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科研机构
上海药物研究所 [26]
内容类型
期刊论文 [26]
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2021 [9]
2020 [3]
2019 [2]
2018 [3]
2017 [4]
2015 [3]
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LS-106, a novel EGFR inhibitor targeting C797S, exhibits antitumor activities both in vitro and in vivo
期刊论文
CANCER SCIENCE, 2021, 页码: 12
作者:
Liu, Yingqiang
;
Lai, Mengzhen
;
Li, Shan
;
Wang, Yanan
;
Feng, Fang
收藏
  |  
浏览/下载:62/0
  |  
提交时间:2022/01/18
C797S
epidermal growth factor receptor
fourth-generation EGFR TKI
non-small cell lung cancer
osimertinib resistance
Rapid nucleic acid detection of Escherichia coli O157:H7 based on CRISPR/ Cas12a system
期刊论文
FOOD CONTROL, 2021, 卷号: 130, 页码: 8
作者:
Wang, Shujuan
;
Fan, Yiling
;
Feng, Zhen
;
Song, Minghui
;
Li, Qiongqiong
收藏
  |  
浏览/下载:50/0
  |  
提交时间:2021/11/04
CRISPR/Cas12a
Fe3O4@PDA@UiO-66-NH2
Nucleic acid
Detection Escherichia coli O157:H7
Discovery of Potent and Selective CDK9 Degraders for Targeting Transcription Regulation in Triple-Negative Breast Cancer
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 64, 期号: 19, 页码: 14822-14847
作者:
Wei, Dan
;
Wang, Hanlin
;
Zeng, Qinghe
;
Wang, Wenjing
;
Hao, Bingbing
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  |  
浏览/下载:30/0
  |  
提交时间:2021/12/16
Supramolecular Antagonists Promote Mitochondrial Dysfunction
期刊论文
NANO LETTERS, 2021, 卷号: 21, 期号: 13, 页码: 5730-5737
作者:
Li, Mingming
;
Song, Yanqiu
;
Song, Na
;
Wu, Guangyao
;
Zhou, Hao
收藏
  |  
浏览/下载:87/0
  |  
提交时间:2021/08/17
Self-Assembly
Peptides
Drug Delivery
Mitochondrion-Targeting
Antagonists
Rh-Catalyzed cascade C-H activation/C-C cleavage/cyclization of carboxylic acids with cyclopropanols
期刊论文
CHEMICAL COMMUNICATIONS, 2021, 页码: 4
作者:
Wang, Siqi
;
Miao, Erfei
;
Wang, Hao
;
Song, Bichao
;
Huang, Wei
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  |  
浏览/下载:25/0
  |  
提交时间:2021/08/17
Natural product 1,2,3,4,6-penta-O-galloyl-beta-D-glucopyranose is a reversible inhibitor of glyceraldehyde 3-phosphate dehydrogenase
期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:
Li, Wen
;
Liao, Li-ping
;
Song, Ning
;
Liu, Yan-jun
;
Ding, Yi-luan
收藏
  |  
浏览/下载:82/0
  |  
提交时间:2021/06/11
glyceraldehyde 3-phosphate dehydrogenase
1,2,3,4,6-penta-O-galloyl-beta-D-glucopyranose
hydrogen deuterium exchange mass spectrometry
reversible inhibitor
glycolysis
Natural product 1,2,3,4,6-penta-O-galloyl-beta-D-glucopyranose is a reversible inhibitor of glyceraldehyde 3-phosphate dehydrogenase
期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 13
作者:
Li, Wen
;
Liao, Li-ping
;
Song, Ning
;
Liu, Yan-jun
;
Ding, Yi-luan
收藏
  |  
浏览/下载:81/0
  |  
提交时间:2021/06/11
glyceraldehyde 3-phosphate dehydrogenase
1,2,3,4,6-penta-O-galloyl-beta-D-glucopyranose
hydrogen deuterium exchange mass spectrometry
reversible inhibitor
glycolysis
Reply to: Binding site for MDL-801 on SIRT6
期刊论文
NATURE CHEMICAL BIOLOGY, 2021, 页码: 5
作者:
Huang, Zhimin
;
Zhao, Junxing
;
Deng, Wei
;
Chen, Yingyi
;
Shang, Jialin
收藏
  |  
浏览/下载:64/0
  |  
提交时间:2021/05/24
Marine furanocembranoids-inspired macrocycles enabled by Pd-catalyzed unactivated C(sp(3))-H olefination mediated by donor/donor carbenes
期刊论文
NATURE COMMUNICATIONS, 2021, 卷号: 12, 期号: 1, 页码: 11
作者:
Hao, Jiping
;
Guo, Xueying
;
He, Shijun
;
Xu, Zhongliang
;
Chen, Lu
收藏
  |  
浏览/下载:29/0
  |  
提交时间:2021/05/24
Engineering Polymeric Prodrug Nanoplatform for Vaccination Immunotherapy of Cancer
期刊论文
NANO LETTERS, 2020, 卷号: 20, 期号: 6, 页码: 4393-4402
作者:
Zhou, Lei
;
Hou, Bo
;
Wang, Dangge
;
Sun, Fang
;
Song, Rundi
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2020/12/24
Polymeric prodrug
Neoantigen
Adaptive immune response
Personalized immunotherapy
Nanoparticles
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