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科研机构
上海药物研究所 [55]
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期刊论文 [52]
会议论文 [3]
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2021 [3]
2020 [3]
2018 [4]
2017 [4]
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GPR84 signaling promotes intestinal mucosal inflammation via enhancing NLRP3 inflammasome activation in macrophages
期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:
Zhang, Qing
;
Chen, Lin-hai
;
Yang, Hui
;
Fang, You-chen
;
Wang, Si-wei
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2022/01/18
GPR84
medium chain fatty acid receptor
GPCR
inflammatory bowel diseases
ulcerative colitis
NLRP3 inflammasome
macrophages
Rapamycin recruits SIRT2 for FKBP12 deacetylation during mTOR activity modulation in innate immunity
期刊论文
ISCIENCE, 2021, 卷号: 24, 期号: 11, 页码: 22
作者:
Hu, Lin
;
Chen, Fuxian
;
Wu, Chao
;
Wang, Jun
;
Chen, Si-si
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2022/01/18
Smart Self-Assembly Amphiphilic Cyclopeptide-Dye for Near-Infrared Window-II Imaging
期刊论文
ADVANCED MATERIALS, 2021, 页码: 13
作者:
Chen, Hao
;
Shou, Kangquan
;
Chen, Si
;
Qu, Chunrong
;
Wang, Zhiming
收藏
  |  
浏览/下载:81/0
  |  
提交时间:2021/05/24
fluorescence‐
imaging‐
guided tumor surgery
NIR‐
II fluorescence imaging
pH‐
responsive materials
self‐
assembly
tumor imaging
Anti-PD-L1 mediating tumor-targeted codelivery of liposomal irinotecan/JQ1 for chemo-immunotherapy
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 8
作者:
He, Zhi-di
;
Zhang, Meng
;
Wang, Yong-hui
;
He, Yang
;
Wang, Hai-rui
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2021/05/24
tumor-targeted delivery
immunogenic cell death
PD-1
PD-L1 blockade
tumor immune microenvironment
irinotecan
JQ1
immune checkpoint
Crystallography-guided discovery of carbazole-based retinoic acid-related orphan receptor gamma-t (ROR gamma t) modulators: insights into different protein behaviors with "short" and "long" inverse agonists
期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 11
作者:
Yu, Ming-cheng
;
Yang, Feng
;
Ding, Xiao-yu
;
Sun, Nan-nan
;
Jiang, Zheng-yuan
收藏
  |  
浏览/下载:83/0
  |  
提交时间:2020/12/24
RORγ
t
cocrystal structures
MD simulation
“
short”
inverse agonists
agonists
“
long”
inverse agonists
Effects of Apatinib on the Pharmacokinetics of Nifedipine and Warfarin in Patients with Advanced Solid Tumors
期刊论文
DRUG DESIGN DEVELOPMENT AND THERAPY, 2020, 卷号: 14, 页码: 1963-1970
作者:
Zhu, Yun-Ting
;
Teng, Zan
;
Zhang, Yi-Fan
;
Li, Wei
;
Guo, Li-Xia
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2020/07/01
apatinib
drug-drug interaction
CYP3A4
CYP2C9
nifedipine
warfarin
The mTOR inhibitor AZD8055 overcomes tamoxifen resistance in breast cancer cells by down-regulating HSPB8
期刊论文
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 8, 页码: 1338-1346
作者:
Shi, Jia-jie
;
Chen, Si-meng
;
Guo, Chen-Liang
;
Li, Yi-xue
;
Ding, Jian
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2019/01/08
tamoxifen resistance
HSPB8
AZD8055
estrogen receptor
mTOR inhibitor
SIRT1 activator E1231 protects from experimental atherosclerosis and lowers plasma cholesterol and triglycerides by enhancing ABCA1 expression
期刊论文
Atherosclerosis, 2018, 卷号: 274, 页码: 172-181
作者:
Feng, Tingting
;
Liu, Peng
;
Wang, Xiao
;
Luo, Jinque
;
Zuo, Xuan
收藏
  |  
浏览/下载:38/0
  |  
提交时间:2019/01/08
Research of pollution-free and precision cultivation system of Chinese herbal medicines
期刊论文
Zhongguo Zhong yao za zhi = Zhongguo zhongyao zazhi = China journal of Chinese materia medica, 2018, 卷号: 43, 期号: 8, 页码: 1517-1528
作者:
Chen, Shi-Lin
;
Dong, Lin-Lin
;
Guo, Qiao-Sheng
;
Wei, Jian-He
;
Li, Xi-Wen
收藏
  |  
浏览/下载:52/0
  |  
提交时间:2019/01/08
Diketopyrrolopyrrole-based semiconducting polymer nanoparticles for in vivo second near-infrared window imaging and image-guided tumor surgery
期刊论文
CHEMICAL SCIENCE, 2018, 卷号: 9, 期号: 12, 页码: 3105-3110
作者:
Shou, Kangquan
;
Tang, Yufu
;
Chen, Hao
;
Chen, Si
;
Zhang, Lei
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2019/01/08
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