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科研机构
复旦大学上海医学院 [20]
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期刊论文 [20]
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2018 [1]
2017 [3]
2016 [1]
2015 [2]
2014 [2]
2013 [2]
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专题:复旦大学上海医学院
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Discovery and anti-inflammatory evaluation of benzothiazepinones (BTZs) as novel non-ATP competitive inhibitors of glycogen synthase kinase-3 beta (GSK-3 beta)
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2018, 卷号: 26, 期号: 20
作者:
Gao, Yang
;
Zhang, Peng
;
Cui, Anfeng
;
Ye, De-Yong
;
Xiang, Meng
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2019/12/05
Glycogen synthase kinase 3 beta
Sirtuin 1
Non-ATP competitive inhibitors
Benzothiazepinones
Inflammation
Augmented O-GlcNAc, signaling via glucosamine attenuates oxidative stress and apoptosis, following contrast-induced acute kidney injury in rats
期刊论文
FREE RADICAL BIOLOGY AND MEDICINE, 2017, 卷号: 103
作者:
Hu, Jiachang
;
Chen, Rongyi
;
Jia, Ping
;
Fang, Yi
;
Liu, Tongqiang
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2019/12/05
Acute kidney injury
Iodinated contrast media
Hexosamine biosynthetic pathway
Glycogen synthase kinase-3 beta
Intranasal BMP9 Ameliorates Alzheimer Disease-Like Pathology and Cognitive Deficits in APP/PS1 Transgenic Mice
期刊论文
FRONTIERS IN MOLECULAR NEUROSCIENCE, 2017, 卷号: 10
作者:
Wang, Zigao
;
Xiong, Lu
;
Wan, Wenbin
;
Duan, Lijie
;
Bai, Xiaojing
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2019/12/05
bone morphogenetic protein 9
Alzheimer's disease
amyloid beta
tau
neuroinflammation
low-density lipoprotein receptor-related protein 1
glycogen synthase kinase-3 beta
The discovery of novel benzothiazinones as highly selective non-ATP competitive glycogen synthase kinase 3 beta inhibitors for the treatment of ovarian cancer
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 135
作者:
Gao, Yang
;
Ye, De-Yong
;
Zhou, Wei-Cheng
;
Chu, Yong
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2019/12/05
Glycogen synthase kinase 3 beta
Non-ATP competitive inhibitors
Benzothiazinones
Ovarian cancer
Antiproliferative activities
HGF alleviates high glucose-induced injury in podocytes by GSK3 beta inhibition and autophagy restoration
期刊论文
BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR CELL RESEARCH, 2016, 卷号: 1863, 期号: 11
作者:
Zhang, Congying
;
Hou, Bo
;
Yu, Siying
;
Chen, Qi
;
Zhang, Nong
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/12/06
Hepatocyte growth factor
Autophagy
Podocyte
Glycogen synthase kinase 3 beta
High glucose
Sulforaphane attenuation of experimental diabetic nephropathy involves GSK-3 beta/Fyn/Nrf2 signaling pathway
期刊论文
JOURNAL OF NUTRITIONAL BIOCHEMISTRY, 2015, 卷号: 26, 期号: 6
作者:
Shang, Guoguo
;
Tang, Xinjun
;
Gao, Pan
;
Guo, Fanli
;
Liu, Hongpeng
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2019/12/13
Sulforaphane
Diabetic nephropathy
Mesangial cells
Glycogen synthase kinase 3 beta
Fyn
Nrf2
Limb ischemic preconditioning protects against contrast-induced acute kidney injury in rats via phosphorylation of GSK-3 beta
期刊论文
FREE RADICAL BIOLOGY AND MEDICINE, 2015, 卷号: 81
作者:
Liu, Tongqiang
;
Fang, Yi
;
Liu, Shaopeng
;
Yu, Xiaofang
;
Zhang, Hui
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2019/12/19
Limb ischemic preconditioning
Acute kidney injury
Iodinated contrast media
Glycogen synthase kinase-3 beta
Beneficial synergistic effects of microdose lithium with pyrroloquinoline quinone in an Alzheimer's disease mouse model
期刊论文
NEUROBIOLOGY OF AGING, 2014, 卷号: 35, 期号: 12
作者:
Zhao, Lei
;
Gong, Neng
;
Liu, Meng
;
Pan, Xiaoli
;
Sang, Shaoming
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/19
Lithium
Pyrroloquinoline quinone
Alzheimer's disease
Glycogen synthase kinase-3
beta-Amyloid-binding alcohol dehydrogenase
Novel benzothiazinones (BTOs) as allosteric modulator or substrate competitive inhibitor of glycogen synthase kinase 3 beta (GSK-3 beta) with cellular activity of promoting glucose uptake
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 24, 期号: 24
作者:
Zhang, Peng
;
Li, Shufen
;
Gao, Yang
;
Lu, Wenbo
;
Huang, Ke
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2019/12/19
GSK-3 beta
Substrate competitive
Allosteric
Benzothiazinones
Anti-diabetes
Design, synthesis and biological evaluation of benzothiazepinones (BTZs) as novel non-ATP competitive inhibitors of glycogen synthase kinase-3 beta (GSK-3 beta)
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 61
作者:
Zhang, Peng
;
Hu, Hai-Rong
;
Bian, Shi-Hui
;
Huang, Zhao-Hui
;
Chu, Yong
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2019/12/19
GSK-3 beta
Kinase inhibitor
Non-ATP competitive
Benzothiazepinones
Selectivity
Docking
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