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Inhibition of Autophagy by a Small Molecule through Covalent Modification of the LC3 Protein 期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2021, 页码: 11
作者:  Fan, Shijie;  Yue, Liyan;  Wan, Wei;  Zhang, Yuanyuan;  Zhang, Bidong
收藏  |  浏览/下载:80/0  |  提交时间:2021/12/16
Discovery of a subtype-selective, covalent inhibitor against palmitoylation pocket of TEAD3 期刊论文
ACTA PHARMACEUTICA SINICA B, 2021, 卷号: 11, 期号: 10, 页码: 3206-3219
作者:  Lu, Tian;  Li, Yong;  Lu, Wenchao;  Spitters, Twgm;  Fang, Xueyu
收藏  |  浏览/下载:41/0  |  提交时间:2021/12/01
Discovery of High-Affinity Inhibitors of the BPTF Bromodomain 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 16, 页码: 12075-12088
作者:  Lu, Tian;  Lu, Haibo;  Duan, Zhe;  Wang, Jun;  Han, Jie
收藏  |  浏览/下载:38/0  |  提交时间:2021/11/04
Facing small and biased data dilemma in drug discovery with enhanced federated learning approaches 期刊论文
SCIENCE CHINA-LIFE SCIENCES, 2021, 页码: 11
作者:  Xiong, Zhaoping;  Cheng, Ziqiang;  Lin, Xinyuan;  Xu, Chi;  Liu, Xiaohong
收藏  |  浏览/下载:45/0  |  提交时间:2021/11/04
SARS-CoV-2 envelope protein causes acute respiratory distress syndrome (ARDS)-like pathological damages and constitutes an antiviral target 期刊论文
CELL RESEARCH, 2021, 页码: 14
作者:  Xia, Bingqing;  Shen, Xurui;  He, Yang;  Pan, Xiaoyan;  Liu, Feng-Liang
收藏  |  浏览/下载:78/0  |  提交时间:2021/08/17
Design, synthesis, and biological evaluation of 4-benzoylamino-1H-pyrazole-3-carboxamide derivatives as potent CDK2 inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 215, 页码: 12
作者:  Lin, Tingting;  Li, Jiacheng;  Liu, Liping;  Li, Yuanqing;  Jiang, Hualiang
收藏  |  浏览/下载:70/0  |  提交时间:2021/05/24
Reply to: Binding site for MDL-801 on SIRT6 期刊论文
NATURE CHEMICAL BIOLOGY, 2021, 页码: 5
作者:  Huang, Zhimin;  Zhao, Junxing;  Deng, Wei;  Chen, Yingyi;  Shang, Jialin
收藏  |  浏览/下载:64/0  |  提交时间:2021/05/24
Sorting Nexin 10 Mediates Metabolic Reprogramming of Macrophages in Atherosclerosis Through the Lyn-Dependent TFEB Signaling Pathway 期刊论文
CIRCULATION RESEARCH, 2020, 卷号: 127, 期号: 4, 页码: 534-549
作者:  You, Yan;  Bao, Wei-Lian;  Zhang, Su-Lin;  Li, Hai-Dong;  Li, Hui
收藏  |  浏览/下载:48/0  |  提交时间:2020/12/24
Structure of M-pro from SARS-CoV-2 and discovery of its inhibitors 期刊论文
NATURE, 2020, 页码: 24
作者:  Jin, Zhenming;  Du, Xiaoyu;  Xu, Yechun;  Deng, Yongqiang;  Liu, Meiqin
收藏  |  浏览/下载:41/0  |  提交时间:2020/07/01
Full-length human GLP-1 receptor structure without orthosteric ligands 期刊论文
naturecommunications, 2020, 卷号: 11, 期号: 1, 页码: 1
作者:  Fan Wu;  Linlin Yang;  Kaini Hang;  Mette Laursen;  Lijie Wu
收藏  |  浏览/下载:26/0  |  提交时间:2020/07/01


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