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广州生物医药与健康研... [8]
海洋研究所 [2]
南海海洋研究所 [1]
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期刊论文 [11]
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2016 [4]
2013 [7]
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Pharmacol... [11]
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浏览/检索结果:
共11条,第1-10条
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学科主题:Pharmacology & Pharmacy
内容类型:期刊论文
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Structure-Based Design of Potent Nicotinamide Phosphoribosyltransferase Inhibitors with Promising in Vitro and in Vivo Antitumor Activities
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5766-5779
作者:
Jiang, Sheng
;
Li, Zheng
;
Qin, Dongguang
;
Qiu, Yatao
;
Chen, Jiaxuan
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2018/12/13
Design, Synthesis, and Biological Evaluation of Substituted Pyrimidines as Potential Phosphatidylinositol 3-Kinase (PI3K) Inhibitors
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 15, 页码: 7268-7274
作者:
Long, Zi-Jie
;
Lai, Xiao-Ju
;
Chen, Hui-Xuan
;
Luo, Yu
;
Weng, Jiang
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2018/12/13
Structure-Based Design of Potent Nicotinamide Phosphoribosyltransferase Inhibitors with Promising in Vitro and in Vivo Antitumor Activities
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5766-5779
Bai, Jinhong
;
Liao, Chenzhong
;
Liu, Yanghan
;
Qin, Xiaochu
;
Chen, Jiaxuan
;
Qiu, Yatao
;
Qin, Dongguang
;
Li, Zheng
;
Tu, Zheng-Chao
;
Jiang, Sheng
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2016/12/16
Design, Synthesis, and Biological Evaluation of Substituted Pyrimidines as Potential Phosphatidylinositol 3-Kinase (PI3K) Inhibitors
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 15, 页码: 7268-7274
Zhang, Ji-Quan
;
Luo, Yong-Jie
;
Xiong, Yan-Shi
;
Yu, Yang
;
Tu, Zheng-Chao
;
Long, Zi-Jie
;
Lai, Xiao-Ju
;
Chen, Hui-Xuan
;
Luo, Yu
;
Weng, Jiang
;
Lu, Gui
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2016/12/16
Discovery of novel bromophenol 3,4-dibromo-5-(2-bromo-3,4-dihydroxy-6-(isobutoxymethyl)benzyl)benzene-1,2-diol as protein tyrosine phosphatase 1B inhibitor and its anti-diabetic properties in C57BL/KsJ-db/db mice
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 64, 页码: 129-136
作者:
Jiang, Bo
;
Guo, Shuju
;
Shi, Dayong
;
Guo, Chao
;
Wang, Tao
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2014/07/17
Type 2 diabetes mellitus
Protein tyrosine phosphatase 1B
Bromophenol
Anti-diabetic activities
HPN, a Synthetic Analogue of Bromophenol from Red Alga Rhodomela confervoides: Synthesis and Anti-Diabetic Effects in C57BL/KsJ-db/db Mice
期刊论文
MARINE DRUGS, 2013, 卷号: 11, 期号: 2, 页码: 350-362
作者:
Shi, Dayong
;
Guo, Shuju
;
Jiang, Bo
;
Guo, Chao
;
Wang, Tao
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2014/07/17
bromophenol
protein tyrosine phosphatase 1B inhibitor
db/db mouse model
anti-diabetes properties
Alkaloids from the Deep-Sea-Derived Fungus Aspergillus westerdijkiae DFFSCS013
期刊论文
JOURNAL OF NATURAL PRODUCTS, 2013, 卷号: 76, 期号: 5
Peng, Jiang
;
Zhang, Xiao-Yong
;
Tu, Zheng-Chao
;
Xu, Xin-Ya
;
Qi, Shu-Hua
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2016/12/16
Alkaloids from the Deep-Sea-Derived Fungus Aspergillus westerdijkiae DFFSCS013
期刊论文
JOURNAL OF NATURAL PRODUCTS, 2013, 卷号: 76, 期号: 5, 页码: 983-987
[Peng, Jiang
;
Zhang, Xiao-Yong
;
Xu, Xin-Ya
;
Qi, Shu-Hua] Chinese Acad Sci, Guangdong Key Lab Marine Mat Med, Key Lab Marine Bioresources Sustainable Utilizat, South China Sea Inst Oceanol,RNAM Ctr Marine Micr, Guangzhou 510301, Guangdong, Peoples R China
;
[Peng, Jiang] Univ Chinese Acad Sci, Chinese Acad Sci, Grad Sch, Beijing 100049, Peoples R China
;
[Tu, Zheng-Chao] Chinese Acad Sci, Guangzhou Inst Biomed & Hlth, Guangzhou 510530, Guangdong, Peoples R China
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2015/01/22
Discovery of potent dipeptidyl peptidase IV inhibitors through pharmacophore hybridization and hit-to-lead optimization
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2013, 卷号: 21, 期号: 7
作者:
Hu, Wenhui
;
Zeng, Shaogao
;
Xie, Hui
;
Zeng, Li-li
;
Lu, Xin
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2018/12/13
Alkaloids from the Deep-Sea-Derived Fungus Aspergillus westerdijkiae DFFSCS013
期刊论文
JOURNAL OF NATURAL PRODUCTS, 2013, 卷号: 76, 期号: 5
作者:
Peng, Jiang
;
Zhang, Xiao-Yong
;
Tu, Zheng-Chao
;
Xu, Xin-Ya
;
Qi, Shu-Hua
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2018/12/13
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