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Crowdsourced identification of multi-target kinase inhibitors for RET- and TAU- based disease: The Multi-Targeting Drug DREAM Challenge 期刊论文
PLOS COMPUTATIONAL BIOLOGY, 2021, 卷号: 17, 期号: 9, 页码: 19
作者:  Xiong, Zhaoping;  Jeon, Minji;  Allaway, Robert J.;  Kang, Jaewoo;  Park, Donghyeon
收藏  |  浏览/下载:22/0  |  提交时间:2021/11/04
Polyoxypregnanes as safe, potent, and specific ABCB1-inhibitory pro-drugs to overcome multidrug resistance in cancer chemotherapy in vitro and in vivo 期刊论文
ACTA PHARMACEUTICA SINICA B, 2021, 卷号: 11, 期号: 7, 页码: 1885-1902
作者:  Wu, Xu;  Yin, Chun;  Ma, Jiang;  Chai, Stella;  Zhang, Chunyuan
收藏  |  浏览/下载:39/0  |  提交时间:2021/11/04
Dual Mechanisms of Novel CD73-Targeted Antibody and Antibody-Drug Conjugate in Inhibiting Lung Tumor Growth and Promoting Antitumor Immune-Effector Function 期刊论文
MOLECULAR CANCER THERAPEUTICS, 2020, 卷号: 19, 期号: 11, 页码: 2340-2352
作者:  Jin, Rui;  Liu, Liang;  Xing, Yun;  Meng, Tao;  Ma, Lanping
收藏  |  浏览/下载:51/0  |  提交时间:2020/12/24
Smart Nanosized Drug Delivery Systems Inducing Immunogenic Cell Death for Combination with Cancer Immunotherapy 期刊论文
ACCOUNTS OF CHEMICAL RESEARCH, 2020, 卷号: 53, 期号: 9, 页码: 1761-1772
作者:  Zhou, Lei;  Zhang, Pengcheng;  Wang, Hao;  Wang, Dangge;  Li, Yaping
收藏  |  浏览/下载:15/0  |  提交时间:2020/12/21
DGAT1 inhibitors protect pancreatic beta-cells from palmitic acid-induced apoptosis 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 8
作者:  Huang, Jun-shang;  Guo, Bin-bin;  Wang, Gai-hong;  Zeng, Li-min;  Hu, You-hong
收藏  |  浏览/下载:57/0  |  提交时间:2020/12/24
YES1amplification confers trastuzumab-emtansine (T-DM1) resistance in HER2-positive cancer 期刊论文
BRITISH JOURNAL OF CANCER, 2020, 页码: 12
作者:  Wang, Lei;  Wang, Quanren;  Xu, Piaopiao;  Fu, Li;  Li, Yun
收藏  |  浏览/下载:16/0  |  提交时间:2020/12/24
A novel M phase blocker, DCZ3301 enhances the sensitivity of bortezomib in resistant multiple myeloma through DNA damage and mitotic catastrophe 期刊论文
Journal of Experimental & Clinical Cancer Research, 2020, 卷号: 39, 期号: 1
作者:  Hu,Liangning;  Li,Bo;  Chen,Gege;  Song,Dongliang;  Xu,Zhijian
收藏  |  浏览/下载:94/0  |  提交时间:2020/07/01
A novel phosphoramide compound, DCZ0847, displays in vitro and in vivo anti-myeloma activity, alone or in combination with bortezomib 期刊论文
CANCER LETTERS, 2020, 卷号: 478, 页码: 45-55
作者:  Chen, Gege;  Hu, Ke;  Sun, Haiguo;  Zhou, Jinfeng;  Song, Dongliang
收藏  |  浏览/下载:97/0  |  提交时间:2020/07/01
Identification of catalytic and non-catalytic activity inhibitors against PRC2-EZH2 complex through multiple high-throughput screening campaigns 期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2020, 页码: 27
作者:  Zhou, Yan;  Du, Dao-Hai;  Wang, Jia;  Cai, Xiao-Qing;  Deng, Alicia X.
收藏  |  浏览/下载:103/0  |  提交时间:2020/07/01
Stepwise targeting and responsive lipid-coated nanoparticles for enhanced tumor cell sensitivity and hepatocellular carcinoma therapy 期刊论文
THERANOSTICS, 2020, 卷号: 10, 期号: 8, 页码: 3722-3736
作者:  Li, Ying;  Miao, Yunqiu;  Chen, Mingshu;  Chen, Xi;  Li, Feifei
收藏  |  浏览/下载:29/0  |  提交时间:2020/07/01


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