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Development of FABP4/5 inhibitors with potential therapeutic effect on type 2 Diabetes Mellitus 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 卷号: 224, 页码: 14
作者:  He, Yu-Long;  Chen, Meng-Ting;  Wang, Ting;  Zhang, Ming-Ming;  Li, Ying-Xia
收藏  |  浏览/下载:63/0  |  提交时间:2021/11/04
Combined treatment with FABP4 inhibitor ameliorates rosiglitazone-induced liver steatosis in obese diabetic db/db mice 期刊论文
BASIC & CLINICAL PHARMACOLOGY & TOXICOLOGY, 2021, 页码: 10
作者:  Chen, Meng-Ting;  Huang, Jun-Shang;  Gao, Ding-Ding;  Li, Ying-Xia;  Wang, He-Yao
收藏  |  浏览/下载:41/0  |  提交时间:2021/08/17
Insights into the molecular mechanism of positive cooperativity between partial agonist MK-8666 and full allosteric agonist AP8 of hGPR40 by Gaussian accelerated molecular dynamics (GaMD) simulations 期刊论文
COMPUTATIONAL AND STRUCTURAL BIOTECHNOLOGY JOURNAL, 2021, 卷号: 19, 页码: 3978-3989
作者:  An, Xiaoli;  Bai, Qifeng;  Bing, Zhitong;  Liu, Huanxiang;  Yao, Xiaojun
收藏  |  浏览/下载:12/0  |  提交时间:2021/12/08
Anti-inflammatory signaling through G protein-coupled receptors 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 8
作者:  Ge, Yun-jun;  Liao, Qi-wen;  Xu, Ye-chun;  Zhao, Qiang;  Wu, Bei-li
收藏  |  浏览/下载:26/0  |  提交时间:2020/12/21
CYC31, A Natural Bromophenol PTP1B Inhibitor, Activates Insulin Signaling and Improves Long Chain-Fatty Acid Oxidation in C2C12 Myotubes 期刊论文
MARINE DRUGS, 2020, 卷号: 18, 期号: 5, 页码: 13
作者:  Luo, Jiao;  Hou, Yufei;  Xie, Mengyue;  Ma, Wanli;  Shi, Dayong
收藏  |  浏览/下载:31/0  |  提交时间:2020/09/25
Exploration of Fragment Binding Poses Leading to Efficient Discovery of Highly Potent and Orally Effective Inhibitors of FABP4 for Anti-inflammation 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 8, 页码: 4090-4106
作者:  Su, Haixia;  Zou, Yi;  Chen, Guofeng;  Dou, Huixia;  Xie, Hang
收藏  |  浏览/下载:32/0  |  提交时间:2020/07/01
Exogenous FABP4 interferes with differentiation, promotes lipolysis and inflammation in adipocytes 期刊论文
ENDOCRINE, 2020, 卷号: 67, 期号: 3, 页码: 587-596
作者:  Dou, Hui-Xia;  Wang, Ting;  Su, Hai-Xia;  Gao, Ding-Ding;  Xu, Ye-Chun
收藏  |  浏览/下载:45/0  |  提交时间:2020/07/01
Identification of new dual FABP4/5 inhibitors based on a naphthalene-1-sulfonamide FABP4 inhibitor 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2019, 卷号: 27, 期号: 19, 页码: 16
作者:  He, Yulong;  Dou, Huixia;  Gao, Dingding;  Wang, Ting;  Zhang, Mingming
收藏  |  浏览/下载:17/0  |  提交时间:2020/07/01
From hit to lead: Structure-based discovery of naphthalene-1-sulfonamide derivatives as potent and selective inhibitors of fatty acid binding protein 4 (vol 154, pg 44, 2018) 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 170, 页码: 235-236
作者:  Gao, Ding-Ding;  Dou, Hui-Xia;  Su, Hai-Xia;  Zhang, Ming-Ming;  Wang, Ting
收藏  |  浏览/下载:9/0  |  提交时间:2020/07/01
FABP5 regulates the proliferation of clear cell renal cell carcinoma cells via the PI3K/AKT signaling pathway 期刊论文
INTERNATIONAL JOURNAL OF ONCOLOGY, 2019, 卷号: 54, 期号: 4
作者:  Le, Wei;  Ding, Qiang;  Wang, Peijun;  Ma, Chunhui;  Lv, Qi
收藏  |  浏览/下载:65/0  |  提交时间:2019/12/05


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