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科研机构
上海药物研究所 [17]
内容类型
期刊论文 [17]
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2021 [3]
2020 [3]
2019 [2]
2017 [5]
2016 [1]
2013 [2]
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Theoretical study and application of 2-phenyl-1,3,4-thiadiazole derivatives with optical and inhibitory activity against SHP1
期刊论文
PHYSICAL CHEMISTRY CHEMICAL PHYSICS, 2021, 页码: 14
作者:
Zhang, Chun
;
Sun, Yi-Tao
;
Gao, Li-Xin
;
Feng, Bo
;
Yan, Xue
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2022/01/18
Molecular recognition of an acyl-peptide hormone and activation of ghrelin receptor
期刊论文
NATURE COMMUNICATIONS, 2021, 卷号: 12, 期号: 1, 页码: 9
作者:
Wang, Yue
;
Guo, Shimeng
;
Zhuang, Youwen
;
Yun, Ying
;
Xu, Peiyu
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2021/11/04
A 36-week multicenter, randomized, double-blind, placebo-controlled, parallel-group, phase 3 clinical trial of sodium oligomannate for mild-to-moderate Alzheimer’s dementia
期刊论文
Alzheimer's Research & Therapy, 2021, 卷号: 13, 期号: 1
作者:
Xiao,Shifu
;
Chan,Piu
;
Wang,Tao
;
Hong,Zhen
;
Wang,Shuzhen
收藏
  |  
浏览/下载:151/0
  |  
提交时间:2021/05/24
Sodium oligomannate
Efficacy
Safety
Alzheimer’s disease
Clinical trial
Identify potent SARS-CoV-2 main protease inhibitors via accelerated free energy perturbation-based virtual screening of existing drugs
期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2020, 卷号: 117, 期号: 44, 页码: 27381-27387
作者:
Li, Zhe
;
Li, Xin
;
Huang, Yi-You
;
Wu, Yaoxing
;
Liu, Runduo
收藏
  |  
浏览/下载:75/0
  |  
提交时间:2020/12/24
virtual screening
SARS-CoV-2
drug repurposing
free energy perturbation
main protease
Structural basis of GPBAR activation and bile acid recognition
期刊论文
NATURE, 2020, 页码: 29
作者:
Yang, Fan
;
Mao, Chunyou
;
Guo, Lulu
;
Lin, Jingyu
;
Ming, Qianqian
收藏
  |  
浏览/下载:46/0
  |  
提交时间:2020/12/24
Microenvironment-Responsive Small-Molecule Probe for Pulmonary Fibrosis Detection
期刊论文
ANALYTICAL CHEMISTRY, 2020, 卷号: 92, 期号: 1, 页码: 699-706
作者:
Dong, Ying
;
Li, Xiao-Rong
;
Chen, Qi
;
Guo, Rui-Ying
;
Tang, Bi-Xi
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2020/07/01
Chain-Length- and Saturation-Tuned Mechanics of Fluid Nanovesicles Direct Tumor Delivery
期刊论文
ACS NANO, 2019, 卷号: 13, 期号: 7, 页码: 7676-7689
作者:
Dai, Zhuo
;
Yu, Miaorong
;
Yi, Xin
;
Wu, Zeming
;
Tian, Falin
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2020/07/01
SUVs
liposome
chain length and saturation
membrane mechanics
vesicle rigidity
ECM penetration
tumor delivery
Temperature- and rigidity-mediated rapid transport of lipid nanovesicles in hydrogels
期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2019, 卷号: 116, 期号: 12, 页码: 5362-5369
作者:
Yu, Miaorong
;
Song, Wenyi
;
Tian, Falin
;
Dai, Zhuo
;
Zhu, Quanlei
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2020/07/01
lipid nanovesicle
liposome
phase transition temperature
diffusion
biological hydrogels
LX2343 alleviates cognitive impairments in AD model rats by inhibiting oxidative stress-induced neuronal apoptosis and tauopathy
期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 8, 页码: 1104-1119
作者:
Guo, Xiao-dan
;
Sun, Guang-long
;
Zhou, Ting-ting
;
Wang, Yi-yang
;
Xu, Xin
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2019/01/08
Alzheimer's disease
LX2343
cognitive deficits
oxidative stress
tauopathy
mitochondria
GSK-3 beta inhibitor
neuroprotection
ICV-STZ rats
Marine-derived chromopeptide A, a novel class I HDAC inhibitor, suppresses human prostate cancer cell proliferation and migration
期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 4, 页码: 551-560
作者:
Sun, Jing-ya
;
Wang, Ji-dong
;
Wang, Xin
;
Liu, Hong-chun
;
Zhang, Min-min
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2019/01/08
HDAC
chromopeptide A
FK228
human prostate cancer
cell cycle arrest
apoptosis
cancer cell migration
PC3 xenograft model
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