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Acid-activatible micelleplex delivering siRNA-PD-L1 for improved cancer immunotherapy of CDK4/6 inhibition 期刊论文
CHINESE CHEMICAL LETTERS, 2021, 卷号: 32, 期号: 6, 页码: 1929-1936
作者:  Gao, Jing;  Zhang, Hanwu;  Zhou, Fengqi;  Hou, Bo;  Chen, Meiwan
收藏  |  浏览/下载:17/0  |  提交时间:2021/08/17
Design, synthesis, and biological evaluation of 4-benzoylamino-1H-pyrazole-3-carboxamide derivatives as potent CDK2 inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 215, 页码: 12
作者:  Lin, Tingting;  Li, Jiacheng;  Liu, Liping;  Li, Yuanqing;  Jiang, Hualiang
收藏  |  浏览/下载:70/0  |  提交时间:2021/05/24
Cyclin-dependent kinase inhibitor roscovitine attenuates liver inflammation and fibrosis by influencing initiating steps of liver injury 期刊论文
CLINICAL SCIENCE, 2021, 卷号: 135, 期号: 7, 页码: 925-941
作者:  Liu, Yanjun;  Li, Jiacheng;  Liao, Liping;  Huang, Heming;  Fan, Shijie
收藏  |  浏览/下载:18/0  |  提交时间:2021/08/17
Multiple functions of p21 in cancer radiotherapy 期刊论文
JOURNAL OF CANCER RESEARCH AND CLINICAL ONCOLOGY, 2021, 卷号: 147, 期号: 4, 页码: -
作者:  Kuang, Yanbei;  Kang, Jian;  Li, Hongbin;  Liu, Bingtao;  Zhao, Xueshan
收藏  |  浏览/下载:9/0  |  提交时间:2021/03/12
EZH2 inhibitors abrogate upregulation of trimethylation of H3K27 by CDK9 inhibitors and potentiate its activity against diffuse large B-cell lymphoma 期刊论文
HAEMATOLOGICA, 2020, 卷号: 105, 期号: 4, 页码: 1021-1031
作者:  Xie, Shao;  Wei, Fan;  Sun, Yi-ming;  Gao, Ying-lei;  Pan, Lu-lu
收藏  |  浏览/下载:38/0  |  提交时间:2020/07/01
Fisetin decreases TET1 activity and CCNY/CDK16 promoter 5hmC levels to inhibit the proliferation and invasion of renal cancer stem cell 期刊论文
JOURNAL OF CELLULAR AND MOLECULAR MEDICINE, 2019, 卷号: 23, 期号: 2
作者:  Si, Yibing;  Liu, Junfeng;  Shen, Hongliang;  Zhang, Chen;  Wu, Yuanhao
收藏  |  浏览/下载:25/0  |  提交时间:2019/12/05
Identification of a cellularly active SIRT6 allosteric activator 期刊论文
NATURE CHEMICAL BIOLOGY, 2018, 卷号: 14, 期号: 12, 页码: 1118-+
作者:  Huang, Zhimin;  Zhao, Junxing;  Deng, Wei;  Chen, Yingyi;  Shang, Jialin
收藏  |  浏览/下载:88/0  |  提交时间:2019/01/08
Discovery of 4-(((4-(5-chloro-2-(((1s,4s)-4-((2-methoxyethyl)amino) cyclohexyl)amino)pyridin-4-yl)thiazol-2-yl)amino)methyl) tetrahydro-2H-pyran-4-carbonitrile (JSH-150) as a novel highly selective and potent CDK9 kinase inhibitor 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 158, 页码: 896-916
作者:  Wang, Beilei;  Wu, Jiaxin;  Wu, Yun;  Chen, Cheng;  Zou, Fengming
收藏  |  浏览/下载:65/0  |  提交时间:2019/12/25
Design, synthesis, and molecular docking study of 3H-imidazole[4,5-c]pyridine derivatives as CDK2 inhibitors 期刊论文
ARCHIV DER PHARMAZIE, 2018, 卷号: 351, 期号: 6
作者:  Wu, Yi-Zhe;  Ying, Hua-Zhou;  Xu, Lei;  Cheng, Gang;  Chen, Jing
收藏  |  浏览/下载:31/0  |  提交时间:2019/01/08
Selective and novel cyclin-dependent kinases 4 inhibitor: synthesis and biological evaluation 期刊论文
Medicinal Chemistry Research, 2018, 卷号: Vol.27 No.6, 页码: 1666-1678
作者:  Qingxiang Guo;  Yongtao Li;  Chao Zhang;  Zhi Huang;  Xin Wang
收藏  |  浏览/下载:7/0  |  提交时间:2019/02/25


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