling
;
Ma, Shanyao
;
Ning, Mengmeng
;
Yang, Wenji
;
Ye, Yangliang
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2020/07/01
TGR5
Glucose homeostasis
Insulin resistance
Skeletal muscle
Type 2 diabetes
Effect of 2,3,7,8-tetrachlorodibenzo-p-dioxin exposure on acetylcholinesterase during myogenic differentiation of contractile rat primary skeletal muscle cells
期刊论文
CHEMICO-BIOLOGICAL INTERACTIONS, 2019, 卷号: 308, 页码: 164-169
作者:
Luo, Yali
;
Xie, Heidi Qunhui
;
Chen, Yangsheng
;
Xia, Yingjie
;
Sha, Rui
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2020/09/10
Dioxin
Acetylcholinesterase
Muscle contraction
Aryl hydrocarbon receptor
Primary skeletal muscle cell
Phosphorylation of TET2 by AMPK is indispensable in myogenic differentiation
期刊论文
EPIGENETICS & CHROMATIN, 2019, 卷号: 12, 页码: -
作者:
Zhang, Ting
;
Guan, Xiaowen
;
Choi, Un Lam
;
Dong, Qiang
;
Lam, Melody M. T.
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2020/10/21
AMPK
TET2
Phosphorylation
Myogenesis
PAX7
Highly Selective Protein Tyrosine Phosphatase Inhibitor, 2,2 ',3,3 '-Tetrabromo-4,4 ',5,5 '-tetrahydroxydiphenylmethane, Ameliorates Type 2 Diabetes Mellitus in BKS db Mice
期刊论文
MOLECULAR PHARMACEUTICS, 2019, 卷号: 16, 期号: 5, 页码: 1839-1850
作者:
Li, Chao
;
Luo, Jiao
;
Guo, Shuju
;
Jia, Xiaoling
;
Guo, Chuanlong
收藏
  |  
浏览/下载:72/0
  |  
提交时间:2019/08/28
type 2 diabetes mellitus
protein tyrosine phosphatase 1B
insulin resistance
hypoglycemic activity
dyslipidemia
Enhancement of Glucose Utilization by Loesenerine through AMPK Activation in Myotubes
期刊论文
CHEMICAL & PHARMACEUTICAL BULLETIN, 2018, 卷号: 66, 期号: 9, 页码: 885-886
作者:
Wang, Luo-Na
;
Jiang, Hao-Wen
;
Li, Jin-Long
;
Li, Jing-Ya
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2019/01/08
loesenerine
spermidine alkaloid
AMP-activated protein kinase activation
glucose uptake
2,3,7,8-Tetrachlorodibenzo-p-dioxin induces alterations in myogenic differentiation of C2C12 cells
期刊论文
ENVIRONMENTAL POLLUTION, 2018, 卷号: 235, 页码: 965-973
作者:
Li, Yunping
;
Fu, Hualing
;
Xie, Heidi Q.
;
Chen, Yangsheng
;
Xu, Tuan
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2019/06/20
2,3,7,8-tetrachlorodibenzo-p-dioxin
Acetylcholinesterase
C2C12 cells
Myogenic differentiation
Aryl hydrocarbon receptor (AhR)
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