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厦门大学 [19]
大连化学物理研究所 [19]
上海药物研究所 [6]
中国科学院大学 [3]
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期刊论文 [63]
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Combining Michaelis-Menten theory and enzyme deactivation reactions for the kinetic study of enzymatic hydrolysis by different pretreated sugarcane bagasse
期刊论文
PROCESS BIOCHEMISTRY, 2021, 卷号: 105, 页码: 72-78
作者:
Zhang, Yu
;
Zhang, Ying
;
Song, Miaojia
;
Topakas, Evangelos
;
Yu, Qiang
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浏览/下载:50/0
  |  
提交时间:2021/10/27
Enzymatic kinetics
Michaelis-Menten theory
Enzyme deactivation
Cellulase
Xylanase
Discovery and characterization of natural products as novel indoleamine 2,3-dioxygenase 1 inhibitors through high-throughput screening
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 卷号: 41, 期号: 3, 页码: 423-431
作者:
Guo, Wei
;
Yao, Sheng
;
Sun, Pu
;
Yang, Tian-biao
;
Tang, Chun-ping
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  |  
浏览/下载:79/0
  |  
提交时间:2020/07/01
indoleamine 2
3-dioxygenase 1 inhibitor
natural product library
high-throughput fluorescence-based screening
discoveryandcharacterizationofnaturalproductsasnovelindoleamine23dioxygenase1inhibitorsthroughhighthroughputscreening
期刊论文
actapharmacologicasinica, 2020, 卷号: 41, 期号: 3, 页码: 423
作者:
Guo Wei
;
Yao Sheng
;
Sun Pu
;
Yang Tianbiao
;
Tang Chunping
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  |  
浏览/下载:81/0
  |  
提交时间:2020/07/01
indoleamine 2
3-dioxygenase 1 inhibitor
natural product library
high-throughput fluorescence-based screening
Cytochrome P450 3A Enzymes Are Key Contributors for Hepatic Metabolism of Bufotalin, a Natural Constitute in Chinese Medicine Chansu
期刊论文
FRONTIERS IN PHARMACOLOGY, 2019, 卷号: 10, 页码: 10
作者:
Ma, Hong-Ping
;
Dai, Zi-Ru
;
Ning, Jing
;
Sun, Gui-Bo
;
Wang, Ping
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  |  
浏览/下载:65/0
  |  
提交时间:2019/06/20
bufotalin
cytochrome P450 3A (CYP3A)
hydroxylation
human liver microsomes (HLMs)
docking simulations
Cytochrome p450 3a enzymes are key contributors for hepatic metabolism of bufotalin, a natural constitute in chinese medicine chansu
期刊论文
Frontiers in pharmacology, 2019, 卷号: 10, 页码: 10
作者:
Dai, Zi-Ru
;
Ning, Jing
;
Sun, Gui-Bo
;
Wang, Ping
;
Zhang, Feng
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  |  
浏览/下载:87/0
  |  
提交时间:2019/05/08
Bufotalin
Cytochrome p450 3a (cyp3a)
Hydroxylation
Human liver microsomes (hlms)
Docking simulations
Resveratroloside Alleviates Postprandial Hyperglycemia in Diabetic Mice by Competitively Inhibiting alpha-Glucosidase
期刊论文
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2019, 卷号: 67, 期号: 10
作者:
Zhao, Xiaohui
;
Tao, Jihong
;
Zhang, Ting
;
Jiang, Sirong
;
Wei, Wei
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  |  
浏览/下载:68/0
  |  
提交时间:2019/11/26
alpha-glucosidase
postprandial blood glucose
diabetes mellitus
resveratroloside
competitive inhibition
Antidiabetic Stilbenes from Peony Seeds with PTP1B, alpha-Glucosidase, and DPPIV Inhibitory Activities
期刊论文
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2019, 卷号: 67, 期号: 24, 页码: 6765-6772
作者:
Zhang,Chen-Chen
;
Geng,Chang-An
;
Huang,Xiao-Yan
;
Zhang,Xue-Mei
;
Chen,Ji-Jun
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  |  
浏览/下载:5/0
  |  
提交时间:2020/04/02
固定化酶的制备及其酶抑制剂筛选的研究
学位论文
北京: 中国科学院大学, 2018
作者:
刘冬梅
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  |  
浏览/下载:14/0
  |  
提交时间:2020/09/21
压力中介微分析
固定化酶
磁性载体
酶动力学研究
抑制剂筛选
Pressure mediated microanalysis
Immobilized enzyme
Magnetic immobilization carrier
Enzyme kinetic and inhibition study
Enzyme inhibitor screening
Inhibition of thrombin by functionalized C-60 nanoparticles revealed via in vitro assays and in silico studies
期刊论文
JOURNAL OF ENVIRONMENTAL SCIENCES-CHINA, 2018, 卷号: 63, 页码: 285-295
作者:
Liu, Yanyan
;
Fu, Jianjie
;
Pan, Wenxiao
;
Xue, Qiao
;
Liu, Xian
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  |  
浏览/下载:35/0
  |  
提交时间:2019/06/20
Thrombin
C-60 nanoparticle (NP)
Surface modification
Activity inhibition
Quantitative nanostructure-activity relationship
Molecular docking
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