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科研机构
华中师范大学 [10]
内容类型
期刊论文 [10]
发表日期
2019 [4]
2017 [3]
2015 [2]
2007 [1]
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专题:华中师范大学
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In silico screening of a novel scaffold for fructose-1,6-bisphosatase (FBPase) inhibitors
期刊论文
Journal of Molecular Graphics and Modelling, 2019, 卷号: 86, 页码: 142-148
作者:
Huang, Yunyuan
;
Chi, Bo
;
Xu, Yanhong
;
Song, Rongrong
;
Wei, Lin
收藏
  |  
浏览/下载:32/0
  |  
提交时间:2019/12/23
Fructose-1,6-bisphosphate (FBPase)
FBPase inhibitors
DOX2.0
FBPase
fructose-1,6-bisphosphatase
FBP
fructose-1,6-biphosphate
IC50
half maximal inhibitory concentration
PAINS
Pan Assay Interference
T2D
Type 2 diabetes
SAR
structure−activity relationship
EGP
endogenous glucose production
GNG
gluconeogenesis
AMP
adenosine monophosphate
DOX
Docking ONIOM eXtended ONIOM (XO)
DOX2.0
Docking PM7@Mopac XO2
LE
ligand efficiency
LELP
lipophilicity-corrected ligand efficiency
Pyrazole-Isoindoline-1,3-dione Hybrid: A Promising Scaffold for 4-Hydroxyphenylpyruvate Dioxygenase Inhibitors.
期刊论文
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2019, 卷号: 67, 期号: 39, 页码: 10844-10852
作者:
He, Bo
;
Dong, Jin
;
Lin, Hong-Yan
;
Wang, Meng-Yao
;
Li, Xian-Kai
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2019/12/23
4-hydroxyphenylpyruvate dioxygenase
X-ray crystallography
inhibition kinetics
isoindoline-1,3-dione
pyrazole
2,7-naphthyridinone-based MET kinase inhibitors: A promising novel scaffold for antitumor drug development
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 178, 页码: 705-714
作者:
Zhuo, Lin-Sheng
;
Xu, Hong-Chuang
;
Wang, Ming-Shu
;
Zhao, Xing-E
;
Ming, Zhi-Hui
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/12/23
2,7-Naphthyridone
Antitumor
In vivo efficacy
MET kinase inhibitor
Design, synthesis and algicides activities of thiourea derivatives as the novel scaffold aldolase inhibitors.
期刊论文
Bioorganic & medicinal chemistry, 2019, 卷号: 27, 期号: 5, 页码: 805-812
作者:
Xiao, Shan
;
Wei, Lin
;
Hong, Zongqin
;
Rao, Li
;
Ren, Yanliang*
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2019/12/23
Aldolases
Algicides activities
De novo discovery
Fragment-based Virtual Screen
Thiourea
A C-H Oxidation/Two-Fold Cyclization Approach to Imidazopyridoindole Scaffold under Mild Oxidizing Conditions
期刊论文
Journal of Organic Chemistry, 2017, 卷号: 82, 期号: 24, 页码: 13671-13677
作者:
Xiang, Jia-Chen
;
Wang, Zi-Xuan
;
Cheng, Yan
;
Ma, Jin-Tian
;
Wang, Miao
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/23
One-step synthesis of carbon nanosheet-decorated carbon nanofibers as a 3D interconnected porous carbon scaffold for lithium-sulfur batteries
期刊论文
Journal of Materials Chemistry A, 2017, 卷号: 5, 期号: 45, 页码: 23737-23743
作者:
Feng, Shuo
;
Song, Junhua
;
Fu, Shaofang
;
Zhu, Chengzhou
;
Shi, Qiurong
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/23
Phosphoprotein/chitosan electrospun nanofibrous scaffold for biomineralization
期刊论文
International Journal of Biological Macromolecules, 2017, 卷号: 102, 页码: 218-224
作者:
Liang, Hongshan
;
Sheng, Feng
;
Zhou, Bin
;
Pei, Yaqiong
;
Li, Bin
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2019/12/23
Phosvitin
Chitosan
Electrospun
Biomineralization
Biocompatibility
Discovery of novel Bruton's tyrosine kinase (BTK) inhibitors bearing a pyrrolo[2,3-d]pyrimidine scaffold
期刊论文
Bioorganic and Medicinal Chemistry, 2015, 卷号: 23, 期号: 4, 页码: 891-901
作者:
Zhao, Xinge
;
Huang, Wei
;
Wang, Yazhou
;
Xin, Minhang
;
Jin, Qiu
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/23
BTK inhibitors
Pyrrolo[23-d]pyrimidine
SAR
Enhanced liver functions of HepG2 cells in the alginate/xyloglucan scaffold
期刊论文
Biotechnology Letters, 2015, 卷号: 37, 期号: 1, 页码: 235-240
作者:
Deng, Xiaojie
;
Cao, Yu
;
Yan, Hao
;
Yang, Jihong
;
Xiong, Guomei
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/23
Albumin synthesis
Ammonia elimination
Encapsulation
HepG2 cell line
Liver tissue engineering
Xyloglucan
Discovery of a new insecticide lead by optimizing a target-diverse scaffold: Tetrazolinone derivatives
期刊论文
Bioorganic and Medicinal Chemistry, 2007, 卷号: 15, 期号: 4, 页码: 1716-1724
作者:
Luo, Yan-Ping(杨光富)
;
Yang, Guang-Fu*
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2019/12/23
1,3,4-Oxadiazole
1,3,4-Thiadiazole
Insecticidal activity
Lead compound
Tetrazolinone
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