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上海药物研究所 [6]
复旦大学上海医学院 [5]
西安交通大学 [3]
武汉大学 [3]
江苏大学 [2]
山东大学 [2]
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期刊论文 [30]
发表日期
2018 [30]
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Design and optimization of 2,3-dihydrobenzo[b][1,4]dioxine propanoic acids as novel GPR40 agonists with improved pharmacokinetic and safety profiles
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 22, 页码: 5780-5791
作者:
Guo, Bin
;
Guo, Shimeng
;
Huang, Jing
;
Li, Jingya
;
Li, Jia
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2019/01/08
GPR40 agonist
2,3-Dihydrobenzo[b][1,4]dioxine
Insulin secretion
Type 2 diabetes mellitus
ETA as a novel Kv2.1 inhibitor ameliorates beta-cell dysfunction and hyperglycaemia
期刊论文
CLINICAL AND EXPERIMENTAL PHARMACOLOGY AND PHYSIOLOGY, 2018, 卷号: 45, 期号: 12, 页码: 1257-1264
作者:
Zhou, Tingting
;
Du, Mengfan
;
Zhao, Tong
;
Quan, Lingling
;
Zhu, Zhiyuan
收藏
  |  
浏览/下载:94/0
  |  
提交时间:2019/01/08
beta cell
apoptosis
glucose-stimulated insulin secretion
T2DM
A novel plectin/integrin-targeted bispecific molecular probe for magnetic Check tat resonance/near-infrared imaging of pancreatic cancer
期刊论文
BIOMATERIALS, 2018, 卷号: 183, 页码: 173-184
作者:
Wang, Qian
;
Yan, Hao
;
Jin, Yushen
;
Wang, Zihua
;
Huang, Wenhui
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2019/12/16
Bispecific peptides
Early diagnosis
Molecular imaging
Pancreatic cancer
Theranostics
A preclinical overview of metformin for the treatment of type 2 diabetes
期刊论文
BIOMEDICINE & PHARMACOTHERAPY, 2018, 卷号: 106, 页码: 1227-1235
作者:
Zhou, Tingting
;
Xu, Xin
;
Du, Mengfan
;
Zhao, Tong
;
Wang, Jiaying
收藏
  |  
浏览/下载:46/0
  |  
提交时间:2019/01/08
Gluconeogenesis
Insulin sensitivity
Mechanism
Metformin
Type 2 diabetes (T2D)
Selection of growth-related genes and dominant genotypes in transgenic Yellow River carp Cyprinus carpio L.
期刊论文
FUNCTIONAL & INTEGRATIVE GENOMICS, 2018, 卷号: 18, 期号: 4, 页码: 425-437
作者:
Luo, Lifei
;
Huang, Rong
;
Zhang, Aidi
;
Yang, Cheng
;
Chen, Liangming
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  |  
浏览/下载:46/0
  |  
提交时间:2019/07/03
Transgenic Yellow River carp
Growth-related genes
Genotype
Bulked segregant analysis (BSA)
Genome-wide association study (GWAS)
Structural characterization of a galactan from Ophiopogon japonicus and anti-pancreatic cancer activity of its acetylated derivative
期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2018, 卷号: 113, 页码: 907-915
作者:
Gu, Dan
;
Huang, Lulin
;
Chen, Xia
;
Wu, Qianhu
;
Ding, Kan
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  |  
浏览/下载:74/0
  |  
提交时间:2019/01/08
Ophiopogon japonicus
Polysaccharide
Acetylated derivative
Apoptosis
Anti-pancreatic cancer
Design, synthesis and structure activity relationship studies of GPR40 agonists containing amide linker
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 152, 页码: 175-194
作者:
Chen, Tingting
;
Ning, Mengmeng
;
Ye, Yangliang
;
Wang, Kai
;
Leng, Ying
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  |  
浏览/下载:31/0
  |  
提交时间:2019/01/08
GPR40
FFAR1
Insulin secretion
Type 2 diabetes mellitus
CNS
Clinical and Physiological Characterization of Elevated Plasma Glucagon-Like Peptide-1 Levels (Hyperglipemia) in a Dipeptidyl Peptidase IV Mutation Carrier
期刊论文
FRONTIERS IN ENDOCRINOLOGY, 2018, 卷号: 9
作者:
Zhao, Dandan
;
Zhao, Shaoqian
;
Wang, Xiao
;
Su, Mingbo
;
Liu, Wen
收藏
  |  
浏览/下载:59/0
  |  
提交时间:2019/01/08
dipeptidyl peptidase IV
glucagon-like peptide-1
beta-cell function
type 2 diabetes
incretin effect
PICK1 is essential for insulin production and the maintenance of glucose homeostasis.
期刊论文
MOLECULAR BIOLOGY OF THE CELL, 2018
作者:
Xia, Jun
;
Li, Jia
;
Mao, Zhuo
;
Huang, Jiandong
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  |  
浏览/下载:23/0
  |  
提交时间:2019/01/31
SNX6 predicts poor prognosis and contributes to the metastasis of pancreatic cancer cells via activating epithelial-mesenchymal transition
期刊论文
ACTA BIOCHIMICA ET BIOPHYSICA SINICA, 2018, 卷号: 50, 期号: 11
作者:
Hu, Pengfei
;
Liang, Yun
;
Hu, Qiangsheng
;
Wang, Hongwei
;
Cai, Zhiwei
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2019/12/05
pancreatic cancer
SNX6
TGF-beta
EMT
ZEB1
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