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Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5911-5916
Wang, Zhen; Bian, Huan; Bartual, Sergio G.; Du, Wenting; Luo, Jinfeng; Zhao, Hu; Zhang, Shasha; Mo, Cheng; Zhou, Yang; Xu, Yong; Tu, Zhengchao; Ren, Xiaomei; Lu, Xiaoyun; Brekken, Rolf A.; Yao, Libo; Bullock, Alex N.; Su, Jin; Ding, Ke
收藏  |  浏览/下载:50/0  |  提交时间:2016/12/16
Structure-Activity Relationship Study of Rakicidins: Overcoming Chronic Myeloid Leukemia Resistance to Imatinib with 4-Methylester-Rakicidin A 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 3, 页码: 1184-1196
作者:  Yang, Guang;  Zhang, Quan;  Chen, Yue;  Sang, Feng;  Ding, Yahui
收藏  |  浏览/下载:25/0  |  提交时间:2018/12/13
Structure-Based Design of Tetrahydroisoquinoline-7-carboxamides as Selective Discoidin Domain Receptor 1 (DDR1) Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 12, 页码: 5911-5916
作者:  Yao, Libo;  Ding, Ke;  Su, Jin;  Bullock, Alex N.;  Brekken, Rolf A.
收藏  |  浏览/下载:32/0  |  提交时间:2018/12/13
Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 4, 页码: 1565-1579
作者:  Tu, Zhengchao;  Zhou, Yulai;  Ding, Ke;  Xu, Yong;  Xue, Xiaoqian
收藏  |  浏览/下载:25/0  |  提交时间:2018/12/13
Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 4, 页码: 1565-1579
Xue, Xiaoqian; Zhang, Yan; Liu, Zhaoxuan; Song, Ming; Xing, Yanli; Xiang, Qiuping; Wang, Zhen; Tu, Zhengchao; Zhou, Yulai; Ding, Ke; Xu, Yong
收藏  |  浏览/下载:20/0  |  提交时间:2016/12/16
Structure-Activity Relationship Study of Rakicidins: Overcoming Chronic Myeloid Leukemia Resistance to Imatinib with 4-Methylester-Rakicidin A 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 3, 页码: 1184-1196
Sang, Feng; Ding, Yahui; Wang, Jinghan; Sun, Bingxia; Sun, Jianlei; Geng, Yan; Zhang, Zhang; Ding, Ke; Wu, Ling-Ling; Liu, Jian-Wei; Ba, Cuigai; Yang, Guang; Zhang, Quan; Li, Lu-Yuan; Chen, Yue
收藏  |  浏览/下载:46/0  |  提交时间:2016/12/16
Small-Molecule BET Inhibitors in Clinical and Preclinical Development and Their Therapeutic Potential 期刊论文
CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2015, 卷号: 15, 期号: 8, 页码: 776-794
Yu, Lei; Wang, Zhen; Zhang, Zhang; Ren, Xiaomei; Lu, Xiaoyun; Ding, Ke
收藏  |  浏览/下载:25/0  |  提交时间:2016/12/16
Design, Synthesis, and Biological Evaluation of Pyrazolo[1,5-a]pyridine-3-carboxamides as Novel Antitubercular Agents 期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 6, 期号: 7, 页码: 814-818
作者:  Ding, Ke;  Tang, Jian;  Wang, Bangxing;  Wu, Tian;  Wan, Junting
收藏  |  浏览/下载:29/0  |  提交时间:2018/12/13
Hybrid pyrimidine alkynyls inhibit the clinically resistance related Bcr-Abl(T315I) mutant 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 17, 页码: 3458-3463
作者:  Ding, Ke;  Pan, Xiaofeng;  Wang, Deping;  Zhuang, Xiaoxi;  Luo, Jingfeng
收藏  |  浏览/下载:22/0  |  提交时间:2018/12/13
Small-Molecule BET Inhibitors in Clinical and Preclinical Development and Their Therapeutic Potential 期刊论文
CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2015, 卷号: 15, 期号: 8, 页码: 776-794
作者:  Wang, Zhen;  Zhang, Zhang;  Ren, Xiaomei;  Lu, Xiaoyun;  Ding, Ke
收藏  |  浏览/下载:10/0  |  提交时间:2018/12/13


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