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Lead discovery, chemical optimization, and biological evaluation studies of novel histone methyltransferase SET7 small-molecule inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 9, 页码: 10
作者:  Hou, Zeng;  Min, Wenjian;  Zhang, Rukang;  Niu, Ao;  Li, Yuanqing
收藏  |  浏览/下载:43/0  |  提交时间:2020/07/01
Amelioration of Uremic Toxin Indoxyl Sulfate-Induced Osteoblastic Calcification by SET Domain Containing Lysine Methyltransferase 7/9 Protein 期刊论文
NEPHRON, 2019, 卷号: 141, 期号: 4
作者:  Hu, Jiachang;  Zhang, Xiaoyan;  Ding, Xiaoqiang;  Shi, Yiqin;  Chen, Jing
收藏  |  浏览/下载:27/0  |  提交时间:2019/12/05
Amelioration of Uremic Toxin Indoxyl Sulfate-Induced Osteoblastic Calcification by SET Domain Containing Lysine Methyltransferase 7/9 Protein. 期刊论文
Nephron, 2019, 页码: 1-8
作者:  Jing Chen;  Yulu Gu;  Han Zhang;  Yichun Ning;  Nana Song
收藏  |  浏览/下载:22/0  |  提交时间:2019/12/13
Resveratrol induces p53 in colorectal cancer through SET7/9 期刊论文
ONCOLOGY LETTERS, 2019, 卷号: 17, 期号: 4, 页码: 3783-3789
作者:  Liu, Zhonglun[1];  Wu, Xiaohong[2];  Lv, Jingjing[3];  Sun, Hui[4];  Zhou, Feiqin[5]
收藏  |  浏览/下载:21/0  |  提交时间:2019/12/24
Discovery and Optimization of Novel, Selective Histone Methyltransferase SET7 Inhibitors by Pharmacophore- and Docking-Based Virtual Screening 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 58, 期号: 20, 页码: 8166-8181
作者:  Meng, Fanwang;  Cheng, Sufang;  Ding, Hong;  Liu, Shien;  Liu, Yan
收藏  |  浏览/下载:30/0  |  提交时间:2019/01/08
Repression of hypoxia-inducible factor alpha signaling by Set7-mediated methylation 期刊论文
NUCLEIC ACIDS RESEARCH, 2015, 卷号: 43, 期号: 10, 页码: 5081-5098
作者:  Liu, Xing;  Chen, Zhu;  Xu, Chenxi;  Leng, Xiaoqian;  Cao, Hong
收藏  |  浏览/下载:39/0  |  提交时间:2015/09/15
Methylation of SUV39H1 by SET7/9 results in heterochromatin relaxation and genome instability 期刊论文
proceedings of the national academy of sciences of the united states of america, 2013
Wang, Donglai; Zhou, Jingyi; Liu, Xiangyu; Lu, Danyu; Shen, Changchun; Du, Yipeng; Wei, Fu-Zheng; Song, Boyan; Lu, Xiaopeng; Yu, Yu; Wang, Lina; Zhao, Ying; Wang, Haiying; Yang, Yang; Akiyama, Yoshimitsu; Zhang, Hongquan; Zhu, Wei-Guo
收藏  |  浏览/下载:3/0  |  提交时间:2015/11/11
Structure of human lysine methyltransferase Smyd2 reveals insights into the substrate divergence in Smyd proteins 期刊论文
JOURNAL OF MOLECULAR CELL BIOLOGY, 2011, 卷号: 3, 期号: 5, 页码: 293-300
作者:  Xu, ST;  Zhong, C;  Zhang, TL;  Ding, JP
收藏  |  浏览/下载:11/0  |  提交时间:2015/07/22


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