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Distal mutation V486M disrupts the catalytic activity of DPP4 by affecting the flap of the propeller domain 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 9
作者:  Li, Teng-teng;  Peng, Cheng;  Wang, Ji-qiu;  Xu, Zhi-jian;  Su, Ming-bo
收藏  |  浏览/下载:42/0  |  提交时间:2022/01/18
Allosteric Modulators Enhancing GLP-1 Binding to GLP-1R via a Transmembrane Site 期刊论文
ACS CHEMICAL BIOLOGY, 2021, 卷号: 16, 期号: 11, 页码: 2444-2452
作者:  Wang, Jiang;  Yang, Dehua;  Cheng, Xi;  Yang, Linlin;  Wang, Zhaohui
收藏  |  浏览/下载:23/0  |  提交时间:2022/01/04
Constitutive signal bias mediated by the human GHRHR splice variant 1 期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2021, 卷号: 118, 期号: 40, 页码: 10
作者:  Cong, Zhaotong;  Zhou, Fulai;  Zhang, Chao;  Zou, Xinyu;  Zhang, Huibing
收藏  |  浏览/下载:24/0  |  提交时间:2021/12/01
Molecular insights into differentiated ligand recognition of the human parathyroid hormone receptor 2 期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2021, 卷号: 118, 期号: 32, 页码: 8
作者:  Wang, Xi;  Cheng, Xi;  Zhao, Lihua;  Wang, Yuzhe;  Ye, Chenyu
收藏  |  浏览/下载:24/0  |  提交时间:2021/11/04
Activation pathway of a G protein-coupled receptor uncovers conformational intermediates as targets for allosteric drug design 期刊论文
NATURE COMMUNICATIONS, 2021, 卷号: 12, 期号: 1, 页码: 15
作者:  Lu, Shaoyong;  He, Xinheng;  Yang, Zhao;  Chai, Zongtao;  Zhou, Shuhua
收藏  |  浏览/下载:35/0  |  提交时间:2021/11/04
Structures of the human dopamine D3 receptor-G(i) complexes 期刊论文
MOLECULAR CELL, 2021, 卷号: 81, 期号: 6, 页码: 1147-+
作者:  Xu, Peiyu;  Huang, Sijie;  Mao, Chunyou;  Krumm, Brian E.;  Zhou, X. Edward
收藏  |  浏览/下载:35/0  |  提交时间:2021/05/24
Discovery of 5-Benzylidene-2-phenyl-1,3-dioxane-4,6-diones as Highly Potent and Selective SIRT1 Inhibitors 期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2021, 卷号: 12, 期号: 3, 页码: 397-403
作者:  Li, Chunpu;  Hu, Sha-Sha;  Yang, Lisheng;  Wang, Min;  Long, Jian-Dong
收藏  |  浏览/下载:57/0  |  提交时间:2021/05/24
Structural insights into the human D1 and D2 dopamine receptor signaling complexes 期刊论文
CELL, 2021, 卷号: 184, 期号: 4, 页码: 931-+
作者:  Zhuang, Youwen;  Xu, Peiyu;  Mao, Chunyou;  Wang, Lei;  Krumm, Brian
收藏  |  浏览/下载:22/0  |  提交时间:2021/05/24
Structural basis for ligand recognition of the neuropeptide Y Y-2 receptor 期刊论文
NATURE COMMUNICATIONS, 2021, 卷号: 12, 期号: 1, 页码: 9
作者:  Tang, Tingting;  Hartig, Christin;  Chen, Qiuru;  Zhao, Wenli;  Kaiser, Anette
收藏  |  浏览/下载:40/0  |  提交时间:2021/05/24
Structural basis for activation of the growth hormone-releasing hormone receptor 期刊论文
NATURE COMMUNICATIONS, 2020, 卷号: 11, 期号: 1, 页码: 10
作者:  Zhou, Fulai;  Zhang, Huibing;  Cong, Zhaotong;  Zhao, Li-Hua;  Zhou, Qingtong
收藏  |  浏览/下载:22/0  |  提交时间:2020/12/21


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