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Design, synthesis and biological evaluation of uncharged catechol derivatives as selective inhibitors of PTP1B 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 136, 页码: 348-359
作者:  Li, Xiang-Qian;  Xu, Qi;  Luo, Jiao;  Wang, Li-Jun;  Jiang, Bo
收藏  |  浏览/下载:24/0  |  提交时间:2017/10/09
A Novel Sarsolenane Diterpene as a PTP1B Inhibitor from Hainan Soft Coral Sarcophyton trocheliophorum Marenzeller 期刊论文
CHINESE JOURNAL OF CHEMISTRY, 2017, 卷号: 35, 期号: 8, 页码: 1246-1250
作者:  Liang, Linfu;  Wang, Jinan;  Shi, Xiaoxuan;  Zhu, Yinghua;  Li, Jia
收藏  |  浏览/下载:23/0  |  提交时间:2019/01/08
Discovery and evaluation of the hybrid of bromophenol and saccharide as potent and selective protein tyrosine phosphatase 1B inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 134, 页码: 24-33
作者:  Zhang, Renshuai;  Yu, Rilei;  Xu, Qi;  Li, Xiangqian;  Luo, Jiao
收藏  |  浏览/下载:22/0  |  提交时间:2017/07/10
5-Alkylpyrrole-2-carboxaldehyde derivatives from the Chinese sponge Mycale lissochela and their PTP1B inhibitory activities 期刊论文
CHINESE CHEMICAL LETTERS, 2017, 卷号: 28, 期号: 6, 页码: 1190-1193
作者:  Xue, Duo-Qing;  Liu, Hai-Li;  Chen, Si-Han;  Mollo, Ernesto;  Gavagnin, Margherita
收藏  |  浏览/下载:25/0  |  提交时间:2019/01/08
Aglaiabbrevins A-D, New Prenylated Bibenzyls from the Leaves of Aglaia abbreviata with Potent PTP1B Inhibitory Activity 期刊论文
CHEMICAL & PHARMACEUTICAL BULLETIN, 2017, 卷号: 65, 期号: 3, 页码: 295-299
作者:  Sun, Pan;  Jiang, Chang-Sheng;  Zhang, Yi;  Liu, Ai -Hong;  Liang, Tong -Jun
收藏  |  浏览/下载:16/0  |  提交时间:2019/01/08
Synthesis, crystal structure and ptps inhibition of a zinc(ii) complex with n-(4-hydroxybenzyl)-l-serine 期刊论文
Chinese journal of structural chemistry, 2017, 卷号: 36, 期号: 2, 页码: 316-323
作者:  Li Yan-Hong;  Lu Li-Ping;  Zhu Miao-Li;  Yuan Cai-Xia;  Feng Si-Si
收藏  |  浏览/下载:45/0  |  提交时间:2019/04/23
Discovery of core-structurally novel PTP1B inhibitors with specific selectivity containing oxindole-fused spirotetrahydrofurochroman by one-pot reaction 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 27, 期号: 4, 页码: 1105-1108
作者:  Dong, Suzhen;  Lei, Yubing;  Jia, Shikun;  Gao, Lixin;  Li, Jia
收藏  |  浏览/下载:22/0  |  提交时间:2019/01/08
Anti-diabetic effect of three new norditerpenoid alkaloids in vitro and potential mechanism via PI3K/Akt signaling pathway 期刊论文
BIOMEDICINE & PHARMACOTHERAPY, 2017, 卷号: 87, 期号: 3, 页码: 145-152
作者:  Tang, D (Tang, Dan);  Chen, QB (Chen, Qi-Bin);  Xin, XL (Xin, Xue-Lei);  Aisa, HA (Aisa, Haji-Akber)
收藏  |  浏览/下载:16/0  |  提交时间:2017/04/05
Synthesis, Crystal Structure and PTPs Inhibition of a Zinc(II) Complex with N-(4-hydroxybenzyl)-L-serine 期刊论文
CHINESE JOURNAL OF STRUCTURAL CHEMISTRY结构化学, 2017, 卷号: 36, 期号: 2, 页码: 316-323
作者:  Zhu, ML;  Yuan, CX;  Feng, SS;  Gao ZQ(高增强);  Gao, ZQ
收藏  |  浏览/下载:16/0  |  提交时间:2019/08/27
Trivaric acid, a new inhibitor of PTP1b with potent beneficial effect on diabetes 期刊论文
LIFE SCIENCES, 2017, 卷号: 169, 页码: 52-64
作者:  Sun, Wenlong;  Zhang, Bowei;  Zheng, Haizhou;  Zhuang, Chunlin;  Li, Xia
收藏  |  浏览/下载:8/0  |  提交时间:2019/12/02


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