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Discovery and development of pyrotinib: A novel irreversible EGFR/HER2 dual tyrosine kinase inhibitor with favorable safety profiles for the treatment of breast cancer
期刊论文
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2017, 卷号: 110, 页码: 51-61
作者:
Li, Xin
;
Yang, Changyong
;
Wan, Hong
;
Zhang, Ge
;
Feng, Jun
收藏
  |  
浏览/下载:136/0
  |  
提交时间:2019/01/08
Pyrotinib
HER2-postive breast cancer
Irreversible EGFR/HER2 dual tyrosine kinase
inhibitor
Preclinical
Clinical
Safety
Drug metabolism
Multifunctionalized mesoporous silica as an efficient reversed-phase/anion exchange mixed-mode sorbent for solid-phase extraction of four acidic nonsteroidal anti-inflammatory drugs in environmental water samples
期刊论文
JOURNAL OF CHROMATOGRAPHY A, 2017, 卷号: 1527, 页码: 10-17
作者:
Li, Yun
;
Huang, Chaonan
;
Yang, Jiajia
;
Peng, Junyu
;
Jin, Jing
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  |  
浏览/下载:38/0
  |  
提交时间:2019/06/20
Multifunctionalized Mesoporous Silica
Mixed-mode Anion-exchanger
Solid Phase Extraction
Acidic Nsaids
Environmental Water Samples
Pharmacologic characterization of SHR8443, a novel dual inhibitor of phosphatidylinositol 3-kinase and mammalian target of rapamycin
期刊论文
ONCOTARGET, 2017, 卷号: 8, 期号: 64, 页码: 107977-107990
作者:
Xie, Chengying
;
Chen, Xiangling
;
Zheng, Mingyue
;
Liu, Xiaohong
;
Wang, Hongbin
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  |  
浏览/下载:27/0
  |  
提交时间:2019/01/08
BEZ235
drug resistance
mTOR
PI3K
SHR8443
The Effect of Electrical Impedance Matching on the Electromechanical Characteristics of Sandwiched Piezoelectric Ultrasonic Transducers
期刊论文
sensors, 2017, 卷号: 17, 期号: 12, 页码: 2832
作者:
Yuan Yang
;
Xiaoyuan Wei
;
Lei Zhang
;
Wenqing Yao
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  |  
浏览/下载:17/0
  |  
提交时间:2022/03/10
sandwiched piezoelectric ultrasonic transducers
effective electro-mechanical coupling coefficient
electro-acoustic power ratio
electro-acoustic gain ratio
electrical impedance matching
The structure-activity relationship between polysaccharides from Sargassum thunbergii and anti-tumor activity
期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2017, 卷号: 105, 页码: 686-692
作者:
Jin, Weihua
;
Zhang, Wenjing
;
Liu, Ge
;
Yao, Jianting
;
Shan, Tifeng
收藏
  |  
浏览/下载:51/0
  |  
提交时间:2019/07/15
Heteropolysaccharide
Anti-tumor activity
Sargassum thunbergii
Structure-activity relationship
Polysaccharides from Sargassum thunbergii: Monthly variations and anti-complement and anti-tumour activities
期刊论文
INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES, 2017, 卷号: 105, 页码: 1526-1531
作者:
Jin, Weihua
;
Liu, Ge
;
Zhong, Weihong
;
Sun, Chaomin
;
Zhang, Quanbin
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  |  
浏览/下载:24/0
  |  
提交时间:2018/01/11
Sargassum Thunbergii
Anti-complement Activities
Anti-tumour Activities
Influence of Calcareous Deposit on Corrosion Behavior of Q235 Carbon Steel with Sulfate-Reducing Bacteria
期刊论文
JOURNAL OF OCEAN UNIVERSITY OF CHINA, 2017, 卷号: 16, 期号: 6, 页码: 1213-1219
作者:
Zhang Jie
;
Li Xiaolong
;
Wang Jiangwei
;
Xu Weichen
;
Duan Jizhou
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2018/01/11
Microbiological Corrosion
Sulfate-reducing Bacteria
Calcareous Deposit
Cathodic Protection
A Simple Push-Pull Algorithm for Blue-Noise Sampling
期刊论文
IEEE TRANSACTIONS ON VISUALIZATION AND COMPUTER GRAPHICS, 2017, 卷号: 23, 期号: 12, 页码: 2496-2508
作者:
Ahmed, Abdalla G. M.
;
Guo, Jianwei
;
Yan, Dong-Ming
;
Franceschia, Jean-Yves
;
Zhang, Xiaopeng
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2017/02/25
Blue-noise Sampling
Push-pull
Surface Sampling
Remeshing
Stippling
Boron Doped ZIF-67@Graphene Derived Carbon Electrocatalyst for Highly Efficient Enzyme-Free Hydrogen Peroxide Biosensor
期刊论文
ADVANCED MATERIALS TECHNOLOGIES, 2017, 卷号: 2, 期号: 12, 页码: 1700224
作者:
Li, Zehui
;
Wang, Wenbo
;
Cao, Hongbin
;
Zhang, Qiang
;
Zhou, Xinyuan
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2018/01/19
Biosensors
Electrocatalysts
Graphene
Hydrogen Peroxide
Zeolitic Imidazolate Frameworks
Benzo[c][1,2,5] thiadiazole derivatives: A new class of potent Src homology-2 domain containing protein tyrosine phosphatase-2 (SHP2) inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 27, 期号: 23, 页码: 5154-5157
作者:
Wang, Wen-Long
;
Chen, Xiao-Yu
;
Gao, Ya
;
Gao, Li-Xin
;
Sheng, Li
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2019/01/08
Benzo[c][1,2,5] thiadiazole derivatives
PTP1B
SHP2
Inhibitors
Structure-activity relationships (SAR)
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