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Discovery of 5-Benzylidene-2-phenyl-1,3-dioxane-4,6-diones as Highly Potent and Selective SIRT1 Inhibitors 期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2021, 卷号: 12, 期号: 3, 页码: 397-403
作者:  Li, Chunpu;  Hu, Sha-Sha;  Yang, Lisheng;  Wang, Min;  Long, Jian-Dong
收藏  |  浏览/下载:57/0  |  提交时间:2021/05/24
S100A11 Promotes Liver Steatosis via FOXO1-Mediated Autophagy and Lipogenesis 期刊论文
CELLULAR AND MOLECULAR GASTROENTEROLOGY AND HEPATOLOGY, 2021, 卷号: 11, 期号: 3, 页码: 697-724
作者:  Zhang, Linqiang;  Zhang, Zhiguo;  Li, Chengbin;  Zhu, Tingting;  Gao, Jing
收藏  |  浏览/下载:48/0  |  提交时间:2021/05/24
Design, Synthesis, and Biological Evaluation of 8-Mercapto-3,7-Dihydro-1H-Purine-2,6-Diones as Potent Inhibitors of SIRT1, SIRT2, SIRT3, and SIRT5 期刊论文
MOLECULES, 2020, 卷号: 25, 期号: 12, 页码: 18
作者:  Han, Haozhen;  Li, Chunpu;  Li, Man;  Yang, Lisheng;  Zhao, Sen
收藏  |  浏览/下载:36/0  |  提交时间:2020/12/24
Structural Insight into the Interactions between Structurally Similar Inhibitors and SIRT6 期刊论文
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2020, 卷号: 21, 期号: 7, 页码: 15
作者:  Zhao, Shuang;  Zhu, Yan-Yan;  Wang, Xiao-Yu;  Liu, Yong-Sheng;  Sun, Yun-Xiang
收藏  |  浏览/下载:30/0  |  提交时间:2020/07/01
Celastrol Protects From Cholestatic Liver Injury Through Modulation of SIRT1-FXR Signaling 期刊论文
MOLECULAR & CELLULAR PROTEOMICS, 2019, 卷号: 18, 期号: 3, 页码: 520-533
作者:  Zhao, Qi;  Liu, Fang;  Cheng, Yan;  Xiao, Xue-Rong;  Hu, Dan-Dan
收藏  |  浏览/下载:57/0  |  提交时间:2019/07/29
Cyclic tripeptide-based potent human SIRT7 inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 3, 页码: 461-465
作者:  Li, Shengchao[1];  Wu, Bo[2];  Zheng, Weiping[3]
收藏  |  浏览/下载:5/0  |  提交时间:2019/12/24
The mimics of N-epsilon-acyl-lysine derived from cysteine as sirtuin inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2018, 卷号: 28, 期号: 14, 页码: 2375-2378
作者:  Wang, Chun;  Wang, Fang;  Chen, Xiaoxue;  Zou, Yefang;  Zhu, Hong
收藏  |  浏览/下载:22/0  |  提交时间:2019/01/08
Discovery and anti-inflammatory evaluation of benzothiazepinones (BTZs) as novel non-ATP competitive inhibitors of glycogen synthase kinase-3 beta (GSK-3 beta) 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 20
作者:  Gao, Yang;  Zhang, Peng;  Cui, Anfeng;  Ye, De-Yong;  Xiang, Meng
收藏  |  浏览/下载:6/0  |  提交时间:2019/12/05
X-ray crystal structure guided discovery of new selective, substrate-mimicking sirtuin 2 inhibitors that exhibit activities against non-small cell lung cancer cells 期刊论文
European Journal of Medicinal Chemistry, 2018
作者:  Ling-Ling Yang;  Hua-Li Wang;  Lei Zhong;  Chen Yuan;  Si-Yu Liu
收藏  |  浏览/下载:5/0  |  提交时间:2019/02/25
Bivalent SIRT1 inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 27, 期号: 2, 页码: 180-186
作者:  Wang, Juan[1];  Zang, Wenwen[2];  Liu, Jiajia[3];  Zheng, Weiping[4]
收藏  |  浏览/下载:8/0  |  提交时间:2019/12/24


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