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上海药物研究所 [14]
厦门大学 [4]
东北农业大学 [3]
大连化学物理研究所 [2]
四川大学 [2]
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期刊论文 [36]
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Synthesis of the analogs of plocabulin and their preliminary structure-activity relationship study
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2021, 卷号: 51, 页码: 5
作者:
Wang, Leiming
;
Li, Xin
;
Cui, Hong
;
Lei, Xinsheng
;
Liu, Hongchun
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2021/12/01
Marine nature products
Plocabulin
PM060184
Synthesis
Antiproliferation
A validated HPLC-MS/MS method for determination of simmitecan and its metabolite chimmitecan in human plasma and its application to a pharmacokinetic study in Chinese patients with advanced solid tumor
期刊论文
JOURNAL OF SEPARATION SCIENCE, 2021, 页码: 8
作者:
Zhou, Jun
;
Zhan, Yan
;
Zhong, Dafang
;
Chen, Xiaoyan
;
Zhang, Yifan
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  |  
浏览/下载:72/0
  |  
提交时间:2021/11/04
chimmitecan
mass spectrometry
pharmacokinetics
simmitecan
solid tumors
Hyperprins A and B, Two Complex Meroterpenoids from Hypericum przewalskii
期刊论文
ORGANIC LETTERS, 2020, 卷号: 22, 期号: 7, 页码: 2797-2800
作者:
Zong, Jian-Fa
;
Hu, Zhu
;
Shao, Ying-Ying
;
Shi, Qing
;
Zhang, Meng-Meng
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  |  
浏览/下载:27/0
  |  
提交时间:2020/07/01
Design, Synthesis and Antiproliferative Activity of Chrysin Derivatives Bearing Triazole Moieties
期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2020, 卷号: 40, 期号: 2, 页码: 440-446
作者:
Luan Tian
;
Quan Zheshan
;
Fang Yingquan
;
Yang Hongjing
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  |  
浏览/下载:36/0
  |  
提交时间:2021/02/02
INHIBITION
CELLS
chrysin
synthesis
triazole
derivatives
antiproliferation
Identification of new NIK inhibitors by discriminatory analysis-based molecular docking and biological evaluation
期刊论文
ARCHIV DER PHARMAZIE, 2019, 卷号: 352, 期号: 7, 页码: 9
作者:
Cheng, Gang
;
Mei, Xiao-Bing
;
Yan, You-You
;
Chen, Jing
;
Zhang, Bo
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  |  
浏览/下载:9/0
  |  
提交时间:2020/07/01
antiproliferation activity
inhibitors
NF-kappa B inducing kinase
virtual screen
Cytotoxic Trichothecene Macrolides Produced by the Endophytic Myrothecium roridum
期刊论文
JOURNAL OF NATURAL PRODUCTS, 2019, 卷号: 82, 期号: 6, 页码: 1503-1509
作者:
Shen, Li
;
Ai, Chun-Zhi
;
Song, Yong-Chun
;
Wang, Feng-Wu
;
Jiao, Rui-Hua
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  |  
浏览/下载:61/0
  |  
提交时间:2019/12/02
Discovery of Novel PRMT5 Inhibitors by Virtual Screening and Biological Evaluations
期刊论文
CHEMICAL & PHARMACEUTICAL BULLETIN, 2019, 卷号: 67, 期号: 4, 页码: 382-388
作者:
Tao, Hongrui
;
Yan, Xue
;
Zhu, Kongkai
;
Zhang, Hua
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  |  
浏览/下载:14/0
  |  
提交时间:2020/07/01
virtual screening
epigenetic inhibitor
antiproliferation
molecular docking
Synthesis and biological evaluation of benzomorpholine derivatives as novel EZH2 inhibitors for anti-non-small cell lung cancer activity.
期刊论文
Molecular diversity, 2019
作者:
Feng Qiang
;
He Hualong
;
Gao Tiantao
;
Zhang Qiangsheng
;
Liu Zhihao
收藏
  |  
浏览/下载:77/0
  |  
提交时间:2019/02/25
Antiproliferation
activity
Benzomorpholine
EZH2
inhibitor
Structure–activity
relationship
Pectic oligosaccharides hydrolyzed from citrus canning processing water by Fenton reaction and their antiproliferation potentials
期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2019, 卷号: Vol.124, 页码: 1025-1032
作者:
Li, Junhui
;
Li, Shan
;
Liu, Shanshan
;
Wei, Chaoyang
;
Yan, Lufeng
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/17
Citrus canning water
Pectic polysaccharide
Depolymerisation
Anti proliferation activity
Rational design of 5-((1H-imidazol-1-yl)methyl)quinolin-8-ol derivatives as novel bromodomain-containing protein 4 inhibitors
期刊论文
European journal of medicinal chemistry, 2018, 卷号: 163, 页码: 281-294
作者:
Xing, Jing
;
Zhang, Rukang
;
Jiang, Xiangrui
;
Hu, Tianwen
;
Wang, Xinjun
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  |  
浏览/下载:86/0
  |  
提交时间:2019/01/08
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