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科研机构
上海药物研究所 [22]
内容类型
期刊论文 [21]
会议论文 [1]
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2016 [2]
2015 [4]
2014 [5]
2013 [2]
2012 [1]
2011 [3]
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Ru(II)-Catalyzed Direct C(sp(2))-H Activation/Selenylation of Arenes with Selenyl Chlorides
期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2016, 卷号: 81, 期号: 13, 页码: 5263-5269
作者:
Shu, Shiqi
;
Fan, Zhoulong
;
Yao, Qizheng
;
Zhang, Ao
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2019/01/08
Ligand-Promoted Pd(II)-Catalyzed Functionalization of Unactivated C(sp(3))-H Bond: Regio- and Stereoselective Synthesis of Arylated Rimantadine Derivatives
期刊论文
ACS CATALYSIS, 2016, 卷号: 6, 期号: 2, 页码: 769-774
作者:
Fan, Zhoulong
;
Shu, Shiqi
;
Ni, Jiabin
;
Yao, Qizheng
;
Zhang, Ao
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2019/01/08
C(sp(3))-H activation
adamantane
rimantadine
regioselectivity
stereoselectivity
Novel tetracyclic benzo[b]carbazolones as highly potent and orally bioavailable ALK inhibitors: Design, synthesis, and structure-activity relationship study
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 105, 页码: 39-56
作者:
Jiang, Xiaolong
;
Zhou, Ji
;
Ai, Jing
;
Song, Zilan
;
Peng, Xia
收藏
  |  
浏览/下载:61/0
  |  
提交时间:2019/01/08
Benzo[b]carbazolones
ALK inhibitors
Anti-cancer
Anti-resistance
Non-small-cell lung cancer
N-(1-Oxy-2-picolyl)oxalamic Acid as an Efficient Ligand for Copper-Catalyzed Amination of Aryl Iodides at Room Temperature
期刊论文
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2015, 期号: 19, 页码: 4153-4161
作者:
Wang, Yongbin
;
Ling, Jing
;
Zhang, Yu
;
Zhang, Ao
;
Yao, Qizheng
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/01/08
Synthetic methods
Ligand design
N
O ligands
Copper
Amination
Discovery and SAR study of c-Met kinase inhibitors bearing an 3-amino-benzo[d] isoxazole or 3-aminoindazole scaffold
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2015, 卷号: 23, 期号: 3, 页码: 564-578
作者:
Jiang, Xiaolong
;
Liu, Hongyan
;
Song, Zilan
;
Peng, Xia
;
Ji, Yinchun
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2019/01/08
c-Met kinase
Inhibitor
3-Amino-benzo[d]isoxazole
3-Aminoindazole
Non-small cell lung cancer
N-(1-Oxy-2-picolyl)oxalamic acids as a new type of O,O-ligands for the Cu-catalyzed N-arylation of azoles with aryl halides in water or organic solvent
期刊论文
ORGANIC & BIOMOLECULAR CHEMISTRY, 2015, 卷号: 13, 期号: 13, 页码: 4101-4114
作者:
Wang, Yongbin
;
Zhang, Yu
;
Yang, Beibei
;
Zhang, Ao
;
Yao, Qizheng
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2019/01/08
Rh-III-Catalysed Hydrazine-Directed C(sp(2))-H Amination of Phenidones with N-Alkyl-O-benzoyl-hydroxylamines
期刊论文
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2014, 期号: 33, 页码: 7481-7488
作者:
Xue, Yu
;
Fan, Zhoulong
;
Jiang, Xiaolong
;
Wu, Kui
;
Wang, Meining
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2019/01/08
C-H activation
Amination
Hydrazines
Hydroxylamines
Amines
Nitrogen heterocycles
Novel 2,4-Diarylanninopyrimidine Analogues (DAAPalogues) Showing Potent c-Met/ALK Multikinase Inhibitory Activities
期刊论文
ACS MEDICINAL CHEMISTRY LETTERS, 2014, 卷号: 5, 期号: 4, 页码: 304-308
作者:
Liu, Zhiqing
;
Ai, Jing
;
Peng, Xia
;
Song, Zilan
;
Wu, Kui
收藏
  |  
浏览/下载:55/0
  |  
提交时间:2019/01/08
C1-Substituted-N3-benzazepine
c-Met/ALK dual inhibitor
structure repurposing
2,4-diarylaminopyrimidine analogues
Rh(III)-Catalyzed Intermolecular C-H Amination of 1-Aryl-1H-pyrazol-5(4H)-ones with Alkylamines
期刊论文
ORGANIC LETTERS, 2014, 卷号: 16, 期号: 1, 页码: 42-45
作者:
Wu, Kui
;
Fan, Zhoulong
;
Xue, Yu
;
Yao, Qizheng
;
Zhang, Ao
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2019/01/08
(D,L)-10-Camphorsulfonic-Acid-Catalysed Synthesis of Diaryl-Fused 2,8-Dioxabicyclo[3.3.1]nonanes from 2-Hydroxychalcones and Naphthol Derivatives
期刊论文
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2014, 期号: 2, 页码: 418-425
作者:
Jiang, Xiaolong
;
Song, Zilan
;
Xu, Chang
;
Yao, Qizheng
;
Zhang, Ao
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2019/01/08
Oxygen heterocycles
Nitrogen heterocycles
Cyclization
Aromatic substitution
Fused-ring systems
Acid catalysis
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