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浏览/检索结果: 共9条，第1-9条 帮助 限定条件 发表日期：2020    专题：上海药物研究所    第一署名单位    第一作者单位    通讯作者单位     已选(0)清除 条数/页：5101520253035404550556065707580859095100   排序方式：请选择作者升序作者降序题名升序题名降序发表日期升序发表日期降序提交时间升序提交时间降序 A Peptide Binder of E3 Ligase Adaptor SPOP Disrupts Oncogenic SPOP-Protein Interactions in Kidney Cancer Cells 期刊论文 CHINESE JOURNAL OF CHEMISTRY, 2020, 页码: 274-280 作者:  Wang, Zhen;  Zhang, Hao;  Chen, Baoen;  Ouyang, Sisheng;  Zheng, Tong 收藏  |  浏览/下载：124/0  |  提交时间：2021/05/24 SPOP  Protein‐  protein interaction  Clear cell Renal Cell Carcinomas  Crystal structure  Peptide inhibitor   Tideglusib and Its Analogues As Inhibitors of Staphylococcus aureus SrtA 期刊论文 JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 15, 页码: 8442-8457 作者:  Yang, Teng;  Zhang, Tao;  Guan, Xiang-Na;  Dong, Ze;  Lan, Lefu 收藏  |  浏览/下载：22/0  |  提交时间：2020/12/24 Structure-Activity Relationship of SPOP Inhibitors against Kidney Cancer 期刊论文 JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 9, 页码: 4849-4866 作者:  Dong, Ze;  Wang, Zhen;  Guo, Zhong-Qiang;  Gong, Shouzhe;  Zhang, Tao 收藏  |  浏览/下载：45/0  |  提交时间：2020/07/01 2-Oxo-3,4-dihydropyrimido[4,5-d] pyrimidines as new reversible inhibitors of EGFR C797S (Cys797 to Ser797) mutant 期刊论文 CHINESE CHEMICAL LETTERS, 2020, 卷号: 31, 期号: 5, 页码: 1281-1287 作者:  Hu, Xianglong;  Xun, Qiuju;  Zhang, Tao;  Zhu, Su-Jie;  Li, Qian 收藏  |  浏览/下载：47/0  |  提交时间：2020/07/01 EGFR(C797S) mutant  SARs  2-Oxo-3,4-dihydropyrimido[4,5-d] pyrimidine  Clinical resistance  Fourth-generation inhibitors   High-throughput screening campaign identifies a small molecule agonist of the relaxin family peptide receptor 4 期刊论文 ACTA PHARMACOLOGICA SINICA, 2020, 页码: 9 作者:  Lin, Guang-yao;  Lin, Lin;  Cai, Xiao-qing;  Dai, An-tao;  Zhu, Yue 收藏  |  浏览/下载：28/0  |  提交时间：2020/07/01 RXFP4  INSL5  high-throughput screening  agonist  JK1   Design and synthesis of Imidazo[1,2-b]pyridazine IRAK4 inhibitors for the treatment of mutant MYD88 L265P diffuse large B-cell lymphoma 期刊论文 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 190, 页码: 14 作者:  Chen, Yun;  Bai, Gang;  Ning, Yi;  Cai, Shi;  Zhang, Tao 收藏  |  浏览/下载：24/0  |  提交时间：2020/07/01 lnterleukin-1 receptor associated kinase 4  Imidazol1,2-6]pyridazine  Diffuse large B-cell lymphoma  Drug design  Antitumor agents   Discovery of novel CBP bromodomain inhibitors through TR-FRET-based high-throughput screening 期刊论文 ACTA PHARMACOLOGICA SINICA, 2020, 卷号: 41, 期号: 2, 页码: 286-292 作者:  Zhang, Feng-cai;  Sun, Zhong-ya;  Liao, Li-ping;  Zuo, Yu;  Zhang, Dan 收藏  |  浏览/下载：31/0  |  提交时间：2020/07/01 CBP bromodomain  small-molecule inhibitor  high-throughput screening  TR-FRET  molecular modeling  human leukemia MV4-11 cells   Introducing "Future of Biochemistry 2020: The Asia-Pacific Issue" 期刊论文 BIOCHEMISTRY, 2020, 卷号: 59, 期号: 1, 页码: 1-7 作者:  Ananthanarayanan, Vaishnavi;  Chattopadhyay, Kausik;  Chen, Lei;  Cheng, Liang;  Edgington-Mitchell, Laura 收藏  |  浏览/下载：17/0  |  提交时间：2020/07/01 Analysis of Four Types of Leukemia Using Gene Ontology Term and Kyoto Encyclopedia of Genes and Genomes Pathway Enrichment Scores 期刊论文 COMBINATORIAL CHEMISTRY & HIGH THROUGHPUT SCREENING, 2020, 卷号: 23, 期号: 4, 页码: 295-303 作者:  Lu, Jing;  Zhang, YuHang;  Wang, ShaoPeng;  Bi, Yi;  Huang, Tao 收藏  |  浏览/下载：35/0  |  提交时间：2020/07/01 Leukemia  protein-drug interactions  GO term  KEGG pathway  enrichment score  mRMR