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Repressing MYC by targeting BET synergizes with selective inhibition of PI3K alpha against B cell lymphoma 期刊论文
CANCER LETTERS, 2022, 卷号: 524, 页码: 206-218
作者:  Chen, Zi-qi;  Cao, Zhe-rui;  Wang, Yi;  Zhang, Xi;  Xu, Lan
收藏  |  浏览/下载:53/0  |  提交时间:2021/12/16
CYH33  MYC  P300  BET  B cell lymphoma  PI3K  
Identify potent SARS-CoV-2 main protease inhibitors via accelerated free energy perturbation-based virtual screening of existing drugs 期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2020, 卷号: 117, 期号: 44, 页码: 27381-27387
作者:  Li, Zhe;  Li, Xin;  Huang, Yi-You;  Wu, Yaoxing;  Liu, Runduo
收藏  |  浏览/下载:75/0  |  提交时间:2020/12/24
Cyclopeptide RA-V Inhibits Organ Enlargement and Tumorigenesis Induced by YAP Activation 期刊论文
CANCERS, 2018, 卷号: 10, 期号: 11
作者:  Ji, Xinyan;  Song, Lihua;  Sheng, Li;  Gao, Anhui;  Zhao, Yang
收藏  |  浏览/下载:78/0  |  提交时间:2019/01/08
Design, synthesis, and molecular docking study of 3H-imidazole[4,5-c]pyridine derivatives as CDK2 inhibitors 期刊论文
ARCHIV DER PHARMAZIE, 2018, 卷号: 351, 期号: 6
作者:  Wu, Yi-Zhe;  Ying, Hua-Zhou;  Xu, Lei;  Cheng, Gang;  Chen, Jing
收藏  |  浏览/下载:32/0  |  提交时间:2019/01/08
Discovery of Novel Inhibitors Targeting the Menin-Mixed Lineage Leukemia Interface Using Pharmacophore- and Docking-Based Virtual Screening 期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2016, 卷号: 56, 期号: 9, 页码: 1847-1855
作者:  Xu, Yuan;  Yue, Liyan;  Wang, Yulan;  Xing, Jin;  Chen, Zhifeng
收藏  |  浏览/下载:20/0  |  提交时间:2019/01/08
Fragment-Based Drug Discovery of 2-Thiazolidinones as BRD4 Inhibitors: 2. Structure-Based Optimization 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 58, 期号: 3, 页码: 1281-1297
作者:  Zhao, Lele;  Wang, Yingqing;  Cao, Danyan;  Chen, Tiantian;  Wang, Qi
收藏  |  浏览/下载:19/0  |  提交时间:2019/01/08
Pharmacokinetic evaluation of the anticancer prodrug simmitecan in different experimental animals 期刊论文
ACTA PHARMACOLOGICA SINICA, 2013, 卷号: 34, 期号: 11, 页码: 1437-1448
作者:  Hu, Zhe-yi;  Li, Xiu-xue;  Du, Fei-fei;  Yang, Jun-ling;  Niu, Wei
收藏  |  浏览/下载:22/0  |  提交时间:2019/01/08


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