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Synthesis and Target Identification of Benzoxepane Derivatives as Potential Anti-Neuroinflammatory Agents for Ischemic Stroke
期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2020, 卷号: 59, 期号: 6, 页码: 2429-2439
作者:
Gao, Cheng-Long
;
Hou, Gui-Ge
;
Liu, Jin
;
Ru, Tong
;
Xu, Ya-Zhou
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2020/07/01
anti-inflammatory
drug discovery
heterocycles
photoaffinity labeling
proteins
Colocalization Strategy Unveils an Underside Binding Site in the Transmembrane Domain of Smoothened Receptor
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 21, 页码: 9983-9989
作者:
Zhou, Fang
;
Ding, Kang
;
Zhou, Yiqing
;
Liu, Yang
;
Liu, Xiaoyan
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  |  
浏览/下载:27/0
  |  
提交时间:2020/07/01
Combinatorial Peptide Ligand Library-Based Photoaffinity Probe for the Identification of Phosphotyrosine-Binding Domain Proteins
期刊论文
ANALYTICAL CHEMISTRY, 2019, 卷号: 91, 期号: 5, 页码: 3221-3226
作者:
Zhang, Kai
;
An, Jinying
;
Zhai, Guijin
;
Guo, Zhenchang
;
Bai, Xue
收藏
  |  
浏览/下载:55/0
  |  
提交时间:2019/06/20
Combinatorial peptide ligand library-based photoaffinity probe for the identification of phosphotyrosine-binding domain proteins
期刊论文
Analytical chemistry, 2019, 卷号: 91, 期号: 5, 页码: 3221-3226
作者:
An, Jinying
;
Zhai, Guijin
;
Guo, Zhenchang
;
Bai, Xue
;
Chen, Pu
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  |  
浏览/下载:69/0
  |  
提交时间:2019/05/08
An Efficient Approach for Selective Enrichment of Histone Modification Readers Using Self-Assembled Multivalent Photoaffinity Peptide Probes
期刊论文
ANALYTICAL CHEMISTRY, 2018, 卷号: 90, 期号: 19, 页码: 11385-11392
作者:
Zhang, Kai
;
Zhai, Guijin
;
Dong, Hanyang
;
Guo, Zhenchang
;
Feng, Wei
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  |  
浏览/下载:49/0
  |  
提交时间:2019/06/20
A diubiquitin-based photoaffinity probe for profiling K27-linkage targeting deubiquitinases
期刊论文
CHEMICAL COMMUNICATIONS, 2017, 卷号: 53, 期号: 73, 页码: 10208-10211
作者:
Tan, Xiao-Dan
;
Pan, Man
;
Gao, Shuai
;
Zheng, Yong
;
Shi, Jing
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  |  
浏览/下载:18/0
  |  
提交时间:2018/08/16
Exploring the Binding Proteins of Glycolipids with Bifunctional Chemical Probes
期刊论文
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2016
Liu, Xiaohui
;
Dong, Ting
;
Zhou, Yu
;
Huang, Niu
;
Lei, Xiaoguang
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  |  
浏览/下载:3/0
  |  
提交时间:2017/12/03
click chemistry
glycolipids
minimalist linker
photoaffinity labeling
target identification
LIPID-A ANALOGS
SIGNAL-TRANSDUCTION
IN-VITRO
ENDOTOXIN ANTAGONIST
TLR4-MD-2 COMPLEX
RECEPTOR 4
LIPOPOLYSACCHARIDE
CELL
SPHINGOLIPIDS
RECOGNITION
Affinity purification in target identification: the specificity challenge
期刊论文
archives of pharmacal research, 2015, 卷号: 38, 期号: 9, 页码: 1661-1685
作者:
Zheng, Wenlu
;
Li, Gang
;
Li, Xiaoyu
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  |  
浏览/下载:133/0
  |  
提交时间:2015/11/17
Target identification
Affinity purification
Small molecule
Phenotypic screening
Protein-ligand interaction
Specificity
Affinity purification in target identification: the specificity challenge
期刊论文
ARCHIVES OF PHARMACAL RESEARCH, 2015
Zheng, Wenlu
;
Li, Gang
;
Li, Xiaoyu
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2017/12/03
Target identification
Affinity purification
Small molecule
Phenotypic screening
Protein-ligand interaction
Specificity
PROTEIN-LIGAND INTERACTIONS
SMALL-MOLECULE PROBES
PHOTOAFFINITY CROSS-LINKING
BIOACTIVE SMALL MOLECULES
QUANTITATIVE CHEMICAL PROTEOMICS
HISTONE DEACETYLASE COMPLEXES
CARBOHYDRATE-BINDING PROTEINS
DIRECTED TOSYL CHEMISTRY
TAGGED TRIAZINE LIBRARY
A1 ADENOSINE RECEPTOR
Photoaffinity labeling of transcription factors by DNA-templated crosslinking
期刊论文
chemical science, 2015
Liu, Ying
;
Zheng, Wenlu
;
Zhang, Wan
;
Chen, Nan
;
Liu, Yang
;
Chen, Li
;
Zhou, Xiaozhou
;
Chen, Xingshuo
;
Zheng, Haifeng
;
Li, Xiaoyu
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2015/11/10
NF-KAPPA-B
ENCODED CHEMICAL LIBRARIES
PROTEIN-DNA
BINDING-PROTEINS
GENE-EXPRESSION
GEL-ELECTROPHORESIS
PHOTOCROSS-LINKING
COMPLEX REVEALS
ASSAY
AFFINITY
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