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Discovery of Novel Allosteric Modulators Targeting an Extra-Helical Binding Site of GLP-1R Using Structure- and Ligand-Based Virtual Screening 期刊论文
BIOMOLECULES, 2021, 卷号: 11, 期号: 7, 页码: 14
作者:  Zhou, Qingtong;  Guo, Wanjing;  Dai, Antao;  Cai, Xiaoqing;  Vass, Marton
收藏  |  浏览/下载:41/0  |  提交时间:2021/08/17
Affinity Mass Spectrometry-Based Fragment Screening Identified a New Negative Allosteric Modulator of the Adenosine A(2A) Receptor Targeting the Sodium Ion Pocket 期刊论文
ACS CHEMICAL BIOLOGY, 2021, 卷号: 16, 期号: 6, 页码: 991-1002
作者:  Lu, Yan;  Liu, Hongyue;  Yang, Dehua;  Zhong, Li;  Xin, Ye
收藏  |  浏览/下载:25/0  |  提交时间:2021/08/17
G protein-coupled receptors: structure- and function-based drug discovery 期刊论文
SIGNAL TRANSDUCTION AND TARGETED THERAPY, 2021, 卷号: 6, 期号: 1, 页码: 27
作者:  Yang, Dehua;  Zhou, Qingtong;  Labroska, Viktorija;  Qin, Shanshan;  Darbalaei, Sanaz
收藏  |  浏览/下载:23/0  |  提交时间:2021/05/24
Targeted Proteomics Combined with Affinity Mass Spectrometry Analysis Reveals Antagonist E7 Acts As an Intracellular Covalent Ligand of Orphan Receptor GPR52 期刊论文
ACS CHEMICAL BIOLOGY, 2020, 卷号: 15, 期号: 12, 页码: 3275-3284
作者:  Ma, Mengna;  Guo, Shimeng;  Lin, Xi;  Li, Shanshan;  Wu, Yiran
收藏  |  浏览/下载:16/0  |  提交时间:2021/05/24
Accelerating the Throughput of Affinity Mass Spectrometry-Based Ligand Screening toward a G Protein-Coupled Receptor (vol 91, pg 8162, 2019) 期刊论文
ANALYTICAL CHEMISTRY, 2020, 卷号: 92, 期号: 6, 页码: 4689-4689
作者:  Lu, Yan;  Qin, Shanshan;  Zhang, Bingjie;  Dai, Antao;  Cai, Xiaoqing
收藏  |  浏览/下载:27/0  |  提交时间:2020/07/01
A Novel G Protein-Biased and Subtype-Selective Agonist for a G Protein-Coupled Receptor Discovered from Screening Herbal Extracts 期刊论文
ACS CENTRAL SCIENCE, 2020, 卷号: 6, 期号: 2, 页码: 213-225
作者:  Zhang, Bingjie;  Zhao, Simeng;  Yang, Dehua;  Wu, Yiran;  Xin, Ye
收藏  |  浏览/下载:36/0  |  提交时间:2020/07/01
Accelerating the Throughput of Affinity Mass Spectrometry-Based Ligand Screening toward a G Protein-Coupled Receptor 期刊论文
ANALYTICAL CHEMISTRY, 2019, 卷号: 91, 期号: 13, 页码: 8162-8169
作者:  Lu, Yan;  Qin, Shanshan;  Zhang, Bingjie;  Dai, Antao;  Cai, Xiaoqing
收藏  |  浏览/下载:12/0  |  提交时间:2020/07/01
Efficient ligand discovery from natural herbs by integrating virtual screening, affinity mass spectrometry and targeted metabolomics 期刊论文
ANALYST, 2019, 卷号: 144, 期号: 9, 页码: 2881-2890
作者:  Wang, Zhihua;  Liang, Hao;  Cao, Haijie;  Zhang, Bingjie;  Li, Jun
收藏  |  浏览/下载:31/0  |  提交时间:2020/07/01
Accelerating the Throughput of Affinity Mass Spectrometry-Based Ligand Screening toward a G Protein-Coupled Receptor 期刊论文
ANALYTICAL CHEMISTRY, 2019, 卷号: 91, 期号: 13
作者:  Lu, Yan;  Qin, Shanshan;  Zhang, Bingjie;  Dai, Antao;  Cai, Xiaoqing
收藏  |  浏览/下载:29/0  |  提交时间:2019/12/05
Crystal structure of the Frizzled 4 receptor in a ligand-free state 期刊论文
NATURE, 2018, 卷号: 560, 期号: 7720, 页码: 666-+
作者:  Yang, Shifan;  Wu, Yiran;  Xu, Ting-Hai;  de Waal, Parker W.;  He, Yuanzheng
收藏  |  浏览/下载:81/0  |  提交时间:2019/01/08


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