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上海药物研究所 [18]
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期刊论文 [18]
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2021 [1]
2020 [2]
2014 [1]
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Synthesis of 5-Phenyl-1,3,4-thiadiazole Derivatives and Their Biochemical Evaluation against Src Homology 2 Domain-Containing Protein Tyrosine Phosphatase 1 (SHP1)
期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 41, 期号: 8, 页码: 3097-3105
作者:
Yu Lijie
;
Feng Bo
;
Wang Zhijia
;
Gao Lixin
;
Zhang Chun
收藏
  |  
浏览/下载:187/0
  |  
提交时间:2021/11/04
5-phenyl-1,3,4-thiadiazole derivatives
Src homology 2 domain-containing protein tyrosine phosphatase 1 (SHP1)
inhibitors
structure-activity relationships
Disrupting phosphatase SHP2 in macrophages protects mice from high-fat diet-induced hepatic steatosis and insulin resistance by elevating IL-18 levels
期刊论文
JOURNAL OF BIOLOGICAL CHEMISTRY, 2020, 卷号: 295, 期号: 31, 页码: 10842-10856
作者:
Liu, Wen
;
Yin, Ye
;
Wang, Meijing
;
Fan, Ting
;
Zhu, Yuyu
收藏
  |  
浏览/下载:182/0
  |  
提交时间:2020/12/24
Src homology 2 domain containing tyrosine phosphatase-2 (SHP2)
hepatic steatosis
insulin resistance
caspase-1
interleukin 18 (IL-18)
fatty liver
metabolic disorder
inflammation
cytokine signaling
caspase 1 (CASP1)
tyrosine-protein phosphatase (tyrosine phosphatase)
macrophage
Synthesis, antifungal activity and potential mechanism of fusidic acid derivatives possessing amino-terminal groups
期刊论文
FUTURE MEDICINAL CHEMISTRY, 2020, 卷号: 12, 期号: 9, 页码: 763-774
作者:
Cao, Yucheng
;
Ni, Jingxuan
;
Ji, Wentao
;
Shang, Kangle
;
Liang, Kaicheng
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2020/12/24
antifungal activity
fusidic acid
homology modeling
molecular docking
molecular dynamics simulations
Design, synthesis, biological evaluation, and comparative docking study of 1,2,4-triazolones as CB1 receptor selective antagonists
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2014, 卷号: 74, 页码: 73-84
作者:
Han, Shuang
;
Zhang, Fei-Fei
;
Xie, Xin
;
Chen, Jian-Zhong
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/01/08
Cannabinoid receptors
Antagonist
1,2,4-Triazolone
Scaffold hopping
Homology model
Computational Models for Predicting Interactions with Membrane Transporters
期刊论文
CURRENT MEDICINAL CHEMISTRY, 2013, 卷号: 20, 期号: 16, 页码: 2118-2136
作者:
Xu, Y.
;
Shen, Q.
;
Liu, X.
;
Lu, J.
;
Li, S.
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08
Computational methods
homology modeling
membrane transporter
phamacophore models
QSAR models
supervised/unsupervised learning algorithms
Structural insights into the homology and differences between mouse protein tyrosine phosphatase-sigma and human protein tyrosine phosphatase-sigma
期刊论文
ACTA BIOCHIMICA ET BIOPHYSICA SINICA, 2011, 卷号: 43, 期号: 12, 页码: 977-988
作者:
Hou, Li
;
Wang, Jianchuan
;
Zhou, Yueyang
;
Li, Jingya
;
Zang, Yi
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2019/01/08
mouse PTP-sigma
crystallization
homology
difference
A novel class of antagonists for the FFAs receptor GPR40
期刊论文
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2009, 卷号: 390, 期号: 3, 页码: 557-563
作者:
Hu, Hui
;
He, Ling Yan
;
Gong, Zhen
;
Li, Ning
;
Lu, Yi Na
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/01/08
GPR40
Antagonist
Type 2 diabetes
Homology modeling
Virtual screening
Sulfonamide
Histidine kinase (YycG) protein of Streptococcus pneumoniae: Homology modeling and analysis
期刊论文
Chinese Journal of Biotechnology, 2009, 卷号: 25, 期号: 2, 页码: 207-214
作者:
Nan Li
;
Fei Wang
;
Wenchun Xu
;
Hong Wang
;
Xiaomin Luo
收藏
  |  
浏览/下载:20/0
  |  
提交时间:2019/01/08
Streptococcus pneumoniae
two-component system
histidine kinase
homology modeling
molecular docking
Probing ligand binding modes of human cytochrome P450 2J2 by homology modeling, molecular dynamics simulation, and flexible molecular docking
期刊论文
PROTEINS-STRUCTURE FUNCTION AND BIOINFORMATICS, 2008, 卷号: 71, 期号: 2, 页码: 938-949
作者:
Li, Weihua
;
Tang, Yun
;
Liu, Hong
;
Cheng, Jiagao
;
Zhu, Weiliang
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
cytochrome P450 2J2
homology modeling
molecular dynamics
molecular docking
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