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科研机构
北京大学 [18]
内容类型
期刊论文 [16]
其他 [2]
发表日期
2017 [1]
2016 [2]
2015 [2]
2014 [3]
2013 [1]
2012 [2]
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专题:北京大学
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Serum polyunsaturated fatty acid metabolites as useful tool for screening potential biomarker of colorectal cancer
期刊论文
PROSTAGLANDINS LEUKOTRIENES AND ESSENTIAL FATTY ACIDS, 2017
Zhang, Li-Jian
;
Chen, Bin
;
Zhang, Jun-jie
;
Li, Jian
;
Yang, Qingjing
;
Zhong, Qi-sheng
;
Zhan, Song
;
Liu, Huwei
;
Cai, Chun
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2017/12/03
Lipidomic
Colorectal cancer
Ultra-high performance liquid chromatography
Mass spectrometry
DRUG-INDUCED APOPTOSIS
CELL LUNG-CANCER
OXIDATIVE STRESS
PPAR-GAMMA
13-HYDROXYOCTADECADIENOIC ACID
PROSTAGLANDIN E-2
ARACHIDONIC-ACID
COLON
GROWTH
15-LIPOXYGENASE-1
Discovery of Novel 15-Lipoxygenase Activators To Shift the Human Arachidonic Acid Metabolic Network toward Inflammation Resolution
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016
Meng, Hu
;
McClendon, Christopher L.
;
Dai, Ziwei
;
Li, Kenan
;
Zhang, Xiaoling
;
He, Shan
;
Shang, Erchang
;
Liu, Ying
;
Lai, Luhua
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2017/12/03
INHIBITION
ENZYMES
MODEL
SITE
BIOSYNTHESIS
PROSTACYCLIN
PROTEINS
EFFECTOR
SYNTHASE
LIGANDS
Motions of Allosteric and Orthosteric Ligand-Binding Sites in Proteins are Highly Correlated
期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2016
Ma, Xiaomin
;
Meng, Hu
;
Lai, Luhua
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2017/12/04
MOLECULAR-DYNAMICS SIMULATIONS
CATABOLITE ACTIVATOR PROTEIN
TRANSCRIPTION ACTIVATION
CYTOCHROME-P450 3A4
SEQUENCE VARIATIONS
3C-LIKE PROTEINASE
RESIDUE POTENTIALS
FOLDED PROTEINS
DRUG DESIGN
DNA-BINDING
Antisense suppression of LOX3 gene expression in rice endosperm enhances seed longevity
期刊论文
PLANT BIOTECHNOLOGY JOURNAL, 2015
Xu, Huibin
;
Wei, Yidong
;
Zhu, Yongsheng
;
Lian, Ling
;
Xie, Hongguang
;
Cai, Qiuhua
;
Chen, Qiushi
;
Lin, Zhongping
;
Wang, Zonghua
;
Xie, Huaan
;
Zhang, Jianfu
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2017/12/03
seed longevity
rice
LOX3
artificial ageing
SITE-SPECIFIC RECOMBINATION
MASS-SPECTROMETRY
PRODUCT SPECIFICITY
TRANSGENIC PLANTS
SOYBEAN SEEDS
MARKER GENES
LIPOXYGENASE
PROTEOMICS
ITRAQ
TOOL
Diverse Ways of Perturbing the Human Arachidonic Acid Metabolic Network To Control Inflammation
期刊论文
ACCOUNTS OF CHEMICAL RESEARCH, 2015
Meng, Hu
;
Liu, Ying
;
Lai, Luhua
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2017/12/03
PROSTAGLANDIN E-2 SYNTHASE-1
TRADITIONAL CHINESE MEDICINE
LEUKOTRIENE A(4) HYDROLASE
DUAL INHIBITORS
DRUG DESIGN
LTA(4) HYDROLASE
5-LIPOXYGENASE
DISCOVERY
DERIVATIVES
CYCLOOXYGENASE-2
Identification of 1, 4-Dihydrothieno[3 ', 2 ':5, 6] thiopyrano [4, 3-c]pyrazole Derivatives as Human 5-Lipo-oxygenase Inhibitors
期刊论文
chemical biology drug design, 2014
Hu, Jianshu
;
Zhu, Wei
;
Meng, Hu
;
Liu, Ying
;
Wang, Xin
;
Hu, Chun
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2015/11/10
bioassay
cross-reactivity
human 5-lipo-oxygenase inhibitors
molecular docking
synthesis
LIPID MEDIATORS
5-LIPOXYGENASE
INFLAMMATION
LIGANDS
Benzo[d] isothiazole 1,1-dioxide derivatives as dual functional inhibitors of 5-lipoxygenase and microsomal prostaglandin E-2 synthase-1
期刊论文
生物有机化学与医药化学通讯, 2014
Shang, Erchang
;
Wu, Yiran
;
Liu, Pei
;
Liu, Ying
;
Zhu, Wei
;
Deng, Xiaobing
;
He, Chong
;
He, Shan
;
Li, Cong
;
Lai, Luhua
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2015/11/10
Benzo[d] isothiazole 1,1-dioxide
5-Lipoxygenase
Microsomal prostaglandin E-2 synthase
Dual functional inhibitor
ANTIINFLAMMATORY DRUGS
MPGES-1
BIOLOGY
TARGET
5-LOX
Development of 3,5-dinitrobenzoate-based 5-lipoxygenase inhibitors
期刊论文
生物有机化学与医药化学, 2014
Shang, Erchang
;
Liu, Ying
;
Wu, Yiran
;
Zhu, Wei
;
He, Chong
;
Lai, Luhua
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2015/11/10
3,5-Dinitrobenzoate
5-Lipoxygenase inhibitors
Cell-free assay
Human whole blood assay
SAR study
DISEASE
BIOSYNTHESIS
LEUKOTRIENES
INFLAMMATION
EICOSANOIDS
MECHANISMS
Optimization of 5-hydroxytryptamines as dual function inhibitors targeting phospholipase A(2) and leukotriene A(4) hydrolase
期刊论文
欧洲医药化学杂志, 2013
Meng, Hu
;
Liu, Ying
;
Zhai, Yujing
;
Lai, Luhua
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2015/11/10
5-Hydroxytryptamine
Optimization
PLA(2)
LTA(4)H
Dual function inhibitor
NMDA RECEPTOR ANTAGONIST
DRUG DISCOVERY
LOW-AFFINITY
5-LIPOXYGENASE
DERIVATIVES
POTENT
DESIGN
CYCLOOXYGENASE
SEROTONIN
BIOLOGY
Dynamic Modeling of Human 5-Lipoxygenase-Inhibitor Interactions Helps To Discover Novel Inhibitors
期刊论文
journal of medicinal chemistry, 2012
Wu, Yiran
;
He, Chong
;
Gao, Yang
;
He, Shan
;
Liu, Ying
;
Lai, Luhua
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2015/11/13
PROSTAGLANDIN E-2 SYNTHASE-1
HUMAN WHOLE-BLOOD
3-DIMENSIONAL STRUCTURES
THERAPEUTIC TARGET
POTENT INHIBITORS
DUAL INHIBITORS
CYCLOOXYGENASE
BIOSYNTHESIS
INFLAMMATION
LICOFELONE
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