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上海药物研究所 [20]
厦门大学 [9]
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期刊论文 [74]
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浏览/检索结果:
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JC-010a, a novel selective SHP2 allosteric inhibitor, overcomes RTK/non-RTK-mediated drug resistance in multiple oncogene-addicted cancers
期刊论文
CANCER LETTERS, 2024, 卷号: 582, 页码: 15
作者:
Lu, Xuxiu
;
Yu, Rilei
;
Li, Zhen
;
Yang, Mengke
;
Dai, Jiajia
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2024/04/07
Acquired resistance
Cancer
NSCLC
JC-010a
SHP2
Hepatoprotective Mechanism and Material Basis of Swertia Plants Based On Network Pharmacology and Molecular Docking Method
期刊论文
LATIN AMERICAN JOURNAL OF PHARMACY, 2023, 卷号: 42, 期号: 2, 页码: 374
作者:
Huang, Xian-Ju
;
Liu, Shi-Quan
;
Dai, Jia-Wei
;
LI, Tian-Cai
;
Wu, Zhou-Yang
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2023/12/01
Anti-Inflammatory Functions of Methanol Extract from Malus baccata (L.) Borkh. Leaves and Shoots by Targeting the NF-κB Pathway
期刊论文
PLANTS-BASEL, 2022, 卷号: 11, 期号: 5
作者:
Song, Chaoran
;
Chen, Hongxi
;
Kim, Soo Ah
;
Lee, Jong Sub
;
Choung, Eui Su
收藏
  |  
浏览/下载:0/0
  |  
提交时间:2024/03/07
Malus baccata (L.) Borkh.
anti-inflammatory
NF-kappa B
Synthesis and biological evaluation of 2,5-diaryl-1,3,4-oxadiazole derivatives as novel Src homology 2 domain-containing protein tyrosine phosphatase 2 (SHP2) inhibitors
期刊论文
BIOORGANIC CHEMISTRY, 2021, 卷号: 116, 页码: 13
作者:
Meng, Xiang-Dong
;
Gao, Li-Xin
;
Wang, Zhi-Jia
;
Feng, Bo
;
Zhang, Chun
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2021/12/01
2,5-diphenyl-1,3,4-oxadiazole derivatives
SHP2
Inhibitors
Structure-activity relationships (SAR)
MD2 blockage prevents the migration and invasion of hepatocellular carcinoma cells via inhibition of the EGFR signaling pathway
期刊论文
JOURNAL OF GASTROINTESTINAL ONCOLOGY, 2021
作者:
Qi, Yajun
;
Fang, Qilu
;
Li, Qinglin
;
Ding, Haiying
;
Shu, Qi
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2021/09/06
Hepatocellular carcinoma (HCC)
myeloid differentiation protein 2 (MD2)
epidermal growth factor receptor (EGFR)
migration
invasion
Synthesis and biological evaluation of heterocyclic bis-aryl amides as novel Src homology 2 domain containing protein tyrosine phosphatase-2 (SHP2) inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 11, 页码: 5
作者:
Satheeshkumar, Rajendran
;
Zhu, Rui
;
Feng, Bo
;
Huang, Chao
;
Gao, Ya
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2020/07/01
Heterocyclic bis-aryl amides
PTP1B
SHP2
Inhibitors
Structure-activity relationships (SAR)
Endosulfan promotes cell migration via PTP4A3-mediated signaling pathways in HUVECs
期刊论文
ECOTOXICOLOGY AND ENVIRONMENTAL SAFETY, 2020, 卷号: 192, 页码: 1-9
作者:
Li, Heng
;
Liu, Shiqi
;
Hu, Yumeng
;
Zhao, Bin
;
Sun, Yeqing
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2021/09/14
Endosulfan
Cell migration
PTP4A3
Signaling pathway
Endothelial cells
Quantitative proteomic and phosphoproteomic studies reveal novel 5-fluorouracil resistant targets in hepatocellular carcinoma
期刊论文
JOURNAL OF PROTEOMICS, 2019, 卷号: 208, 页码: 10
作者:
Liu, Zhen
;
Wang, Yan
;
Yao, Yating
;
Fang, Zheng
;
Miao, Qing R.
收藏
  |  
浏览/下载:92/0
  |  
提交时间:2019/12/02
Hepatocellular carcinoma
5-Fu resistance
LC-MS/MS
GnRH signaling pathway
Blocking ROR1 enhances the roles of erlotinib in lung adenocarcinoma cell lines
期刊论文
ONCOLOGY LETTERS, 2019, 卷号: 18, 期号: 3, 页码: 2977-2984
作者:
Wang, Hui-Li
;
Liu, Yan-Chun
;
Long, Ming-Peng
;
Zheng, Chuan
;
Yang, Jia-Hui
收藏
  |  
浏览/下载:96/0
  |  
提交时间:2019/11/07
receptor tyrosine kinase-like orphan receptor 1
lung adenocarcinoma
erlotinib resistance
AKT
mammalian target of rapamycin
small interfering RNA
Mechanical features of endothelium regulate cell adhesive molecule-induced calcium response in neutrophils
期刊论文
APL BIOENGINEERING, 1, 2019, 卷号: 3, 页码: 16104
作者:
Xu YH(徐艳红)
;
Huang DD(黄丹丹)
;
Lv SQ(吕守芹)
;
Zhang Y(章燕)
;
Long M(龙勉)
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2022/10/25
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