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上海药物研究所 [13]
西北高原生物研究所 [9]
昆明植物研究所 [6]
复旦大学上海医学院 [4]
武汉植物园 [3]
新疆理化技术研究所 [2]
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期刊论文 [41]
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Novel tetrahydrobenzo[b]thiophen-2-yl)urea derivatives as novel alpha-glucosidase inhibitors: Synthesis, kinetics study, molecular docking, and in vivo anti-hyperglycemic evaluation
期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 115, 页码: 17
作者:
Xie, Hong-Xu
;
Zhang, Juan
;
Li, Yue
;
Zhang, Jin-He
;
Liu, Shan-Kui
收藏
  |  
浏览/下载:68/0
  |  
提交时间:2021/11/04
Tetrahydrobenzo[b]thiophen-2-yl)urea
alpha-Glucosidase inhibitors
Non-competitive inhibitor
Molecular docking
Anti-hyperglycaemic activity
Type 2 diabetes
New cembrane-type diterpenoids from the South China Sea soft coral Sinularia crassa and their alpha-glucosidase inhibitory activity
期刊论文
BIOORGANIC CHEMISTRY, 2020, 卷号: 104, 页码: 6
作者:
Wu, Meng-Jun
;
Wang, Hong
;
Jiang, Cheng-Shi
;
Guo, Yue-Wei
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2021/05/24
Sinularia crassa
Cembranoid
Modified Mosher's method
ECD calculation
alpha-Glucosidase inhibitor
Chemical Composition, Antioxidant, and Antimicrobial Activities of the Essential Oils From Artemisia annua L. Growing Wild in Tajikistan
期刊论文
NATURAL PRODUCT COMMUNICATIONS, 2020, 卷号: 15, 期号: 5, 页码: 1-7
作者:
Sharopov, FS (Sharopov, Farukh S.)[ 1,2 ]
;
Salimov, A (Salimov, Aminjon)[ 3 ]
;
Numonov, S (Numonov, Sodik)[ 1,2 ]
;
Safomuddin, A (Safomuddin, Abduahad)[ 4 ]
;
Bakri, M (Bakri, Mahinur)[ 2 ]
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  |  
浏览/下载:3/0
  |  
提交时间:2020/07/06
chemotype
Artemisia annua
essential oil
cluster analysis
camphor
1,8-cineole
Phytochemical Study on the Essential Oils of Tarragon (Artemisia dracunculus L.) Growing in Tajikistan and Its Comparison With the Essential Oil of the Species in the Rest of the World
期刊论文
NATURAL PRODUCT COMMUNICATIONS, 2020, 卷号: 15, 期号: 12, 页码: 1-7
作者:
Sharopov, FS (Sharopov, Farukh S.)[ 1,2 ]
;
Salimov, A (Salimov, Aminjon)[ 3 ]
;
Numonov, S (Numonov, Sodik)[ 1,2 ]
;
Bakri, M (Bakri, Mahinur)[ 2 ]
;
Sangov, Z (Sangov, Zafar)[ 4 ]
收藏
  |  
浏览/下载:116/0
  |  
提交时间:2021/03/19
Artemisia dracunculus
essential oil
GC-MS
cluster analysis
chemotype
sabinene
estragole
Biomimetic synthesis of the natural product salviadione and its hybrids: discovery of tissue-specific anti-inflammatory agents for acute lung injury
期刊论文
CHEMICAL SCIENCE, 2019, 卷号: 10, 期号: 17, 页码: 4667-4672
作者:
Ding, Chunyong
;
Chen, Hongjin
;
Liang, Bin
;
Jiao, Mingkun
;
Liang, Guang
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  |  
浏览/下载:10/0
  |  
提交时间:2020/07/01
Bioactive polyoxygenated cembranoids from a novel Hainan chemotype of the soft coral Sinularia flexibilis
期刊论文
Bioorganic & medicinal chemistry letters, 2019, 卷号: 29, 期号: 2, 页码: 185-188
作者:
Wu, Qihao
;
Li, Xu-Wen
;
Li, Heng
;
Yao, Li-Gong
;
Tang, Wei
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  |  
浏览/下载:70/0
  |  
提交时间:2019/01/08
Discovery and synthesis of 6,7,8,9-tetrahydro-5H-pyrido[4,3-c]azepin-5-one-based novel chemotype CCR2 antagonists via scaffold hopping strategy
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 12, 页码: 3559-3572
作者:
Qin, Li-Huai
;
Wang, Zhi-Long
;
Xie, Xin
;
Long, Ya-Qiu
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2019/01/08
6,7,8,9-Tetrahydro-5H-pyrido[43-c]azepin-5-one
3,4-Dihydro-2,6-naphthyridin-1(2H)-one
CCR2 antagonist
Scaffold hopping
Structure-activity relationship
Selectivity of CCR2 over CCR5
Acid-Promoted D-A-D Type Far-Red Fluorescent Probe with High Photostability for Lysosomal Nitric Oxide Imaging
期刊论文
ANALYTICAL CHEMISTRY, 2018, 卷号: 90, 期号: 13, 页码: 7953-7962
作者:
Wang, Fengyang
;
Yu, Shujuan
;
Xu, Zhiai
;
Li, Lingling
;
Dang, Yijing
收藏
  |  
浏览/下载:53/0
  |  
提交时间:2019/01/08
Genotypic and Environmental Effects on the Volatile Chemotype of Valeriana jatamansi Jones
期刊论文
FRONTIERS IN PLANT SCIENCE, 2018, 卷号: 9
作者:
He, Xingchao
;
Wang, Shiyu
;
Shi, Jiayi
;
Sun, Zhonglin
;
Lei, Zhentian
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2019/12/05
Valerianae Jatamansi Rhizoma et Radix
Valeriana jatamansi
genotype
chemotype
volatile profile
wild population
common-garden sample
Discovery of Potent and Orally Bioavailable GPR40 Full Agonists Bearing Thiophen-2-ylpropanoic Acid Scaffold
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 7, 页码: 2697-2717
作者:
Li, He
;
Huang, Qi
;
Chen, Cheng
;
Xu, Bin
;
Wang, He-Yao
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08
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