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S3I-201 derivative incorporating naphthoquinone unit as effective STAT3 inhibitors: Design, synthesis and anti-gastric cancer evaluation 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2022, 卷号: 71
作者:  Li, Haobin;  Cai, Maohua;  Cao, Fei;  Yu, Dehua;  Yang, Jing
收藏  |  浏览/下载:14/0  |  提交时间:2022/12/22
Inhibition of STAT3 Signaling Pathway by Terphenyllin Suppresses Growth and Metastasis of Gastric Cancer 期刊论文
FRONTIERS IN PHARMACOLOGY, 2022, 卷号: 13
作者:  Yu, Dehua;  Qi, Simin;  Guan, Xiaoqing;  Yu, Wenkai;  Yu, Xuefei
收藏  |  浏览/下载:15/0  |  提交时间:2022/12/23
Allosteric Modulators Enhancing GLP-1 Binding to GLP-1R via a Transmembrane Site 期刊论文
ACS CHEMICAL BIOLOGY, 2021, 卷号: 16, 期号: 11, 页码: 2444-2452
作者:  Wang, Jiang;  Yang, Dehua;  Cheng, Xi;  Yang, Linlin;  Wang, Zhaohui
收藏  |  浏览/下载:27/0  |  提交时间:2022/01/04
Constitutive signal bias mediated by the human GHRHR splice variant 1 期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2021, 卷号: 118, 期号: 40, 页码: 10
作者:  Cong, Zhaotong;  Zhou, Fulai;  Zhang, Chao;  Zou, Xinyu;  Zhang, Huibing
收藏  |  浏览/下载:26/0  |  提交时间:2021/12/01
Discovery of Novel Allosteric Modulators Targeting an Extra-Helical Binding Site of GLP-1R Using Structure- and Ligand-Based Virtual Screening 期刊论文
BIOMOLECULES, 2021, 卷号: 11, 期号: 7, 页码: 14
作者:  Zhou, Qingtong;  Guo, Wanjing;  Dai, Antao;  Cai, Xiaoqing;  Vass, Marton
收藏  |  浏览/下载:41/0  |  提交时间:2021/08/17
Structures of G(i)-bound metabotropic glutamate receptors mGlu2 and mGlu4 期刊论文
NATURE, 2021, 卷号: 594, 期号: 7864, 页码: 583-+
作者:  Lin, Shuling;  Han, Shuo;  Cai, Xiaoqing;  Tan, Qiuxiang;  Zhou, Kexiu
收藏  |  浏览/下载:37/0  |  提交时间:2021/11/16
Structures of Gi-bound metabotropic glutamate receptors mGlu2 and mGlu4 期刊论文
NATURE, 2021, 页码: 23
作者:  Lin, Shuling;  Han, Shuo;  Cai, Xiaoqing;  Tan, Qiuxiang;  Zhou, Kexiu
收藏  |  浏览/下载:25/0  |  提交时间:2021/08/17
A unique hormonal recognition feature of the human glucagon-like peptide-2 receptor 期刊论文
CELL RESEARCH, 2020, 页码: 11
作者:  Sun, Wen;  Chen, Li-Nan;  Zhou, Qingtong;  Zhao, Li-Hua;  Yang, Dehua
收藏  |  浏览/下载:86/0  |  提交时间:2020/12/24
Transcriptional and proteomic insights into the host response in fatal COVID-19 cases 期刊论文
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2020, 卷号: 117, 期号: 45, 页码: 28336-28343
作者:  Wu, Meng;  Chen, Yaobing;  Xia, Han;  Wang, Changli;  Tan, Chin Yee
收藏  |  浏览/下载:57/0  |  提交时间:2020/12/24
Structural basis for activation of the growth hormone-releasing hormone receptor 期刊论文
NATURE COMMUNICATIONS, 2020, 卷号: 11, 期号: 1, 页码: 10
作者:  Zhou, Fulai;  Zhang, Huibing;  Cong, Zhaotong;  Zhao, Li-Hua;  Zhou, Qingtong
收藏  |  浏览/下载:24/0  |  提交时间:2020/12/21


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