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浏览/检索结果: 共7条，第1-7条 帮助 限定条件 发表日期：2017     已选(0)清除 条数/页：5101520253035404550556065707580859095100   排序方式：请选择作者升序作者降序题名升序题名降序发表日期升序发表日期降序提交时间升序提交时间降序 Discovery of novel BET inhibitors by drug repurposing of nitroxoline and its analogues 期刊论文 ORGANIC & BIOMOLECULAR CHEMISTRY, 2017, 卷号: 15, 期号: 44, 页码: 9352-9361 作者:  Jiang, Hao;  Xing, Jing;  Wang, Chen;  Zhang, Hao;  Yue, Liyan 收藏  |  浏览/下载：108/0  |  提交时间：2019/01/08 JQ1 synergizes with the Bcl-2 inhibitor ABT-263 against MYCN-amplified small cell lung cancer 期刊论文 ONCOTARGET, 2017, 卷号: 8, 期号: 49, 页码: 86312-86324 作者:  Wang, Huogang;  Hong, Bo;  Li, Xuemin;  Deng, Ke;  Li, Hong 收藏  |  浏览/下载：25/0  |  提交时间：2018/08/17 Small Cell Lung Cancer  N-myc  Bcl-2  Jq1  Abt-263   Discovery of a series of dihydroquinoxalin-2(1H)-ones as selective BET inhibitors from a dual PLK1-BRD4 inhibitor 期刊论文 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 137, 页码: 176-195 作者:  Hu, Jianping;  Wang, Yingqing;  Li, Yanlian;  Xu, Lin;  Cao, Danyan 收藏  |  浏览/下载：32/0  |  提交时间：2019/01/08 BRD4 inhibitor  Kinase  BI-2536  Dihydroquinoxalin-2(1H)-one   Structure-Based Discovery of 4-(6-Methoxy-2-methyl-4-(quinolin-4-yl)-9H-pyrimido[4,5-b]indol-7-yl)-3,5-dimethylisoxazole (CD161) as a Potent and Orally Bioavailable BET Bromodomain Inhibitor 期刊论文 JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 9, 页码: 3887-3901 作者:  Zhao, Yujun;  Bai, Longchuan;  Liu, Liu;  McEachern, Donna;  Stuckey, Jeanne A. 收藏  |  浏览/下载：27/0  |  提交时间：2019/01/08 Discovery of novel BRD4 inhibitors by high-throughput screening, crystallography, and cell-based assays 期刊论文 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 27, 期号: 9, 页码: 2003-2009 作者:  Sun, Zhongya;  Zhang, Hao;  Chen, Zhifeng;  Xie, Yiqian;  Jiang, Hao 收藏  |  浏览/下载：89/0  |  提交时间：2019/01/08 BRD4 inhibitor  High-throughput screening  Crystallography   BET N-terminal bromodomain inhibition selectively blocks Th17 cell differentiation and ameliorates colitis in mice 期刊论文 PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2017, 卷号: 114, 期号: 11 作者:  Cheung, Kalung;  Lu, Geming;  Sharma, Rajal;  Vincek, Adam;  Zhang, Ruihua 收藏  |  浏览/下载：9/0  |  提交时间：2019/12/05 Synergistic immunostimulatory effects and therapeutic benefit of combined histone deacetylase and bromodomain inhibition in non–small cell lung cancer 期刊论文 Cancer Discovery, 2017, 卷号: 7, 期号: 8, 页码: 852-867 作者:  Adeegbe D.O.;  Liu Y.;  Lizotte P.H.;  Kamihara Y.;  Aref A.R. 收藏  |  浏览/下载：2/0  |  提交时间：2019/12/12