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Inhibition of Autophagy by a Small Molecule through Covalent Modification of the LC3 Protein 期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2021, 页码: 11
作者:  Fan, Shijie;  Yue, Liyan;  Wan, Wei;  Zhang, Yuanyuan;  Zhang, Bidong
收藏  |  浏览/下载:80/0  |  提交时间:2021/12/16
Dynamics of Post-Translational Modification Inspires Drug Design in the Kinase Family 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 20, 页码: 15111-15125
作者:  Zhang, Huimin;  He, Jixiao;  Hu, Guang;  Zhu, Fei;  Jiang, Hao
收藏  |  浏览/下载:36/0  |  提交时间:2022/01/04
Drug target inference by mining transcriptional data using a novel graph convolutional network framework 期刊论文
PROTEIN & CELL, 2021, 页码: 21
作者:  Zhong, Feisheng;  Wu, Xiaolong;  Yang, Ruirui;  Li, Xutong;  Wang, Dingyan
收藏  |  浏览/下载:22/0  |  提交时间:2021/12/01
Introducing the authors 期刊论文
CELL METABOLISM, 2021, 卷号: 33, 期号: 10, 页码: 1896-1900
作者:  Li, Jingya;  Jiang, Hui;  Li, Hongliang;  Jiang, Changtao;  Liu, Junli
收藏  |  浏览/下载:16/0  |  提交时间:2022/01/18
Discovery of a subtype-selective, covalent inhibitor against palmitoylation pocket of TEAD3 期刊论文
ACTA PHARMACEUTICA SINICA B, 2021, 卷号: 11, 期号: 10, 页码: 3206-3219
作者:  Lu, Tian;  Li, Yong;  Lu, Wenchao;  Spitters, Twgm;  Fang, Xueyu
收藏  |  浏览/下载:41/0  |  提交时间:2021/12/01
A hybrid framework for improving uncertainty quantification in deep learning-based QSAR regression modeling 期刊论文
JOURNAL OF CHEMINFORMATICS, 2021, 卷号: 13, 期号: 1, 页码: 17
作者:  Wang, Dingyan;  Yu, Jie;  Chen, Lifan;  Li, Xutong;  Jiang, Hualiang
收藏  |  浏览/下载:60/0  |  提交时间:2021/11/04
Discovery of High-Affinity Inhibitors of the BPTF Bromodomain 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 16, 页码: 12075-12088
作者:  Lu, Tian;  Lu, Haibo;  Duan, Zhe;  Wang, Jun;  Han, Jie
收藏  |  浏览/下载:38/0  |  提交时间:2021/11/04
Facing small and biased data dilemma in drug discovery with enhanced federated learning approaches 期刊论文
SCIENCE CHINA-LIFE SCIENCES, 2021, 页码: 11
作者:  Xiong, Zhaoping;  Cheng, Ziqiang;  Lin, Xinyuan;  Xu, Chi;  Liu, Xiaohong
收藏  |  浏览/下载:46/0  |  提交时间:2021/11/04
Intestinal MYC modulates obesity-related metabolic dysfunction 期刊论文
NATURE METABOLISM, 2021, 页码: 37
作者:  Luo, Yuhong;  Yang, Shoumei
收藏  |  浏览/下载:30/0  |  提交时间:2021/08/17
Structure-Guided Development of Small-Molecule PRC2 Inhibitors Targeting EZH2-EED Interaction 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 12, 页码: 8194-8207
作者:  Du, Daohai;  Xu, Dandan;  Zhu, Licheng;  Stazi, Giulia;  Zwergel, Clemens
收藏  |  浏览/下载:74/0  |  提交时间:2021/08/17


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