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Inhibition of PTP1B blocks pancreatic cancer progression by targeting the PKM2/AMPK/mTOC1 pathway 期刊论文
CELL DEATH & DISEASE, 2019, 卷号: 10, 页码: 15
作者:  Xu, Qi;  Wu, Ning;  Li, Xiangqian;  Guo, Chuanlong;  Li, Chao
收藏  |  浏览/下载:25/0  |  提交时间:2020/03/20
Synthesis and PTP1B/TCPTP Inhibitory Activity Evaluation of Novel 2,5-Disubstituted-1,3,4-thiadiazolamide Derivatives Containing Carbazole/Benzimidazole Moity 期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2019, 卷号: 39, 期号: 9, 页码: 2599-2608
作者:  Li Yingjun;  Zhao Yue;  Jin Kun;  Gao Lixin;  Sheng Li
收藏  |  浏览/下载:34/0  |  提交时间:2020/07/01
Frondoplysins A and B, Unprecedented Terpene-Alkaloid Bioconjugates from Dysidea frondosa 期刊论文
ORGANIC LETTERS, 2019, 卷号: 21, 期号: 16, 页码: 6190-6193
作者:  Jiao, Wei-Hua;  Li, Jing;  Zhang, Meng-Meng;  Cui, Jie;  Gui, Yu-Han
收藏  |  浏览/下载:2/0  |  提交时间:2020/07/01
Synthesis and biological evaluation of tryptophan-derived rhodanine derivatives as PTP1B inhibitors and anti-bacterial agents 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 172, 页码: 163-173
作者:  Liu, Hongyan;  Sun, Danwen;  Du, Hang;  Zheng, Changji;  Li, Jingya
收藏  |  浏览/下载:13/0  |  提交时间:2020/07/01
Discovery of 1,3-diphenyl-1H-pyrazole derivatives containing rhodanine-3-alkanoic acid groups as potential PTP1B inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 10, 页码: 1187-1193
作者:  Sun, Liangpeng;  Wang, Peipei;  Xu, Lili;  Gao, Lixin;  Li, Jia
收藏  |  浏览/下载:4/0  |  提交时间:2020/07/01
Highly Selective Protein Tyrosine Phosphatase Inhibitor, 2,2 ',3,3 '-Tetrabromo-4,4 ',5,5 '-tetrahydroxydiphenylmethane, Ameliorates Type 2 Diabetes Mellitus in BKS db Mice 期刊论文
MOLECULAR PHARMACEUTICS, 2019, 卷号: 16, 期号: 5, 页码: 1839-1850
作者:  Li, Chao;  Luo, Jiao;  Guo, Shuju;  Jia, Xiaoling;  Guo, Chuanlong
收藏  |  浏览/下载:73/0  |  提交时间:2019/08/28
Synthesis and PTP1B Inhibitory Activity of Novel Chalcone Derivatives Bearing 1H-Benzo[d]imidazol or 1H-Benzo[d][1,2,3]triazol Moieties 期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2019, 卷号: 39, 期号: 4, 页码: 1029-1036
作者:  Fu Yang;  Sheng Li;  Gao Lixin;  Li Jia;  Sun Liangpeng
收藏  |  浏览/下载:3/0  |  提交时间:2020/07/01
Toward a treatment of diabesity: In vitro and in vivo evaluation of uncharged bromophenol derivatives as a new series of PTP1B inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 166, 页码: 178-185
作者:  Li, Xiangqian;  Xu, Qi;  Li, Chao;  Luo, Jiao;  Li, Xiuxue
收藏  |  浏览/下载:59/0  |  提交时间:2019/05/15


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