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上海药物研究所 [6]
复旦大学上海医学院 [2]
南华大学 [1]
北京大学 [1]
昆明医科大学 [1]
湖南大学 [1]
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期刊论文 [12]
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Intestinal farnesoid X receptor signaling controls hepatic fatty acid oxidation
期刊论文
BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR AND CELL BIOLOGY OF LIPIDS, 2022, 卷号: 1867, 期号: 2, 页码: 13
作者:
Lu, Dasheng
;
Liu, Yameng
;
Luo, Yuhong
;
Zhao, Jie
;
Feng, Chao
收藏
  |  
浏览/下载:49/0
  |  
提交时间:2022/01/18
Fatty acid oxidation
Acylcarnitines
FXR
FGF15/19
PGC1 alpha
Transcriptomics
Metabolomics
Discovery of a Potential Liver Fibrosis Inhibitor from a Mushroom Endophytic Fungus by Genome Mining of a Silent Biosynthetic Gene Cluster
期刊论文
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2021, 卷号: 69, 期号: 38, 页码: 11303-11310
作者:
Cheng, Jin-Tao
;
Wang, Han-Min
;
Yu, Jia-Hui
;
Sun, Chen-Fan
;
Cao, Fei
收藏
  |  
浏览/下载:28/0
  |  
提交时间:2021/12/01
fungus
Calcarisporium arbuscula
natural product
gene cluster activation
liver fibrosis
Discovery of novel ketoxime ether derivatives with potent FXR agonistic activity, oral effectiveness and high liver/blood ratio
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 43, 页码: 13
作者:
Tang, Xuehang
;
Ning, Mengmeng
;
Ye, Yangliang
;
Gu, Yipei
;
Yan, Hongyi
收藏
  |  
浏览/下载:49/0
  |  
提交时间:2021/11/04
FXR agonist
Ketoxime ether
Target genes
Liver
blood ratio
Systemic activation
A new mechanism of obeticholic acid on NASH treatment by inhibiting NLRP3 inflammasome activation in macrophage
期刊论文
METABOLISM-CLINICAL AND EXPERIMENTAL, 2021, 卷号: 120, 页码: 12
作者:
Huang, Suling
;
Wu, Yanwei
;
Zhao, Zhuohui
;
Wu, Bing
;
Sun, Kai
收藏
  |  
浏览/下载:90/0
  |  
提交时间:2021/08/17
Macrophage
NLRP3 inflammasome
Hepatic lipid accumulation
NASH
FXR
Discovery and Optimization of Non-bile Acid FXR Agonists as Preclinical Candidates for the Treatment of Nonalcoholic Steatohepatitis
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 21, 页码: 12748-12772
作者:
Li, Junyou
;
Liu, Mengqi
;
Li, Yazhou
;
Sun, Dan-dan
;
Shu, Zhihao
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2021/05/24
A novel bile acid analog, A17, ameliorated non-alcoholic steatohepatitis in high-fat diet-fed hamsters
期刊论文
TOXICOLOGY AND APPLIED PHARMACOLOGY, 2020, 卷号: 404, 页码: 14
作者:
Wang, Ying
;
Zhu, Yao
;
Niu, Junxing
;
Deng, Qiangqiang
;
Guo, Shimeng
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  |  
浏览/下载:60/0
  |  
提交时间:2020/12/21
Bile acid analog
NASH
TGR5
Cd36
AMPK alpha
The protective effect and mechanism of the FXR agonist obeticholic acid via targeting gut microbiota in non-alcoholic fatty liver disease
期刊论文
DRUG DESIGN DEVELOPMENT AND THERAPY, 2019, 卷号: 13
作者:
Zhang, Dan-Ying
;
Zhu, Lin
;
Liu, Hai-Ning
;
Tseng, Yu-Jen
;
Weng, Shu-Qiang
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  |  
浏览/下载:25/0
  |  
提交时间:2019/12/05
non-alcoholic fatty liver disease
farnesoid X receptor
gastrointestinal microbiome
bile acid
metabolic diseases
FXR-Dependent Modulation of the Human Small Intestinal Microbiome by the Bile Acid Derivative Obeticholic Acid
期刊论文
Gastroenterology, 2018, 卷号: Vol.155 No.6, 页码: 1741-1752(e5)
作者:
Elliot S. Friedman
;
Yun Li
;
Ting-Chin David Shen
;
Jack Jiang
;
Lillian Chau
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2019/12/26
Nuclear
Hormone
Receptor
Genetics
Gene
Regulation
Metabolism
Mechanisms of MAFG Dysregulation in Cholestatic Liver Injury and Development of Liver Cancer
期刊论文
Gastroenterology, 2018, 卷号: 155, 期号: 2, 页码: 557-571.e14
作者:
Liu, Ting
;
Yang, Heping
;
Fan, Wei
;
Tu, Jian
;
Li, Tony W. H.
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/12/27
FXR
Obeticholic Acid
S-Adenosylmethionine
Ursodeoxycholic Acid
Chemoproteomic Profiling of Bile Acid Interacting Proteins
期刊论文
ACS CENTRAL SCIENCE, 2017
Zhuang, Shentian
;
Li, Qiang
;
Cai, Lirong
;
Wang, Chu
;
Lei, Xiaoguang
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2017/12/03
NONALCOHOLIC-FATTY-LIVER
FARNESOID-X-RECEPTOR
NUCLEAR RECEPTOR
TAUROURSODEOXYCHOLIC ACID
ALZHEIMERS-DISEASE
EMERGING ROLE
OBETICHOLIC ACID
BINDING-PROTEINS
VIBRIO-CHOLERAE
HOST METABOLISM
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