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科研机构
北京大学 [6]
化学研究所 [2]
中国医学科学院 北京... [1]
生态环境研究中心 [1]
内容类型
期刊论文 [9]
其他 [1]
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2018 [2]
2016 [2]
2014 [5]
2009 [1]
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Small molecules capable of activating DNA methylation-repressed genes targeted by the p38 mitogen-activated protein kinase pathway
期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2018, 卷号: 293, 期号: 19, 页码: 7423-7436
作者:
Shao, Wei
;
Wang, Hailin
;
Zheng, Yong
;
Li, Xiang
;
Zhao, Zuodong
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2019/06/20
DNA methylation
high-throughput screening (HTS)
p38
mitogen-activated protein kinase (MAPK)
gene regulation
gene activation
Small molecules capable of activating DNA methylation-repressed genes targeted by the p38 mitogen-activated protein kinase pathway
期刊论文
2018, 卷号: 293, 期号: 19, 页码: 7423-7436
作者:
Li, Xiang
;
Shang, Erchang
;
Dong, Qiang
;
Li, Yingfeng
;
Zhang, Jing
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2020/01/03
DNA methylation
high-throughput screening (HTS)
p38
mitogen-activated protein kinase (MAPK)
gene regulation
gene activation
Syntheses of [1,2,4]triazolo[1,5-a]benzazoles enabled by the transition-metal-free oxidative N-N bond formation
期刊论文
CHEMICAL COMMUNICATIONS, 2016
Shang, Erchang
;
Zhang, Junzhi
;
Bai, Jinyi
;
Wang, Zhan
;
Li, Xiang
;
Zhu, Bing
;
Lei, Xiaoguang
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2017/12/03
AZO-COMPOUNDS
ONE-POT
C-N
1,2,4-TRIAZOLES
1,2,3-TRIAZOLES
CYCLIZATION
EFFICIENT
TOSYLHYDRAZONES
ANILINES
OXIDANT
Discovery of Novel 15-Lipoxygenase Activators To Shift the Human Arachidonic Acid Metabolic Network toward Inflammation Resolution
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016
Meng, Hu
;
McClendon, Christopher L.
;
Dai, Ziwei
;
Li, Kenan
;
Zhang, Xiaoling
;
He, Shan
;
Shang, Erchang
;
Liu, Ying
;
Lai, Luhua
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2017/12/03
INHIBITION
ENZYMES
MODEL
SITE
BIOSYNTHESIS
PROSTACYCLIN
PROTEINS
EFFECTOR
SYNTHASE
LIGANDS
Benzo[d] isothiazole 1,1-dioxide derivatives as dual functional inhibitors of 5-lipoxygenase and microsomal prostaglandin E-2 synthase-1
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 12, 页码: 2764-2767
作者:
Shang, Erchang
;
Wu, Yiran
;
Liu, Pei
;
Liu, Ying
;
Zhu, Wei
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2019/04/09
5-lipoxygenase
Microsomal Prostaglandin E-2 Synthase
Dual Functional Inhibitor
Benzo[d] Isothiazole 1
1-dioxide
De Novo Design of Multitarget Ligands with an Iterative Fragment-Growing Strategy
期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2014, 卷号: 54, 期号: 4, 页码: 1235-1241
作者:
Shang, Erchang
;
Yuan, Yaxia
;
Chen, Xinyi
;
Liu, Ying
;
Pei, Jianfeng
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/04/09
De Novo Design of Multitarget Ligands with an Iterative Fragment-Growing Strategy
期刊论文
journal of chemical information and modeling, 2014
Shang, Erchang
;
Yuan, Yaxia
;
Chen, Xinyi
;
Liu, Ying
;
Pei, Jianfeng
;
Lai, Luhua
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2015/11/10
HUMAN WHOLE-BLOOD
DRUG DISCOVERY
MULTIPLE LIGANDS
LEAD DISCOVERY
CYCLOOXYGENASE
INHIBITORS
BIOSYNTHESIS
NETWORK
BIOLOGY
Benzo[d] isothiazole 1,1-dioxide derivatives as dual functional inhibitors of 5-lipoxygenase and microsomal prostaglandin E-2 synthase-1
期刊论文
生物有机化学与医药化学通讯, 2014
Shang, Erchang
;
Wu, Yiran
;
Liu, Pei
;
Liu, Ying
;
Zhu, Wei
;
Deng, Xiaobing
;
He, Chong
;
He, Shan
;
Li, Cong
;
Lai, Luhua
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2015/11/10
Benzo[d] isothiazole 1,1-dioxide
5-Lipoxygenase
Microsomal prostaglandin E-2 synthase
Dual functional inhibitor
ANTIINFLAMMATORY DRUGS
MPGES-1
BIOLOGY
TARGET
5-LOX
Development of 3,5-dinitrobenzoate-based 5-lipoxygenase inhibitors
期刊论文
生物有机化学与医药化学, 2014
Shang, Erchang
;
Liu, Ying
;
Wu, Yiran
;
Zhu, Wei
;
He, Chong
;
Lai, Luhua
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2015/11/10
3,5-Dinitrobenzoate
5-Lipoxygenase inhibitors
Cell-free assay
Human whole blood assay
SAR study
DISEASE
BIOSYNTHESIS
LEUKOTRIENES
INFLAMMATION
EICOSANOIDS
MECHANISMS
SOLUTION STRUCTURE OF DROSOPHILA SNF:IMPLICATIONS FOR ITS ROLE IN SEX-LETHAL SPLICING
其他
2009-01-01
Jicheng HU
;
Gaofeng CUI
;
Congmin LI
;
Cong LIU
;
Erchang SHANG
;
Luhua LAI
;
Changwen JIN
;
Jiwu WANG
;
Bin XIA
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2017/12/03
lethal
Drosophila
switch
splicing
tracts
RNA
mammalian
homologue
specifically
inhibit
lethal
Drosophila
switch
splicing
tracts
RNA
mammalian
homologue
specifically
inhibit
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