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Bufalin exerts antitumor effects in neuroblastoma via the induction of reactive oxygen species-mediated apoptosis by targeting the electron transport chain 期刊论文
INTERNATIONAL JOURNAL OF MOLECULAR MEDICINE, 2020, 卷号: 46, 期号: 6, 页码: 2137-2149
作者:  Pan, Lijia;  Nie, Litong;  Yao, Sheng;  Bi, Aiwei;  Ye, Yang
收藏  |  浏览/下载:26/0  |  提交时间:2020/12/24
cudc907displayspotentantitumoractivityagainsthumanpancreaticadenocarcinomainvitroandinvivothroughinhibitionofhdac6todownregulatecmycexpression 期刊论文
actapharmacologicasinica, 2019, 卷号: 40, 期号: 5, 页码: 677
作者:  Fu Xuhong;  Zhang Xiong;  Yang Hong;  Xu Xiaowei;  Hu Zonglong
收藏  |  浏览/下载:48/0  |  提交时间:2020/07/01
CUDC-907 displays potent antitumor activity against human pancreatic adenocarcinoma in vitro and in vivo through inhibition of HDAC6 to downregulate c-Myc expression 期刊论文
Acta pharmacologica Sinica, 2018
作者:  Fu, Xu-Hong;  Zhang, Xiong;  Yang, Hong;  Xu, Xiao-Wei;  Hu, Zong-Long
收藏  |  浏览/下载:27/0  |  提交时间:2019/01/08
SOMCL-085, a novel multi-targeted FGFR inhibitor, displays potent anticancer activity in FGFR-addicted human cancer models 期刊论文
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 2, 页码: 243-250
作者:  Jiang, Xi-fei;  Dai, Yang;  Peng, Xia;  Shen, Yan-yan;  Su, Yi
收藏  |  浏览/下载:53/0  |  提交时间:2019/01/08
15, 16-Dihydrotanshinone I Inhibits Hemangiomas through Inducing Pro-apoptotic and Anti-angiogenic Mechanisms in Vitro and in Vivo 期刊论文
FRONTIERS IN PHARMACOLOGY, 2018, 卷号: 9
作者:  Cai, Yihong;  Lv, Fan;  Kaldybayeva, Nurshat;  Zhamilya, Abilova;  Wu, Zhixiang
收藏  |  浏览/下载:40/0  |  提交时间:2019/01/08
somcl085anovelmultitargetedfgfrinhibitordisplayspotentanticanceractivityinfgfraddictedhumancancermodels 期刊论文
actapharmacologicasinica, 2018, 卷号: 39, 期号: 2, 页码: 243
作者:  Jiang Xifei;  Dai Yang;  Peng Xia;  Shen Yanyan;  Su Yi
收藏  |  浏览/下载:3/0  |  提交时间:2020/07/01
HER2-targeted antibody drug conjugates for ovarian cancer therapy 期刊论文
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2016, 卷号: 93, 页码: 274-286
作者:  Jiang, Jing;  Dong, Lihou;  Wang, Lei;  Wang, Ling;  Zhang, Jing
收藏  |  浏览/下载:52/0  |  提交时间:2019/01/08
Yhhu3813 is a novel selective inhibitor of c-Met kinase that inhibits c-Met-dependent neoplastic phenotypes of human cancer cells 期刊论文
ACTA PHARMACOLOGICA SINICA, 2014, 卷号: 35, 期号: 1, 页码: 89-97
作者:  He, Chang-xi;  Ai, Jing;  Xing, Wei-qiang;  Chen, Yi;  Zhang, Hao-tian
收藏  |  浏览/下载:35/0  |  提交时间:2019/01/08
Design, Synthesis, and Biological Evaluation of Novel Conformationally Constrained Inhibitors Targeting Epidermal Growth Factor Receptor Threonine(790) -> Methionine(790) Mutant 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2012, 卷号: 55, 期号: 6, 页码: 2711-2723
作者:  Chang, Shaohua;  Zhang, Lianwen;  Xu, Shilin;  Luo, Jinfeng;  Lu, Xiaoyun
收藏  |  浏览/下载:18/0  |  提交时间:2019/01/08
Combined Src and Aromatase Inhibition Impairs Human Breast Cancer Growth In vivo and Bypass Pathways Are Activated in AZD0530-Resistant Tumors 期刊论文
CLINICAL CANCER RESEARCH, 2009, 卷号: 15, 期号: 10, 页码: 3396-3405
作者:  Chen, Yi;  Guggisberg, Natalia;  Jorda, Merce;  Gonzalez-Angulo, Ana;  Hennessy, Bryan
收藏  |  浏览/下载:14/0  |  提交时间:2019/01/08


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