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The discovery of novel and selective fatty acid binding protein 4 inhibitors by virtual screening and biological evaluation 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 18, 页码: 4310-4317
作者:  Song, Ming;  Xu, Yong;  Zhang, Yan;  Nie, Tao;  Zhou, Yang
收藏  |  浏览/下载:21/0  |  提交时间:2018/12/13
Design and synthesis of N-(4-aminopyridin-2-yl)amides as B-Raf(V600E) inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 12, 页码: 2760-2763
Li, Xiaokai; Shen, Jiayi; Tan, Li; Zhang, Zhang; Gao, Donglin; Luo, Jinfeng; Cheng, Huimin; Zhou, Xiaoping; Ma, Jie; Ding, Ke; Lu, Xiaoyun
收藏  |  浏览/下载:42/0  |  提交时间:2016/12/16
Design and synthesis of N-(4-aminopyridin-2-yl)amides as B-Raf(V600E) inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 12, 页码: 2760-2763
作者:  Lu, Xiaoyun;  Luo, Jinfeng;  Cheng, Huimin;  Zhou, Xiaoping;  Ma, Jie
收藏  |  浏览/下载:20/0  |  提交时间:2018/12/13
The discovery of novel and selective fatty acid binding protein 4 inhibitors by virtual screening and biological evaluation 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 18, 页码: 4310-4317
Zhou, Yang; Nie, Tao; Zhang, Yan; Song, Ming; Li, Kuai; Ding, Mengxiao; Ding, Ke; Wu, Donghai; Xu, Yong
收藏  |  浏览/下载:20/0  |  提交时间:2016/12/16
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M) 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 19, 页码: 4277-4281
Chan, Shingpan; Han, Kun; Qu, Rong; Tong, Linjiang; Li, Yingjun; Zhang, Zhang; Cheng, Huimin; Lu, Xiaoyun; Patterson, Adam; Smaill, Jeff; Ren, Xiaomei; Ding, Jian; Xie, Hua; Ding, Ke
收藏  |  浏览/下载:246/0  |  提交时间:2016/12/16
2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L858R/T790M) 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 19, 页码: 4277-4281
作者:  Smaill, Jeff;  Lu, Xiaoyun;  Cheng, Huimin;  Zhang, Zhang;  Li, Yingjun
收藏  |  浏览/下载:48/0  |  提交时间:2018/12/13
Evaluation of spiropiperidine hydantoins as a novel class of antimalarial agents 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2015, 卷号: 23, 期号: 16, 页码: 5144-5150
Meyers, Marvin J.; Anderson, Elizabeth J.; McNitt, Sarah A.; Krenning, Thomas M.; Singh, Megh; Xu, Jing; Zeng, Wentian; Qin, Limei; Xu, Wanwan; Zhao, Siting; Qin, Li; Eickhoff, Christopher S.; Oliva, Jonathan; Campbell, Mary A.; Arnett, Stacy D.; Prinsen, Michael J.; Griggs, David W.; Ruminski, Peter G.; Goldberg, Daniel E.; Ding, Ke; Liu, Xiaorong; Tu, Zhengchao; Tortorella, Micky D.; Sverdrup, Francis M.; Chen, Xiaoping
收藏  |  浏览/下载:54/0  |  提交时间:2016/12/16
Evaluation of spiropiperidine hydantoins as a novel class of antimalarial agents 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2015, 卷号: 23, 期号: 16, 页码: 5144-5150
作者:  Eickhoff, Christopher S.;  Meyers, Marvin J.;  Anderson, Elizabeth J.;  McNitt, Sarah A.;  Krenning, Thomas M.
收藏  |  浏览/下载:22/0  |  提交时间:2018/12/13
Synthesis, Skeletal Rearrangement, and Biological Activities of Spirooxindoles: Exploration of a Stepwise C-Piancatelli Rearrangement 期刊论文
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2014, 期号: 2, 页码: 338-349
作者:  Zheng, Wenxu;  Huang, Li;  Zhang, Xiaoyu;  Li, Jing;  Ding, Ke
收藏  |  浏览/下载:25/0  |  提交时间:2018/12/13
New benzimidazole-2-urea derivates as tubulin inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 17, 页码: 4250-4253
作者:  Cheng, Huimin;  Wang, Wenna;  Kong, Dexin;  Tan, Li;  Zhang, Zhang
收藏  |  浏览/下载:22/0  |  提交时间:2018/12/13


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