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期刊论文 [8]
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Lead discovery, chemical optimization, and biological evaluation studies of novel histone methyltransferase SET7 small-molecule inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 9, 页码: 10
作者:
Hou, Zeng
;
Min, Wenjian
;
Zhang, Rukang
;
Niu, Ao
;
Li, Yuanqing
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2020/07/01
Histone methylation
SET7
Small-molecule inhibitor
Virtual screening
Molecular probe
Amelioration of Uremic Toxin Indoxyl Sulfate-Induced Osteoblastic Calcification by SET Domain Containing Lysine Methyltransferase 7/9 Protein
期刊论文
NEPHRON, 2019, 卷号: 141, 期号: 4
作者:
Hu, Jiachang
;
Zhang, Xiaoyan
;
Ding, Xiaoqiang
;
Shi, Yiqin
;
Chen, Jing
收藏
  |  
浏览/下载:27/0
  |  
提交时间:2019/12/05
Chronic kidney disease
Vascular calcification
SET domain containing lysine methyltransferase 7/9
Indoxyl sulfate
Amelioration of Uremic Toxin Indoxyl Sulfate-Induced Osteoblastic Calcification by SET Domain Containing Lysine Methyltransferase 7/9 Protein.
期刊论文
Nephron, 2019, 页码: 1-8
作者:
Jing Chen
;
Yulu Gu
;
Han Zhang
;
Yichun Ning
;
Nana Song
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2019/12/13
Chronic
kidney
disease
Indoxyl
sulfate
SET
domain
containing
lysine
methyltransferase
7/9
Vascular
calcification
Resveratrol induces p53 in colorectal cancer through SET7/9
期刊论文
ONCOLOGY LETTERS, 2019, 卷号: 17, 期号: 4, 页码: 3783-3789
作者:
Liu, Zhonglun[1]
;
Wu, Xiaohong[2]
;
Lv, Jingjing[3]
;
Sun, Hui[4]
;
Zhou, Feiqin[5]
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2019/12/24
resveratrol
colorectal cancer
tumour protein p53
SET domain containing lysine methyltransferase 7/9
apoptosis
Discovery and Optimization of Novel, Selective Histone Methyltransferase SET7 Inhibitors by Pharmacophore- and Docking-Based Virtual Screening
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2015, 卷号: 58, 期号: 20, 页码: 8166-8181
作者:
Meng, Fanwang
;
Cheng, Sufang
;
Ding, Hong
;
Liu, Shien
;
Liu, Yan
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2019/01/08
Repression of hypoxia-inducible factor alpha signaling by Set7-mediated methylation
期刊论文
NUCLEIC ACIDS RESEARCH, 2015, 卷号: 43, 期号: 10, 页码: 5081-5098
作者:
Liu, Xing
;
Chen, Zhu
;
Xu, Chenxi
;
Leng, Xiaoqian
;
Cao, Hong
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  |  
浏览/下载:39/0
  |  
提交时间:2015/09/15
Methylation of SUV39H1 by SET7/9 results in heterochromatin relaxation and genome instability
期刊论文
proceedings of the national academy of sciences of the united states of america, 2013
Wang, Donglai
;
Zhou, Jingyi
;
Liu, Xiangyu
;
Lu, Danyu
;
Shen, Changchun
;
Du, Yipeng
;
Wei, Fu-Zheng
;
Song, Boyan
;
Lu, Xiaopeng
;
Yu, Yu
;
Wang, Lina
;
Zhao, Ying
;
Wang, Haiying
;
Yang, Yang
;
Akiyama, Yoshimitsu
;
Zhang, Hongquan
;
Zhu, Wei-Guo
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  |  
浏览/下载:3/0
  |  
提交时间:2015/11/11
histone methylation
nonhistone posttranslational modifications
DNA-DAMAGE RESPONSE
HISTONE H3 METHYLATION
LYSINE METHYLATION
TRANSFERASE SUV39H1
TUMOR SUPPRESSION
P53 ACTIVITY
METHYLTRANSFERASE
CHROMATIN
SIRT1
HP1
Structure of human lysine methyltransferase Smyd2 reveals insights into the substrate divergence in Smyd proteins
期刊论文
JOURNAL OF MOLECULAR CELL BIOLOGY, 2011, 卷号: 3, 期号: 5, 页码: 293-300
作者:
Xu, ST
;
Zhong, C
;
Zhang, TL
;
Ding, JP
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2015/07/22
Smyd2
Smyd proteins
SET family
histone lysine methyltransferase
epigenetics
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