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期刊论文 [11]
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Bioassay-guided isolation of saikosaponins with agonistic activity on 5-hydroxytryptamine 2C receptor from Bupleurum chinense and their potential use for the treatment of obesity
期刊论文
CHINESE JOURNAL OF NATURAL MEDICINES, 2017, 卷号: 15, 期号: 6, 页码: 467-473
作者:
Sun Chang-Li
;
Geng Chang-An
;
Huang Xiao-Yan
;
Ma Yun-Bao
;
Zheng Xiao-Hong
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2017/10/23
Bupleurum Chinense
5-hydroxytryptamine 2c (5-ht2c) Receptor
Anti-obesity
Saikosaponins
Nitric oxide production inhibition and mechanism of phenanthrene analogs in lipopolysaccharide-stimulated RAW264.7 macrophages
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 卷号: 26, 期号: 10, 页码: 2521-2525
作者:
Yuan, XH (reprint author), Southwest Univ Sci & Technol, Sch Life Sci & Engn, Mianyang, Peoples R China.
;
Chen, LQ
;
Shen, XF
;
Hu, BY
;
Lin, Y
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  |  
浏览/下载:26/0
  |  
提交时间:2017/11/09
Phenanthrene
Anti-inflammatory Activity
P38
Ijba
Macrophage
Structure-Activity Relationship Study of Rakicidins: Overcoming Chronic Myeloid Leukemia Resistance to Imatinib with 4-Methylester-Rakicidin A
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 3, 页码: 1184-1196
作者:
Yang, Guang
;
Zhang, Quan
;
Chen, Yue
;
Sang, Feng
;
Ding, Yahui
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  |  
浏览/下载:25/0
  |  
提交时间:2018/12/13
Structure-Activity Relationship Study of Rakicidins: Overcoming Chronic Myeloid Leukemia Resistance to Imatinib with 4-Methylester-Rakicidin A
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 59, 期号: 3, 页码: 1184-1196
Sang, Feng
;
Ding, Yahui
;
Wang, Jinghan
;
Sun, Bingxia
;
Sun, Jianlei
;
Geng, Yan
;
Zhang, Zhang
;
Ding, Ke
;
Wu, Ling-Ling
;
Liu, Jian-Wei
;
Ba, Cuigai
;
Yang, Guang
;
Zhang, Quan
;
Li, Lu-Yuan
;
Chen, Yue
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浏览/下载:46/0
  |  
提交时间:2016/12/16
Ligand Efficiency Outperforms pIC(50) on Both 2D MLR and 3D CoMFA Models: A Case Study on AR Antagonists
期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2015, 卷号: 86, 期号: 6, 页码: 1501-1517
作者:
Li, JZ
;
Bai, F
;
Liu, HX
;
Gramatica, P
;
Li, JZ (reprint author), Lanzhou Univ, Sch Pharm, 199 West Donggang Rd, Lanzhou 730000, Peoples R China.
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浏览/下载:3/0
  |  
提交时间:2017/01/11
androgen receptor antagonist
comparative molecular field analysis
ligand efficiency
multiple linear regression
surface efficiency index
Lathyrol Diterpenes as Modulators of P-Glycoprotein Dependent Multidrug Resistance: Structure-Activity Relationship Studies on Euphorbia Factor L-3 Derivatives
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 58, 期号: 9, 页码: 3720-3738
作者:
Jiao, Wei
;
Wan, Zhongmin
;
Chen, Shuang
;
Lu, Runhua
;
Chen, Xiaozhen
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  |  
浏览/下载:45/0
  |  
提交时间:2016/12/22
MOUSE LYMPHOMA-CELLS
JATROPHANE DITERPENES
BREAST-CANCER
MACROCYCLIC DITERPENES
PROTEIN STRUCTURES
DRUG-BINDING
DISCOVERY
TRANSPORTERS
GENERATION
DATABASE
Noncovalent interactions between hydroxylated polycyclic aromatic hydrocarbon and DNA: Molecular docking and QSAR study
期刊论文
ENVIRONMENTAL TOXICOLOGY AND PHARMACOLOGY, 2011, 卷号: 32, 期号: 3, 页码: 373-381
作者:
Li, Fei
;
Li, Xuehua
;
Liu, Xiaoli
;
Zhang, Linbao
;
You, Liping
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  |  
浏览/下载:29/0
  |  
提交时间:2012/03/06
Hydroxylated Polycyclic Aromatic Hydrocarbon (Ho-pah)
Dna
Quantitative Structure-activity Relationship (Qsar)
Binding Interaction
Docking
Antioxidative and antitumor activity of derivatives of 4-beta-amino-4 '-demethylepipodophyllotoxin and their structure-activity relationship
期刊论文
PHARMAZIE, 2007, 卷号: 62, 期号: 6, 页码: 432-438
作者:
Zhang, XY
;
Li, WG
;
Wu, YJ
;
Tian, X
;
Zhang, XY (reprint author), Lanzhou Univ, Coll Basic Med Sci, Lanzhou 730000, Peoples R China.
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  |  
浏览/下载:4/0
  |  
提交时间:2015/12/22
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